YU44185B - Process of a selective acylated n-protected derivatives of an amino-glycoside antibiotic - Google Patents
Process of a selective acylated n-protected derivatives of an amino-glycoside antibioticInfo
- Publication number
- YU44185B YU44185B YU2743/79A YU274379A YU44185B YU 44185 B YU44185 B YU 44185B YU 2743/79 A YU2743/79 A YU 2743/79A YU 274379 A YU274379 A YU 274379A YU 44185 B YU44185 B YU 44185B
- Authority
- YU
- Yugoslavia
- Prior art keywords
- acylated
- selective
- amino
- protected derivatives
- glycoside antibiotic
- Prior art date
Links
- 229940126574 aminoglycoside antibiotic Drugs 0.000 title 1
- 239000002647 aminoglycoside antibiotic agent Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H23/00—Compounds containing boron, silicon or a metal, e.g. chelates or vitamin B12
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
- C07H15/20—Carbocyclic rings
- C07H15/22—Cyclohexane rings, substituted by nitrogen atoms
- C07H15/222—Cyclohexane rings substituted by at least two nitrogen atoms
- C07H15/226—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings
- C07H15/234—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings attached to non-adjacent ring carbon atoms of the cyclohexane rings, e.g. kanamycins, tobramycin, nebramycin, gentamicin A2
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Biochemistry (AREA)
- Biotechnology (AREA)
- General Health & Medical Sciences (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Saccharide Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP13840278A JPS5564598A (en) | 1978-11-11 | 1978-11-11 | Preparation of aminoglycoside antibiotic having selectively protected amino group |
| JP7306479A JPS55164696A (en) | 1979-06-12 | 1979-06-12 | Preparation of protected derivative of aminoglycoside antibiotic substance wherein amino groups other than 1-position are selectively protected, and preparation of 1-n- alpha-hydroxy-omega-aminoalkanoyl -aminoglycoside antibiotic substance |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| YU274379A YU274379A (en) | 1983-02-28 |
| YU44185B true YU44185B (en) | 1990-04-30 |
Family
ID=26414188
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| YU2743/79A YU44185B (en) | 1978-11-11 | 1979-11-08 | Process of a selective acylated n-protected derivatives of an amino-glycoside antibiotic |
Country Status (20)
Families Citing this family (22)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS55105699A (en) * | 1979-02-05 | 1980-08-13 | Microbial Chem Res Found | 3',4'-dideoxykanamycin a and its 1-n-aminoalkanoyl derivative |
| US4468512A (en) * | 1980-09-22 | 1984-08-28 | Eli Lilly And Company | 1-N-Acylated and 1-N-alkylated derivatives of 4-O-substituted-2-deoxystreptamine aminoglycosides |
| US4424344A (en) | 1980-09-22 | 1984-01-03 | Eli Lilly And Company | 2-N-Acylated and 2-N-alkylated derivatives of 4-O-substituted-2-deoxystreptamine aminoglycosides and process |
| US4424345A (en) | 1980-09-22 | 1984-01-03 | Eli Lilly And Company | 1-N-Acylated and 1-N-alkylated derivatives of 4-O-substituted-2-deoxystreptamine aminoglycosides and process |
| IT1200774B (it) * | 1985-10-10 | 1989-01-27 | Pierrel Spa | Procedimento di sentisi dell'amikacina |
| US4833232A (en) * | 1986-05-02 | 1989-05-23 | Exxon Research And Engineering Company | Synthesis of novel highly intrinsic conducting organic polymers |
| US5442047A (en) * | 1991-12-04 | 1995-08-15 | Schering Corporation | Process for preparing isepamicin |
| ATE152094T1 (de) * | 1989-06-21 | 1997-05-15 | Schering Corp | N-geschützte (s)-isoserin-verbindungen |
| IT1237490B (it) * | 1989-09-22 | 1993-06-07 | Chementecno S R L Monza Milano | Procedimento per la sintesi della 1 n (s delta ammino alfa idrossibutirril)kamanycin a basato sul trattamento della 1 n (s delta benzilossicarbonilammino alfa idrossibutirril) 3,6' di n benzilossicarbonilkanamycin a con acido formico |
| EP0446670B1 (en) * | 1990-03-08 | 1994-09-21 | Biochimica Opos Spa | Method of preparation of amikacin precursors |
| US5488038A (en) | 1992-11-27 | 1996-01-30 | Zaidan Hojin Biseibutsu Kagaku Kenkyu Kai | Dibekacin derivatives and arbekacin derivatives active against resistant bacteria |
| KR0139021B1 (ko) * | 1995-02-09 | 1998-04-30 | 김은영 | 1-엔(n)-에틸시소마이신의 제조방법 |
