YU48079B - Heterociklična jedinjenja - Google Patents

Heterociklična jedinjenja

Info

Publication number
YU48079B
YU48079B YU142791A YU142791A YU48079B YU 48079 B YU48079 B YU 48079B YU 142791 A YU142791 A YU 142791A YU 142791 A YU142791 A YU 142791A YU 48079 B YU48079 B YU 48079B
Authority
YU
Yugoslavia
Prior art keywords
group
alkyl
heterocyclic units
alkyl group
formula
Prior art date
Application number
YU142791A
Other languages
English (en)
Other versions
YU142791A (sh
Inventor
A. Perboni
T. Rossi
G. Gaviraghi
G. Tarzia
A. Ursini
Original Assignee
Glaxo S.P.A.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB909018330A external-priority patent/GB9018330D0/en
Priority claimed from GB919104770A external-priority patent/GB9104770D0/en
Application filed by Glaxo S.P.A. filed Critical Glaxo S.P.A.
Priority to SI9111427A priority Critical patent/SI9111427B/sl
Publication of YU142791A publication Critical patent/YU142791A/sh
Priority to HR940556A priority patent/HRP940556B1/xx
Publication of YU48079B publication Critical patent/YU48079B/sh

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D477/00—Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Heat Sensitive Colour Forming Recording (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

HETEROCIKLIČNA JEDINJENJA edinjenja opšte formule (I): naznačena time, što u formuli R1 pretstavlja grupu: gde R4 pretstavlja vodonik ili C1-4 alkil grupu; p je nula ili jedan; R5 pretstavlja grupu koja je izabrana od C1-6 alkil, C5-6 cik-loalkil koji je opciono supstituisan sa C1-3 alkil grupom, fenil ili C1-4 alkil koji je supstituisan sa C1-3 alkoksi grupom; i R2 pretstavlja grupu OR3 gde R3 pretstavlja C1-5 alkil grupu. Prijava sadrži još 1 nezavisan i 8 zavisnih zahteva.
YU142791A 1990-08-21 1991-08-20 Heterociklična jedinjenja YU48079B (sh)

Priority Applications (2)

Application Number Priority Date Filing Date Title
SI9111427A SI9111427B (sl) 1990-08-21 1991-08-20 Heterociklične spojine
HR940556A HRP940556B1 (en) 1990-08-21 1994-09-16 Heterocyclic compounds

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB909018330A GB9018330D0 (en) 1990-08-21 1990-08-21 Heterocyclic compounds
GB919104770A GB9104770D0 (en) 1991-03-07 1991-03-07 Heterocyclic compounds

Publications (2)

Publication Number Publication Date
YU142791A YU142791A (sh) 1994-01-20
YU48079B true YU48079B (sh) 1997-01-08

Family

ID=26297540

Family Applications (1)

Application Number Title Priority Date Filing Date
YU142791A YU48079B (sh) 1990-08-21 1991-08-20 Heterociklična jedinjenja

Country Status (32)

