ZA200202518B - Certain alkylene diamine-substituted heterocycles. - Google Patents

Certain alkylene diamine-substituted heterocycles.

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Publication number
ZA200202518B
ZA200202518B ZA200202518A ZA200202518A ZA200202518B ZA 200202518 B ZA200202518 B ZA 200202518B ZA 200202518 A ZA200202518 A ZA 200202518A ZA 200202518 A ZA200202518 A ZA 200202518A ZA 200202518 B ZA200202518 B ZA 200202518B
Authority
ZA
South Africa
Prior art keywords
alkylene diamine
substituted heterocycles
certain alkylene
certain
novel compounds
Prior art date
Application number
ZA200202518A
Other languages
English (en)
Inventor
Raymond F Horvath
Jennifer Tran
Stephane De Lombaert
Hodgetts Keven Julian
Philip A Carpino
David A Griffith
Original Assignee
Neurogen Corp Pfizer Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Neurogen Corp Pfizer Inc filed Critical Neurogen Corp Pfizer Inc
Publication of ZA200202518B publication Critical patent/ZA200202518B/xx

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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
    • C07D213/73—Unsubstituted amino or imino radicals
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    • C07D215/38—Nitrogen atoms
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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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ZA200202518A 1999-09-30 2002-03-28 Certain alkylene diamine-substituted heterocycles. ZA200202518B (en)

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Application Number Priority Date Filing Date Title
US15687099P 1999-09-30 1999-09-30

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ZA200202518B true ZA200202518B (en) 2003-08-27

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ZA200202518A ZA200202518B (en) 1999-09-30 2002-03-28 Certain alkylene diamine-substituted heterocycles.

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US (3) US6506762B1 (pl)
EP (1) EP1224187B1 (pl)
JP (2) JP2003510327A (pl)
KR (1) KR20020043223A (pl)
CN (1) CN1377356A (pl)
AT (1) ATE318267T1 (pl)
AU (1) AU7738000A (pl)
BG (1) BG106508A (pl)
CA (1) CA2379640C (pl)
CZ (1) CZ20021086A3 (pl)
DE (1) DE60026155T2 (pl)
EA (1) EA200200424A1 (pl)
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HU (1) HUP0202636A3 (pl)
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OA (1) OA12050A (pl)
PL (1) PL354784A1 (pl)
WO (1) WO2001023389A2 (pl)
ZA (1) ZA200202518B (pl)

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US20030158197A1 (en) 2003-08-21
CA2379640A1 (en) 2001-04-05
PL354784A1 (pl) 2004-02-23
WO2001023389A3 (en) 2002-05-10
DE60026155D1 (de) 2006-04-27
AU7738000A (en) 2001-04-30
DE60026155T2 (de) 2006-08-10
EA200200424A1 (ru) 2002-12-26
HUP0202636A3 (en) 2004-06-28
US20040229870A1 (en) 2004-11-18
OA12050A (en) 2006-05-02
JP2008007515A (ja) 2008-01-17
CZ20021086A3 (cs) 2002-10-16
US6506762B1 (en) 2003-01-14
WO2001023389A2 (en) 2001-04-05
CN1377356A (zh) 2002-10-30
IL148903A0 (en) 2002-09-12
JP2003510327A (ja) 2003-03-18
EP1224187A2 (en) 2002-07-24
US6696445B2 (en) 2004-02-24
US7074929B2 (en) 2006-07-11
NO20021358D0 (no) 2002-03-19
KR20020043223A (ko) 2002-06-08
BG106508A (en) 2003-02-28
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ATE318267T1 (de) 2006-03-15
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EP1224187B1 (en) 2006-02-22

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