ZA200504339B - 2-(1H-indazol-6-ylamino)-benzamide compounds as protein kinases inhibitors useful for the treatment of ophtalmic diseases - Google Patents
2-(1H-indazol-6-ylamino)-benzamide compounds as protein kinases inhibitors useful for the treatment of ophtalmic diseases Download PDFInfo
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
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| US20060182783A1 (en) * | 2004-04-30 | 2006-08-17 | Allergan, Inc. | Sustained release intraocular drug delivery systems |
| WO2006043172A1 (en) * | 2004-10-19 | 2006-04-27 | Pfizer Inc. | Pharmaceutical compositions and methods for sub-tenon delivery |
| WO2006048745A1 (en) * | 2004-11-02 | 2006-05-11 | Pfizer Inc. | Methods for preparing indazole compounds |
| US20060160863A1 (en) * | 2005-01-05 | 2006-07-20 | Agouron Pharmaceuticals, Inc. | Polymorphic and amorphous forms of 2-{3-[(E)-2-(4,6-dimethyl-pyridin-2-yl)-vinyl]-1H-indazol-6-ylamino}-N-(4-hydroxy-but-2-ynyl)benzamide |
| WO2006117666A2 (en) * | 2005-04-29 | 2006-11-09 | Pfizer Inc. | Dosage forms, pharmaceutical compositions and methods for sub-tenon delivery |
| US7974856B2 (en) | 2005-11-30 | 2011-07-05 | The Invention Science Fund I, Llc | Computational systems and methods related to nutraceuticals |
| US10296720B2 (en) | 2005-11-30 | 2019-05-21 | Gearbox Llc | Computational systems and methods related to nutraceuticals |
| US8297028B2 (en) | 2006-06-14 | 2012-10-30 | The Invention Science Fund I, Llc | Individualized pharmaceutical selection and packaging |
| US7827042B2 (en) | 2005-11-30 | 2010-11-02 | The Invention Science Fund I, Inc | Methods and systems related to transmission of nutraceutical associated information |
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| US7927787B2 (en) | 2006-06-28 | 2011-04-19 | The Invention Science Fund I, Llc | Methods and systems for analysis of nutraceutical associated components |
| US8340944B2 (en) | 2005-11-30 | 2012-12-25 | The Invention Science Fund I, Llc | Computational and/or control systems and methods related to nutraceutical agent selection and dosing |
| US8068991B2 (en) * | 2005-11-30 | 2011-11-29 | The Invention Science Fund I, Llc | Systems and methods for transmitting pathogen related information and responding |
| US20100048660A1 (en) * | 2006-02-10 | 2010-02-25 | Graham Michael Wynne | Treatment of duchenne muscular dystrophy |
| WO2008020606A1 (fr) * | 2006-08-16 | 2008-02-21 | Kyowa Hakko Kirin Co., Ltd. | Agent anti-angiogénique |
| WO2008128538A1 (en) * | 2007-04-19 | 2008-10-30 | Leo Pharma A/S | Src family kinase inhibitors |
| CN101686665B (zh) | 2007-04-20 | 2014-04-23 | 奥克塞拉有限公司 | 用于治疗眼科疾病和紊乱的苯乙烯基衍生化合物 |
| US20090081277A1 (en) * | 2007-09-21 | 2009-03-26 | Allergan, Inc. | Pharmaceutical formulations and methods for treating ocular conditions |
| DK2346827T3 (da) | 2008-08-27 | 2014-02-03 | Leo Pharma As | Pyridinderivater som VEGFR-2 receptor og proteintyrosinkinasehæmmere |
| CN103804349A (zh) * | 2012-11-01 | 2014-05-21 | 杨子娇 | 一类治疗青光眼的化合物及其用途 |
| JO3425B1 (ar) | 2013-07-15 | 2019-10-20 | Novartis Ag | مشتقات البابيريدينيل-اندول واستخدامها كعامل متمم لمثبطات b |
| CN106458920B (zh) * | 2014-03-31 | 2019-02-15 | 千寿制药株式会社 | 炔基吲唑衍生物及其用途 |
| CN104744338A (zh) * | 2015-03-31 | 2015-07-01 | 天津维智精细化工有限公司 | 一种6-氯羟吲哚的合成方法 |
| WO2017024968A1 (zh) * | 2015-08-07 | 2017-02-16 | 南京明德新药研发股份有限公司 | 作为fgfr和vegfr抑制剂的乙烯基化合物 |
| CN109942544B (zh) * | 2017-12-21 | 2021-06-11 | 中国科学院合肥物质科学研究院 | 一类新型吲唑类衍生物激酶抑制剂 |
| WO2024032584A1 (zh) * | 2022-08-08 | 2024-02-15 | 苏州必扬医药科技有限公司 | 一种蛋白酪氨酸激酶抑制剂及其医疗用途 |
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2003
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- 2003-12-08 DE DE60314013T patent/DE60314013T2/de not_active Expired - Fee Related
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- 2003-12-08 DK DK03777064T patent/DK1585743T3/da active
- 2003-12-08 WO PCT/IB2003/005854 patent/WO2004056806A1/en active IP Right Grant
- 2003-12-08 NZ NZ540340A patent/NZ540340A/en unknown
- 2003-12-08 PL PL377713A patent/PL377713A1/pl not_active Application Discontinuation
- 2003-12-08 EP EP03777064A patent/EP1585743B1/en not_active Expired - Lifetime
- 2003-12-08 RS YUP-2005/0430A patent/RS20050430A/sr unknown
- 2003-12-08 CN CNA2003801096976A patent/CN1747950A/zh active Pending
- 2003-12-08 AU AU2003286321A patent/AU2003286321A1/en not_active Abandoned
- 2003-12-08 AP AP2005003341A patent/AP2005003341A0/xx unknown
- 2003-12-08 SI SI200330833T patent/SI1585743T1/sl unknown
- 2003-12-08 JP JP2004561821A patent/JP3814285B2/ja not_active Expired - Fee Related
- 2003-12-08 KR KR1020057011551A patent/KR100730267B1/ko not_active IP Right Cessation
- 2003-12-08 AT AT03777064T patent/ATE362928T1/de not_active IP Right Cessation
- 2003-12-08 BR BR0317548-0A patent/BR0317548A/pt not_active IP Right Cessation
- 2003-12-11 PE PE2003001269A patent/PE20041006A1/es not_active Application Discontinuation
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2005
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- 2005-06-15 EC EC2005005858A patent/ECSP055858A/es unknown
- 2005-06-16 HR HR20050559A patent/HRP20050559A2/hr not_active Application Discontinuation
- 2005-06-17 TN TNP2005000164A patent/TNSN05164A1/fr unknown
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- 2005-06-17 CR CR7882A patent/CR7882A/es not_active Application Discontinuation
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- 2005-07-18 NO NO20053486A patent/NO20053486L/no not_active Application Discontinuation
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