UY33317A - Nuevos derivados de pirazol - Google Patents

Nuevos derivados de pirazol

Info

Publication number
UY33317A
UY33317A UY0001033317A UY33317A UY33317A UY 33317 A UY33317 A UY 33317A UY 0001033317 A UY0001033317 A UY 0001033317A UY 33317 A UY33317 A UY 33317A UY 33317 A UY33317 A UY 33317A
Authority
UY
Uruguay
Prior art keywords
pirazol
new derivatives
sphingosine
agonists
disease
Prior art date
Application number
UY0001033317A
Other languages
English (en)
Inventor
Eloisa Navarro Romero
Nuria Aguilar Izquierdo
Monserrat Erra Sola
Marta Carrascal Riera
Lorena Taboada Martinez
Bernat Vidal Juan
Original Assignee
Almirall Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Almirall Sa filed Critical Almirall Sa
Publication of UY33317A publication Critical patent/UY33317A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond

Abstract

La presente invención se refiere a un compuesto de fórmula (I), al procedimiento para preparar dichos compuestos y a su uso en el tratamiento de una condición patológica o enfermedad susceptible de mejorar por agonistas de los receptores de 1-fosfato de esfingosina (S1P1).
UY0001033317A 2010-05-19 2011-04-06 Nuevos derivados de pirazol UY33317A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP10382128A EP2390252A1 (en) 2010-05-19 2010-05-19 New pyrazole derivatives

Publications (1)

Publication Number Publication Date
UY33317A true UY33317A (es) 2011-10-31

Family

ID=42664897

Family Applications (1)

Application Number Title Priority Date Filing Date
UY0001033317A UY33317A (es) 2010-05-19 2011-04-06 Nuevos derivados de pirazol

Country Status (4)

Country Link
EP (1) EP2390252A1 (es)
TW (1) TW201141858A (es)
UY (1) UY33317A (es)
WO (1) WO2011144338A1 (es)

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US9034884B2 (en) 2010-11-19 2015-05-19 Incyte Corporation Heterocyclic-substituted pyrrolopyridines and pyrrolopyrimidines as JAK inhibitors
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MY195091A (en) 2013-08-07 2023-01-10 Incyte Corp Sustained Release Dosage Forms for a JAK1 Inhibitor
RU2016132324A (ru) * 2014-01-21 2018-03-01 Ф. Хоффманн-Ля Рош Аг Имидазолы для лечения и профилактики респираторной синцитиальной вирусной инфекции
WO2015184305A1 (en) 2014-05-30 2015-12-03 Incyte Corporation TREATMENT OF CHRONIC NEUTROPHILIC LEUKEMIA (CNL) AND ATYPICAL CHRONIC MYELOID LEUKEMIA (aCML) BY INHIBITORS OF JAK1
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KR20180036415A (ko) 2016-09-30 2018-04-09 재단법인 한국파스퇴르연구소 신규 헤테로아릴 화합물, 이의 거울상 이성질체, 부분 입체 이성질체 또는 약학적으로 허용가능한 염, 및 이를 유효성분으로 함유하는 항바이러스용 조성물
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TW202220651A (zh) * 2020-09-28 2022-06-01 南韓商Ｌｇ化學股份有限公司 神經鞘胺醇－１－磷酸受體促效劑的用途
WO2022065939A1 (ko) * 2020-09-28 2022-03-31 주식회사 엘지화학 스핑고신-1-인산 수용체 효능제의 용도
WO2022080812A1 (ko) * 2020-10-13 2022-04-21 주식회사 엘지화학 스핑고신-1-인산 수용체 효능제 합성을 위한 중간체의 제조 방법
KR20220142377A (ko) * 2021-04-14 2022-10-21 주식회사 엘지화학 입도가 조절된 스핑고신-1-인산 수용체 효능제를 포함하는 약제학적 조성물
CN117120038A (zh) * 2021-04-14 2023-11-24 株式会社Lg化学 包含鞘氨醇-1-磷酸受体激动剂的固体制剂的制备方法
WO2022220596A1 (ko) * 2021-04-14 2022-10-20 주식회사 엘지화학 습식과립법에 의한 스핑고신-1-인산 수용체 효능제를 포함하는 경구용 고형 제제의 제조 방법
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Also Published As

Publication number Publication date
TW201141858A (en) 2011-12-01
WO2011144338A1 (en) 2011-11-24
EP2390252A1 (en) 2011-11-30

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Effective date: 20130802