ZA200502341B - Novel piperidine derivatives for use in the tretment of chemokine mediated disease states. - Google Patents
Novel piperidine derivatives for use in the tretment of chemokine mediated disease states. Download PDFInfo
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- ZA200502341B ZA200502341B ZA200502341A ZA200502341A ZA200502341B ZA 200502341 B ZA200502341 B ZA 200502341B ZA 200502341 A ZA200502341 A ZA 200502341A ZA 200502341 A ZA200502341 A ZA 200502341A ZA 200502341 B ZA200502341 B ZA 200502341B
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- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/40—Oxygen atoms
- C07D211/44—Oxygen atoms attached in position 4
- C07D211/46—Oxygen atoms attached in position 4 having a hydrogen atom as the second substituent in position 4
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CN (1) | CN1684952A (es) |
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AR033517A1 (es) * | 2000-04-08 | 2003-12-26 | Astrazeneca Ab | Derivados de piperidina, proceso para su preparacion y uso de estos derivados en la fabricacion de medicamentos |
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JP2009511582A (ja) | 2005-10-11 | 2009-03-19 | シェーリング コーポレイション | Cxcr3拮抗薬活性を有する置換複素環式化合物 |
TWI433838B (zh) * | 2008-06-25 | 2014-04-11 | 必治妥美雅史谷比公司 | 作為趨化因子受體活性調節劑之六氫吡啶衍生物 |
GB0908394D0 (en) | 2009-05-15 | 2009-06-24 | Univ Leuven Kath | Novel viral replication inhibitors |
GB0913636D0 (en) * | 2009-08-05 | 2009-09-16 | Univ Leuven Kath | Novel viral replication inhibitors |
BR112013011737A2 (pt) | 2010-11-15 | 2016-08-09 | Univ Leuven Kath | composto, uso de um composto composição farmacêutica, e, método de tratamento ou prevenção de uma infecção por hiv |
KR101699822B1 (ko) | 2011-12-21 | 2017-01-25 | 노비라 테라퓨틱스, 인코포레이티드 | B형 간염의 항바이러스성 제제 |
AR092270A1 (es) | 2012-08-28 | 2015-04-08 | Janssen R&D Ireland | Sulfamoilarilamidas y su uso como medicamentos para el tratamiento de la hepatitis b |
PT2961732T (pt) | 2013-02-28 | 2017-06-26 | Janssen Sciences Ireland Uc | Sulfamoil-arilamidas e utilização das mesmas como medicamentos para o tratamento de hepatite b |
EA027068B1 (ru) | 2013-04-03 | 2017-06-30 | Янссен Сайенсиз Айрлэнд Юси | Производные n-фенилкарбоксамида и их применение в качестве лекарственных препаратов для лечения гепатита b |
JO3603B1 (ar) | 2013-05-17 | 2020-07-05 | Janssen Sciences Ireland Uc | مشتقات سلفامويل بيرولاميد واستخدامها كادوية لمعالجة التهاب الكبد نوع بي |
JP6441315B2 (ja) | 2013-05-17 | 2018-12-19 | ヤンセン・サイエンシズ・アイルランド・ユーシー | スルファモイルチオフェンアミド誘導体およびb型肝炎を治療するための医薬品としてのその使用 |
US10450270B2 (en) | 2013-07-25 | 2019-10-22 | Janssen Sciences Ireland Uc | Glyoxamide substituted pyrrolamide derivatives and the use thereof as medicaments for the treatment of hepatitis B |
MX368158B (es) | 2013-10-23 | 2019-09-20 | Janssen Sciences Ireland Uc | Derivados de carboxamida y su uso como medicamentos para el tratamiento de la hepatitis b. |
US10392349B2 (en) | 2014-01-16 | 2019-08-27 | Novira Therapeutics, Inc. | Azepane derivatives and methods of treating hepatitis B infections |
US9169212B2 (en) | 2014-01-16 | 2015-10-27 | Novira Therapeutics, Inc. | Azepane derivatives and methods of treating hepatitis B infections |