Country Link
US (1) US5587374A (sh)
EP (1) EP0495953B1 (sh)
JP (2) JP3151215B2 (sh)
KR (1) KR0169147B1 (sh)
CN (1) CN1030917C (sh)
AP (1) AP238A (sh)
AT (1) ATE106887T1 (sh)
AU (1) AU647178B2 (sh)
CA (1) CA2067741C (sh)
CY (1) CY2037A (sh)
CZ (1) CZ280942B6 (sh)
DE (1) DE69102415T2 (sh)
DK (1) DK0495953T3 (sh)
ES (1) ES2054502T3 (sh)
FI (1) FI97136C (sh)
HK (1) HK19495A (sh)
HR (1) HRP940556B1 (sh)
HU (2) HUT61024A (sh)
IE (1) IE66122B1 (sh)
IL (1) IL99248A (sh)
MX (1) MX9100743A (sh)
MY (1) MY106997A (sh)
NO (1) NO300176B1 (sh)
NZ (1) NZ239474A (sh)
OA (1) OA09578A (sh)
PL (1) PL169425B1 (sh)
PT (1) PT98729B (sh)
SG (1) SG169494G (sh)
SI (1) SI9111427B (sh)
SK (1) SK121392A3 (sh)
WO (1) WO1992003437A1 (sh)
YU (1) YU48079B (sh)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9104838D0 (en) * 1991-03-07 1991-04-17 Glaxo Spa Heterocyclic compounds
AP294A (en) * 1992-08-31 1993-12-28 Glaxo Spa "10-(1-Hydroxyethyl)-11-oxo-1-azatricyclo-(7.2.0.0.3.8) undec-2-ene-2-carboxylic acid derivatives".
GB9218781D0 (en) * 1992-09-04 1992-10-21 Glaxo Spa Heterocyclic derivatives
IN188720B (sh) * 1997-11-06 2002-11-02 Panacea Biotec Ltd
JP4377231B2 (ja) 2001-11-05 2009-12-02 大日本住友製薬株式会社 新規なカルバペネム化合物
WO2004089954A1 (ja) * 2003-04-08 2004-10-21 Sumitomo Pharmaceuticals Co., Ltd. 新規なカルバペネム化合物
EP1785426A4 (en) * 2004-09-03 2008-02-20 Dainippon Sumitomo Pharma Co NEW CARBAPENEM DERIVATIVE
WO2006103999A1 (ja) * 2005-03-25 2006-10-05 Dainippon Sumitomo Pharma Co., Ltd. 新規なカルバペネム化合物
EP2085084A1 (en) 2008-01-29 2009-08-05 LEK Pharmaceuticals D.D. Use of inhibitor of beta-lactamases and its combination with beta-lactam antibiotics
EP2135871A1 (en) * 2008-06-18 2009-12-23 LEK Pharmaceuticals D.D. New trinem antibiotics and inhibitors of beta-lactamases
CN110869016B (zh) 2017-05-08 2023-09-12 葛兰素史密斯克莱知识产权发展有限公司 用于治疗分枝杆菌感染的山费培南或其盐或酯

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1425571A (en) * 1972-03-13 1976-02-18 Astra Laekemedel Ab Penicillins and cephaosporins
GB1433131A (en) * 1972-03-13 1976-04-22 Astra Laekemedel Ab Penicillins
DE2811514A1 (de) * 1977-03-19 1978-09-21 Beecham Group Ltd Ester der 7-oxo-1-azabicyclo eckige klammer auf 3.2.0 eckige klammer zu hept- 2-en-2-carbonsaeure und deren derivate, verfahren zur herstellung dieser verbindungen und diese verbindungen enthaltende pharmazeutische zubereitungen
US4374849A (en) * 1981-09-14 1983-02-22 Merck & Co., Inc. 6-Amidocyclonocardicins
US4374848A (en) * 1981-09-14 1983-02-22 Merck & Co., Inc. 6-(1-Hydroxyethyl)cyclonocardicin
CZ285778B6 (cs) * 1989-09-08 1999-11-17 Glaxo S.P.A. Kyselina 10-(1-hydroxyethyl)-11-oxo-1-azatricyklo/7,2,0,03,8/-undec-2en-2-karboxylová a její deriváty, způsob jejich výroby, použití pro výrobu farmaceutických prostředků a farmaceutické prostředky s jejich obsahem
AU636913B2 (en) * 1989-10-11 1993-05-13 Takeda Chemical Industries Ltd. Tricyclic carbapenem compounds
GB9104832D0 (en) * 1991-03-07 1991-04-17 Glaxo Spa Heterocyclic compounds
GB9104838D0 (en) * 1991-03-07 1991-04-17 Glaxo Spa Heterocyclic compounds