| KR100927626B1 (ko) * | 2002-09-18 | 2009-11-20 | 쯔지앙 하이썬 파머슈티컬 컴퍼니, 리미티드 | 이세파마이신의 제조 방법 |
| KR100467506B1 (ko) * | 2002-10-01 | 2005-01-24 | 경동제약 주식회사 | 이세파마이신의 제조방법 |
| US7794713B2 (en) | 2004-04-07 | 2010-09-14 | Lpath, Inc. | Compositions and methods for the treatment and prevention of hyperproliferative diseases |
| US7862812B2 (en) | 2006-05-31 | 2011-01-04 | Lpath, Inc. | Methods for decreasing immune response and treating immune conditions |
| CN102256989B (zh) | 2008-10-03 | 2016-01-06 | 聚糖生物科学有限责任公司 | 糖基化细菌代谢物的阴离子轭合物 |
| CN101928310B (zh) * | 2010-03-26 | 2012-09-05 | 常州方圆制药有限公司 | 3,2’,6’-三-N-乙酰基庆大霉素C1a的制备方法 |
| CN102250166A (zh) * | 2010-05-21 | 2011-11-23 | 江西济民可信集团有限公司 | 一种依替米星硫酸盐的制备方法 |
| CN102746349B (zh) * | 2012-06-27 | 2014-07-30 | 常州方圆制药有限公司 | 一种硫酸依替米星中间体3，2’，6’-三-N-乙酰基庆大霉素Cla的合成方法 |
| CN111138505B (zh) * | 2020-02-17 | 2021-10-08 | 山东安信制药有限公司 | 一种阿米卡星的制备方法 |
| CN116333011A (zh) * | 2023-03-31 | 2023-06-27 | 江西师范大学 | 一种全脱乙酰化壳寡糖及其制备方法和应用 |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FI52847C (fi) * | 1971-09-15 | 1977-12-12 | Suomen Sokeri Oy | Menetelmä ainakin kaksi hydroksyyliryhmää sisältävien yhdisteiden alky yli-, alkenyyli- tai asyylijohdannaisten valmistamiseksi |
| US3781268A (en) * | 1972-01-27 | 1973-12-25 | Bristol Myers Co | Antibiotic derivatives of kanamycin |
| GB1402427A (en) * | 1972-05-03 | 1975-08-06 | Ranks Hovis Mcdougall Ltd | Antibiotics |
| US4107424A (en) * | 1972-10-06 | 1978-08-15 | Zaidan Hojin Biseibutsu Kagaku Kenkyu Kai | 1-N-[(S)-α-hydroxy-ω-aminoacyl] derivatives of 3',4'-dideoxykanamycin B and 3'-deoxykanamycin B antibiotics |
| US4001208A (en) * | 1972-10-06 | 1977-01-04 | Zaidan Hojin Biseibutsu Kagaku Kenkyo Kai | 1-N-[(S)-α-hydroxy-ω-aminoacyl] |
| JPS5324415B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) * | 1972-10-06 | 1978-07-20 | ||
| GB1441202A (en) * | 1973-05-15 | 1976-06-30 | Microbial Chem Res Found | 1-n-isoserylkanamycins and the production thereof |
| JPS554118B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) * | 1973-08-29 | 1980-01-29 | ||
| JPS5635195B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) * | 1974-01-24 | 1981-08-15 | ||
| US4136254A (en) * | 1976-06-17 | 1979-01-23 | Schering Corporation | Process of selectively blocking amino functions in aminoglycosides using transition metal salts and intermediates used thereby |
-
1979
- 1979-10-23 IE IE2026/79A patent/IE48972B1/en not_active IP Right Cessation
- 1979-10-24 IN IN1104/CAL/79A patent/IN151454B/en unknown
- 1979-10-25 SE SE7908850A patent/SE446632B/sv not_active IP Right Cessation
- 1979-10-26 NL NL7907892A patent/NL7907892A/nl not_active Application Discontinuation
- 1979-10-29 CH CH184/84A patent/CH650005A5/de not_active IP Right Cessation
- 1979-10-29 CH CH9682/79A patent/CH650004A5/de not_active IP Right Cessation
- 1979-11-02 US US06/090,591 patent/US4297485A/en not_active Expired - Lifetime
- 1979-11-02 AT AT0707979A patent/AT367066B/de not_active IP Right Cessation
- 1979-11-08 YU YU2743/79A patent/YU44185B/xx unknown
- 1979-11-08 FR FR7928015A patent/FR2441631A1/fr active Granted
- 1979-11-08 AU AU52622/79A patent/AU529682B2/en not_active Expired
- 1979-11-08 DE DE2945010A patent/DE2945010C2/de not_active Expired
- 1979-11-08 DE DE2953878A patent/DE2953878C2/de not_active Expired
- 1979-11-08 MX MX798478U patent/MX6181E/es unknown
- 1979-11-08 PH PH23263A patent/PH16263A/en unknown
- 1979-11-08 ES ES485830A patent/ES485830A1/es not_active Expired
- 1979-11-09 GB GB8103076A patent/GB2065123B/en not_active Expired
- 1979-11-09 CA CA000339531A patent/CA1118416A/en not_active Expired
- 1979-11-09 LU LU81881A patent/LU81881A1/fr unknown
- 1979-11-09 DK DK476679A patent/DK476679A/da not_active Application Discontinuation
- 1979-11-09 GB GB7938894A patent/GB2036020B/en not_active Expired
- 1979-11-09 AR AR79278828A patent/AR241915A1/es active
- 1979-11-12 IT IT09592/79A patent/IT1166021B/it active
-
1980
- 1980-06-16 ES ES492479A patent/ES8105747A1/es not_active Expired
- 1980-12-22 PH PH25015A patent/PH15906A/en unknown
-
1981
- 1981-06-03 FR FR8110968A patent/FR2482109A1/fr active Granted
-
1984
- 1984-12-13 SE SE8406344A patent/SE463264B/sv not_active IP Right Cessation
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