ZA200502326B - Therapeutic piperazine compounds - Google Patents

Therapeutic piperazine compounds Download PDF

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Publication number
ZA200502326B
ZA200502326B ZA200502326A ZA200502326A ZA200502326B ZA 200502326 B ZA200502326 B ZA 200502326B ZA 200502326 A ZA200502326 A ZA 200502326A ZA 200502326 A ZA200502326 A ZA 200502326A ZA 200502326 B ZA200502326 B ZA 200502326B
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ZA
South Africa
Prior art keywords
compound
halo
phenyl
alkyl
membered
Prior art date
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ZA200502326A
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English (en)
Inventor
Qun Sun
Xiaoming Zhou
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Euro Celtique Sa
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Publication of ZA200502326B publication Critical patent/ZA200502326B/en

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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A61P29/02—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID] without antiinflammatory effect
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/02—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
    • C07D241/10—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
    • C07D241/14—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D241/20—Nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond

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  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Addiction (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Psychology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
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  • Urology & Nephrology (AREA)
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  • Diabetes (AREA)
  • Otolaryngology (AREA)
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  • Nutrition Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
ZA200502326A 2002-09-24 2005-03-18 Therapeutic piperazine compounds ZA200502326B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US41284702P 2002-09-24 2002-09-24

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ZA200502326B true ZA200502326B (en) 2006-05-31

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ZA200502326A ZA200502326B (en) 2002-09-24 2005-03-18 Therapeutic piperazine compounds

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Country Link
US (4) US7157462B2 (enExample)
EP (2) EP1810970B8 (enExample)
JP (1) JP4560610B2 (enExample)
KR (1) KR20050052514A (enExample)
CN (1) CN100393713C (enExample)
AT (2) ATE356817T1 (enExample)
AU (1) AU2003272685A1 (enExample)
BR (1) BR0314699A (enExample)
CA (1) CA2500113C (enExample)
CY (1) CY1106634T1 (enExample)
DE (2) DE60312544T2 (enExample)
DK (1) DK1562936T3 (enExample)
ES (1) ES2285170T3 (enExample)
MX (1) MXPA05003302A (enExample)
NZ (1) NZ539205A (enExample)
PT (1) PT1562936E (enExample)
SI (1) SI1562936T1 (enExample)
WO (1) WO2004029031A2 (enExample)
ZA (1) ZA200502326B (enExample)

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BR0314699A (pt) 2005-08-09
ATE467627T1 (de) 2010-05-15
MXPA05003302A (es) 2005-10-18
US20110082152A1 (en) 2011-04-07
US7855210B2 (en) 2010-12-21
US7157462B2 (en) 2007-01-02
CA2500113A1 (en) 2004-04-08
JP2006508067A (ja) 2006-03-09
SI1562936T1 (sl) 2007-08-31
EP1562936A2 (en) 2005-08-17
HK1083216A1 (en) 2006-06-30
US20050059671A1 (en) 2005-03-17
PT1562936E (pt) 2007-06-12
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CN100393713C (zh) 2008-06-11
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