Also Published As

Publication number Publication date
EP0495953A1 (en) 1992-07-29
KR0169147B1 (en) 1999-01-15
SK278470B6 (en) 1997-06-04
DK0495953T3 (da) 1994-07-18
JPH05502044A (ja) 1993-04-15
CN1030917C (zh) 1996-02-07
JP3151215B2 (ja) 2001-04-03
ES2054502T3 (es) 1994-08-01
WO1992003437A1 (en) 1992-03-05
AP238A (en) 1993-02-04
IE912944A1 (en) 1992-02-26
FI921717A0 (fi) 1992-04-16
HU211584A9 (en) 1995-12-28
MY106997A (en) 1995-08-30
SG169494G (en) 1995-04-28
HU9201303D0 (en) 1992-07-28
PT98729A (pt) 1992-07-31
NO921521L (no) 1992-06-22
EP0495953B1 (en) 1994-06-08
HK19495A (en) 1995-02-17
IE66122B1 (en) 1995-12-13
NZ239474A (en) 1994-06-27
CA2067741A1 (en) 1992-02-22
OA09578A (en) 1993-01-31
CN1060094A (zh) 1992-04-08
SI9111427B (sl) 2000-10-31
HUT61024A (en) 1992-11-30
SK121392A3 (en) 1997-06-04
YU142791A (sh) 1994-01-20
PT98729B (pt) 1999-01-29
AU647178B2 (en) 1994-03-17
DE69102415T2 (de) 1994-10-13
NO300176B1 (no) 1997-04-21
HRP940556A2 (en) 1996-06-30
PL169425B1 (pl) 1996-07-31
JP2000351730A (ja) 2000-12-19
AU8421291A (en) 1992-03-17
CZ280942B6 (cs) 1996-05-15
DE69102415D1 (de) 1994-07-14
FI97136B (fi) 1996-07-15
JP3461786B2 (ja) 2003-10-27
FI921717A (fi) 1992-04-16
AP9100320A0 (en) 1991-10-31
CA2067741C (en) 2002-01-01
NO921521D0 (no) 1992-04-15
CZ121392A3 (en) 1993-04-14
KR920702361A (ko) 1992-09-03
HRP940556B1 (en) 2000-06-30
US5587374A (en) 1996-12-24
IL99248A (en) 1996-01-31
FI97136C (fi) 1996-10-25
SI9111427A (en) 1996-12-31
CY2037A (en) 1998-02-20
ATE106887T1 (de) 1994-06-15
MX9100743A (es) 1992-04-01
IL99248A0 (en) 1992-07-15

Similar Documents

Publication Publication Date Title
FI862621A0 (fi) Estrar av (met)-akrylsyror och deras anvaendning.
CO5050332A1 (es) Composiciones fungicidas que comprenden 2-metoxibenzofenonas
HUP9900582A2 (hu) Halogén-pirimidin-származékok, intermedierjeik, előállításuk és alkalmazásuk, a vegyületeket hatóanyagként tartalmazó kártevőirtó készítmények
HUP9802304A2 (hu) Piridazin-3-on-származékok, intermedierjeik, alkalmazásuk, a vegyületeket hatóanyagként tartalmazó herbicid készítmények
MY132009A (en) Pharmaceutical compounds.
YU48079B (sh) Heterociklična jedinjenja
ES2177058T3 (es) Compuestos eter piperidinilaminometil trifluorometil ciclicos como antagonistas de la sustancia p.
FI834730A (fi) 1-karboxialkanoylperhydro-indol-2- karboxylsyror och deras derivat.
ES482799A1 (es) Un metodo de preparar nuevas diaminas.
NO861563L (no) Neglelakk.
YU47047B (sh) Supstituisani 3-amino-2-benzoilcikloheks-2-enoni, postupak za njihovo dobijanje i primena za dobijanje herbicica
MX9303976A (es) Derivados de 2-amino-n-{{((4-(aminocarbonil)-pirimidin-2-il-amino)-alquil}-pirimidi n-4-carboxamida, su preparacion y su aplicacion en terapeutica.
ES8100238A1 (es) Un procedimiento para la preparacion de derivados del acido oxisustituido-ciclohexilacetico
ATE120453T1 (de) Inhibitoren fur angiotensin umwandelnde enzyme.
FI824407L (fi) Foerfarande foer framstaellning av vid behandling av magsaor anvaendbara pyrimidinderivat
FI942265A (fi) 2-aminopyratsin-5-karboksamidijohdannaiset, niiden valmistus ja terapeuttinen käyttö
ECSP951529A (es) Compuestos farmaceuticos
CO4810303A1 (es) Derivados de n-[3-[2-[(2,3-dihidro-1h-inden-2-il)alquilami- no]-etil]fenil]carboxamida, su preparacion y su aplicacion en terapeutica
YU47071B (sh) Spiro jedinjenje
YU86391A (sh) Nova antidijabetska i hipoglikemijska jedinjenja