UY36466A - Formulaciones inyectables de paracetamol - Google Patents

Formulaciones inyectables de paracetamol

Info

Publication number
UY36466A
UY36466A UY0001036466A UY36466A UY36466A UY 36466 A UY36466 A UY 36466A UY 0001036466 A UY0001036466 A UY 0001036466A UY 36466 A UY36466 A UY 36466A UY 36466 A UY36466 A UY 36466A
Authority
UY
Uruguay
Prior art keywords
paracetamol
intravenous
slow
injectable formulations
formulations
Prior art date
Application number
UY0001036466A
Other languages
English (en)
Inventor
Ketan R Patel
Milan R Patel
Asheel K Patel
Prakashchandra J Shah
Original Assignee
Troikaa Pharmaceuticals Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=55022620&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UY36466(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Troikaa Pharmaceuticals Ltd filed Critical Troikaa Pharmaceuticals Ltd
Publication of UY36466A publication Critical patent/UY36466A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/22Heterocyclic compounds, e.g. ascorbic acid, tocopherol or pyrrolidones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • A61K31/165Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A61K31/167Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the nitrogen of a carboxamide group directly attached to the aromatic ring, e.g. lidocaine, paracetamol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/02Inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/10Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/08Solutions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Pain & Pain Management (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Dermatology (AREA)
  • Engineering & Computer Science (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Inorganic Chemistry (AREA)
  • Neurosurgery (AREA)
  • Rheumatology (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

La presente invención se relaciona con la disminución del volumen de las inyecciones intravenosas de paracetamol, o de su sal farmacéuticamente aceptada, y del método de preparación. Las formulaciones proveen altas concentraciones de paracetamol, o su sal farmacéuticamente aceptada, en un sistema solvente. Tales formulaciones no sólo pueden ser administradas a través de rutas intra-musculares e infusiones intravenosas, sino también mediante bolos IV lentos después de ser diluidas con fluidos acuosos a un volumen final no mayor a 20 Ml, y permanecen estables y son aptas para la administración mediante una ruta intravenosa lenta con efectos secundarios minimizados.
UY0001036466A 2014-12-20 2015-12-21 Formulaciones inyectables de paracetamol UY36466A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IN4102MU2014 2014-12-20

Publications (1)

Publication Number Publication Date
UY36466A true UY36466A (es) 2016-07-29

Family

ID=55022620

Family Applications (1)

Application Number Title Priority Date Filing Date
UY0001036466A UY36466A (es) 2014-12-20 2015-12-21 Formulaciones inyectables de paracetamol

Country Status (28)

Country Link
US (1) US20180000940A1 (es)
EP (1) EP3233055A1 (es)
JP (1) JP2017538762A (es)
KR (1) KR20170099911A (es)
CN (1) CN107205924A (es)
AR (1) AR103188A1 (es)
AU (1) AU2015365533A1 (es)
BR (1) BR112017012975B1 (es)
CA (1) CA2969303A1 (es)
CL (1) CL2017001629A1 (es)
CO (1) CO2017006268A2 (es)
CU (1) CU20170088A7 (es)
DO (1) DOP2017000134A (es)
EA (1) EA201791409A1 (es)
EC (1) ECSP17038668A (es)
IL (1) IL252729A0 (es)
JO (1) JO3689B1 (es)
MA (1) MA40599A1 (es)
MD (1) MD20170071A2 (es)
MX (1) MX2017008264A (es)
PE (1) PE20171305A1 (es)
PH (1) PH12017501005A1 (es)
SG (1) SG11201704435PA (es)
TN (1) TN2017000232A1 (es)
TW (1) TWI649097B (es)
UA (1) UA122136C2 (es)
UY (1) UY36466A (es)
WO (1) WO2016097899A1 (es)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN107229455B (zh) 2016-03-24 2019-09-17 阿里巴巴集团控股有限公司 一种业务处理方法、装置及系统

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2751875B1 (fr) 1996-08-05 1998-12-24 Scr Newpharm Nouvelles formulations liquides stables a base de paracetamol et leur mode de preparation
IT1301976B1 (it) * 1998-07-31 2000-07-20 Angelini Ricerche Spa Composizione farmaceutica iniettabile a base di paracetamolo
IT1313579B1 (it) 1999-07-30 2002-09-09 Acraf Composizione farmaceutica liquida a base di paracetamolo.
ITMI20012135A1 (it) 2001-10-16 2003-04-16 Bioren S A Soluzioni iniettabili pronte all'uso di paracetamolo
MX2007014862A (es) * 2005-05-27 2008-02-21 Panacea Biotec Ltd Composiciones inyectables y procedimiento para la preparacion de dichas composiciones.
DK1973527T3 (da) * 2005-12-15 2010-02-01 Acusphere Inc Fremgangsmåder til fremstilling af partikelbaserede farmaceutiske formulationer til parenteral indgivelse
EP2170313A2 (en) 2007-06-18 2010-04-07 Combino Pharm, S.L. Aqueous formulations of acetaminophen for injection
WO2009098716A2 (en) 2008-01-17 2009-08-13 Aptuit Laurus Private Limited Stable pharmaceutical aqueous compositions
CN102159184B (zh) * 2008-10-09 2013-09-04 方济各安吉利克化学联合股份有限公司 含有对乙酰氨基酚的液体药物制剂
BR112012031928B1 (pt) 2010-06-30 2021-08-31 Troikaa Pharmaceuticals Ltd Composições farmacêuticas as quais incluem paracetamol e processo para preparação do mesmo
TWI577377B (zh) * 2010-09-16 2017-04-11 Viiv醫療保健公司 醫藥組合物
CN102258485A (zh) * 2011-01-11 2011-11-30 北京润德康医药技术有限公司 一种含对乙酰氨基酚的注射用制剂及其应用
CN102600068A (zh) * 2011-01-24 2012-07-25 联康药业克雷恩特塞提斯制药实验室有限责任公司 稳定即用的可注射扑热息痛制剂

Also Published As

Publication number Publication date
CA2969303A1 (en) 2016-06-23
CU20170088A7 (es) 2018-03-13
MX2017008264A (es) 2017-10-02
CN107205924A (zh) 2017-09-26
EP3233055A1 (en) 2017-10-25
SG11201704435PA (en) 2017-06-29
WO2016097899A1 (en) 2016-06-23
ECSP17038668A (es) 2017-12-01
KR20170099911A (ko) 2017-09-01
CL2017001629A1 (es) 2018-03-16
PH12017501005A1 (en) 2017-12-11
JP2017538762A (ja) 2017-12-28
JO3689B1 (ar) 2020-08-27
TW201622703A (zh) 2016-07-01
TWI649097B (zh) 2019-02-01
MA40599A1 (fr) 2017-11-30
BR112017012975A2 (pt) 2018-02-27
TN2017000232A1 (en) 2018-10-19
IL252729A0 (en) 2017-08-31
UA122136C2 (uk) 2020-09-25
AR103188A1 (es) 2017-04-19
DOP2017000134A (es) 2017-09-15
PE20171305A1 (es) 2017-09-05
US20180000940A1 (en) 2018-01-04
MD20170071A2 (ro) 2017-09-30
AU2015365533A1 (en) 2017-07-06
BR112017012975B1 (pt) 2023-09-26
EA201791409A1 (ru) 2017-10-31
CO2017006268A2 (es) 2017-10-20

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