MX2016009449A (es) | 2014-02-05 | 2016-10-13 | Novira Therapeutics Inc | Terapia de combinacion para el tratamiento de infecciones por virus de la hepatitis b (vhb). |
EA035848B1 (ru) | 2014-02-06 | 2020-08-20 | Янссен Сайенсиз Айрлэнд Юси | Производные сульфамоилпирроламида и их применение в качестве медикаментов для лечения гепатита b |
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US10875876B2 (en) | 2015-07-02 | 2020-12-29 | Janssen Sciences Ireland Uc | Cyclized sulfamoylarylamide derivatives and the use thereof as medicaments for the treatment of hepatitis B |
AU2016330964B2 (en) | 2015-09-29 | 2021-04-01 | Novira Therapeutics, Inc. | Crystalline forms of a hepatitis B antiviral agent |
SG11201808949SA (en) | 2016-04-15 | 2018-11-29 | Novira Therapeutics Inc | Combinations and methods comprising a capsid assembly inhibitor |
CA3090125A1 (en) | 2018-03-14 | 2019-09-19 | Janssen Sciences Ireland Unlimited Company | Capsid assembly modulator dosing regimen |
US11096931B2 (en) | 2019-02-22 | 2021-08-24 | Janssen Sciences Ireland Unlimited Company | Amide derivatives useful in the treatment of HBV infection or HBV-induced diseases |
EP3966205A1 (en) | 2019-05-06 | 2022-03-16 | Janssen Sciences Ireland Unlimited Company | Amide derivatives useful in the treatment of hbv infection or hbv-induced diseases |
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US4588722A (en) * | 1984-01-09 | 1986-05-13 | Janssen Pharmaceutica N.V. | N-(4-piperidinyl) bicyclic condensed 2-imidazolamine derivatives |
US4695575A (en) * | 1984-11-13 | 1987-09-22 | Janssen Pharmaceutica, N.V. | 4-[(bicycle heterocyclyl)-methyl and -hetero]-piperidines |
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- 2003-09-12 BR BR0314688-0A patent/BR0314688A/pt not_active IP Right Cessation
- 2003-09-12 CA CA002497280A patent/CA2497280A1/en not_active Abandoned
- 2003-09-12 EP EP07010143A patent/EP1816123A1/en not_active Withdrawn
- 2003-09-12 EP EP03798620A patent/EP1546130B1/en not_active Expired - Lifetime
- 2003-09-12 DE DE60315323T patent/DE60315323T2/de not_active Expired - Fee Related
- 2003-09-12 KR KR1020057004938A patent/KR20050052511A/ko not_active Application Discontinuation
- 2003-09-12 PL PL03376119A patent/PL376119A1/xx not_active Application Discontinuation
-
2005
- 2005-03-18 ZA ZA200502341A patent/ZA200502341B/en unknown
- 2005-04-20 IS IS7813A patent/IS7813A/is unknown
- 2005-04-22 NO NO20051965A patent/NO20051965L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
NO20051965L (no) | 2005-06-23 |
NO20051965D0 (no) | 2005-04-22 |
DE60315323T2 (de) | 2008-04-17 |
AU2003259004B2 (en) | 2007-02-08 |
BR0314688A (pt) | 2005-08-02 |
WO2004029041A1 (en) | 2004-04-08 |
EP1546130A1 (en) | 2005-06-29 |
AU2003259004A1 (en) | 2004-04-19 |
EP1816123A1 (en) | 2007-08-08 |
KR20050052511A (ko) | 2005-06-02 |
SE0202838D0 (sv) | 2002-09-24 |
ATE368656T1 (de) | 2007-08-15 |
ES2289354T3 (es) | 2008-02-01 |
IS7813A (is) | 2005-04-20 |
EP1546130B1 (en) | 2007-08-01 |
PL376119A1 (en) | 2005-12-12 |
MXPA05003007A (es) | 2005-06-22 |
CN1684952A (zh) | 2005-10-19 |
DE60315323D1 (de) | 2007-09-13 |
RU2005105053A (ru) | 2005-12-10 |
CA2497280A1 (en) | 2004-04-08 |
NZ538527A (en) | 2006-10-27 |
JP2006503066A (ja) | 2006-01-26 |
US20060040984A1 (en) | 2006-02-23 |
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