UY34973A - Proceso para la preparación de derivados de éster heterocíclicos inhibidores de c-fms quinasa - Google Patents

Proceso para la preparación de derivados de éster heterocíclicos inhibidores de c-fms quinasa

Info

Publication number
UY34973A
UY34973A UY0001034973A UY34973A UY34973A UY 34973 A UY34973 A UY 34973A UY 0001034973 A UY0001034973 A UY 0001034973A UY 34973 A UY34973 A UY 34973A UY 34973 A UY34973 A UY 34973A
Authority
UY
Uruguay
Prior art keywords
preparation
fms
ester derivatives
quinasa
heterocyclic ester
Prior art date
Application number
UY0001034973A
Other languages
English (en)
Inventor
Jean Pierre Andre Marc Bongartz
Alfred Elisabeth Stappers
Christopher A Teleha
Koen Johan Herman Weerts
Kenneth J Wilson
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of UY34973A publication Critical patent/UY34973A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02Silicon compounds
    • C07F7/08Compounds having one or more C—Si linkages
    • C07F7/0803Compounds with Si-C or Si-Si linkages
    • C07F7/0825Preparations of compounds not comprising Si-Si or Si-cyano linkages
    • C07F7/083Syntheses without formation of a Si-C bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02Silicon compounds
    • C07F7/08Compounds having one or more C—Si linkages
    • C07F7/0803Compounds with Si-C or Si-Si linkages
    • C07F7/081Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te
    • C07F7/0812Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te comprising a heterocyclic ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02Silicon compounds
    • C07F7/08Compounds having one or more C—Si linkages
    • C07F7/10Compounds having one or more C—Si linkages containing nitrogen having a Si-N linkage

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

La presente invención se dirige a un proceso para la preparación de derivados de éster heterocíclico de la Fórmula I, en donde A1, SEM y W1 son como se definen en la presente descripción. Los compuestos son útiles como productos intermedios en la síntesis de derivados útiles como inhibidores de proteína tirosina, más particularmente, inhibidores de c-fms quinasa.
UY0001034973A 2012-08-07 2013-08-07 Proceso para la preparación de derivados de éster heterocíclicos inhibidores de c-fms quinasa UY34973A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201261680412P 2012-08-07 2012-08-07

Publications (1)

Publication Number Publication Date
UY34973A true UY34973A (es) 2014-02-28

Family

ID=48985861

Family Applications (1)

Application Number Title Priority Date Filing Date
UY0001034973A UY34973A (es) 2012-08-07 2013-08-07 Proceso para la preparación de derivados de éster heterocíclicos inhibidores de c-fms quinasa

Country Status (13)

Country Link
US (2) US9303046B2 (es)
EP (1) EP2882757B1 (es)
JP (1) JP6359537B2 (es)
CN (1) CN104870454B (es)
AR (1) AR092071A1 (es)
AU (1) AU2013299922B2 (es)
ES (1) ES2608628T3 (es)
HK (2) HK1209753A1 (es)
IN (1) IN2015DN00659A (es)
JO (1) JO3185B1 (es)
TW (1) TWI608009B (es)
UY (1) UY34973A (es)
WO (1) WO2014025675A1 (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2014025675A1 (en) * 2012-08-07 2014-02-13 Janssen Pharmaceutica Nv Process for the preparation of heterocyclic ester derivatives
AU2018208422B2 (en) 2017-01-10 2021-11-11 Bayer Aktiengesellschaft Heterocyclene derivatives as pest control agents

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Also Published As

Publication number Publication date
US20160168170A1 (en) 2016-06-16
AR092071A1 (es) 2015-03-18
CN104870454B (zh) 2020-03-03
TW201427986A (zh) 2014-07-16
ES2608628T3 (es) 2017-04-12
WO2014025675A1 (en) 2014-02-13
HK1210617A1 (en) 2016-04-29
US20140046072A1 (en) 2014-02-13
JO3185B1 (ar) 2018-03-08
US9303046B2 (en) 2016-04-05
HK1209753A1 (en) 2016-04-08
TWI608009B (zh) 2017-12-11
AU2013299922B2 (en) 2018-06-21
EP2882757A1 (en) 2015-06-17
AU2013299922A8 (en) 2015-03-12
AU2013299922A1 (en) 2015-02-12
EP2882757B1 (en) 2016-10-05
IN2015DN00659A (es) 2015-06-26
JP2015525796A (ja) 2015-09-07
JP6359537B2 (ja) 2018-07-18
CN104870454A (zh) 2015-08-26

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