UY33079A - Derivados de difenil -pirazolopiridinas, su preparación y su aplicación en terapeutica - Google Patents
Derivados de difenil -pirazolopiridinas, su preparación y su aplicación en terapeuticaInfo
- Publication number
- UY33079A UY33079A UY33079A UY33079A UY33079A UY 33079 A UY33079 A UY 33079A UY 33079 A UY33079 A UY 33079A UY 33079 A UY33079 A UY 33079A UY 33079 A UY33079 A UY 33079A
- Authority
- UY
- Uruguay
- Prior art keywords
- pirazolopiridinas
- difenil
- therapeutics
- derivatives
- preparation
- Prior art date
Links
- 239000003814 drug Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Physical Education & Sports Medicine (AREA)
- Rheumatology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Psychology (AREA)
- Addiction (AREA)
- Hospice & Palliative Care (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0958651A FR2953520B1 (fr) | 2009-12-04 | 2009-12-04 | Derives de diphenyl-pyrazolopyridines, leur preparation et leur application en therapeutique |
Publications (1)
Publication Number | Publication Date |
---|---|
UY33079A true UY33079A (es) | 2011-06-01 |
Family
ID=42111360
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
UY33079A UY33079A (es) | 2009-12-04 | 2010-12-03 | Derivados de difenil -pirazolopiridinas, su preparación y su aplicación en terapeutica |
Country Status (24)
Country | Link |
---|---|
US (1) | US8680096B2 (es) |
EP (1) | EP2507238B1 (es) |
JP (1) | JP5738310B2 (es) |
KR (1) | KR101696959B1 (es) |
CN (1) | CN102762559B (es) |
AR (1) | AR079250A1 (es) |
AU (1) | AU2010326429B2 (es) |
BR (1) | BR112012013511A2 (es) |
CA (1) | CA2782704C (es) |
CL (1) | CL2012001461A1 (es) |
CO (1) | CO6551713A2 (es) |
EA (1) | EA020652B1 (es) |
FR (1) | FR2953520B1 (es) |
HK (1) | HK1169984A1 (es) |
IL (1) | IL220060A (es) |
JO (1) | JO3098B1 (es) |
MA (1) | MA33893B1 (es) |
MX (1) | MX2012006421A (es) |
MY (1) | MY157676A (es) |
NZ (1) | NZ600368A (es) |
SG (1) | SG181138A1 (es) |
TW (1) | TWI481606B (es) |
UY (1) | UY33079A (es) |
WO (1) | WO2011067544A1 (es) |
Families Citing this family (15)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2950345B1 (fr) * | 2009-09-18 | 2011-09-23 | Sanofi Aventis | Derives acetyleniques de 5-phenyl-pyrazolopyridine, leur preparation et leur application en therapeutique |
FR2950344B1 (fr) * | 2009-09-18 | 2011-11-25 | Sanofi Aventis | Derives de 5-phenyl-pyrazolopyridine, leur preparation et leur aplication en therapeutique. |
WO2018098499A1 (en) | 2016-11-28 | 2018-05-31 | Praxis Precision Medicines, Inc. | Compounds and their methods of use |
US11261188B2 (en) | 2016-11-28 | 2022-03-01 | Praxis Precision Medicines, Inc. | Fused heteroaryl compounds, and methods thereof for treating diseases, disorders, and conditions relating to aberrant function of a sodium channel |
WO2018098500A1 (en) * | 2016-11-28 | 2018-05-31 | Praxis Precision Medicines, Inc. | Compounds and their methods of use |
EP3551616A1 (de) * | 2016-12-08 | 2019-10-16 | Bayer CropScience Aktiengesellschaft | Verfahren zur herstellung von 5-(1-phenyl-1h-pyrazol-4-yl)-nicotinamid-derivaten und ähnlicher verbindungen ohne isolierung oder aufreinigung der phenylhydrazin-zwischenstufe |
US11492345B2 (en) | 2017-02-13 | 2022-11-08 | Praxis Precision Medicines, Inc. | Compounds and their methods of use |
US11731966B2 (en) | 2017-04-04 | 2023-08-22 | Praxis Precision Medicines, Inc. | Compounds and their methods of use |
US11278535B2 (en) | 2017-08-15 | 2022-03-22 | Praxis Precision Medicines, Inc. | Compounds and their methods of use |
CN117756800A (zh) | 2018-05-30 | 2024-03-26 | 普拉克西斯精密药物股份有限公司 | 离子通道调节剂 |
US11773099B2 (en) | 2019-05-28 | 2023-10-03 | Praxis Precision Medicines, Inc. | Compounds and their methods of use |
US11505554B2 (en) | 2019-05-31 | 2022-11-22 | Praxis Precision Medicines, Inc. | Substituted pyridines as ion channel modulators |
US11279700B2 (en) | 2019-05-31 | 2022-03-22 | Praxis Precision Medicines, Inc. | Ion channel modulators |
US11767325B2 (en) | 2019-11-26 | 2023-09-26 | Praxis Precision Medicines, Inc. | Substituted [1,2,4]triazolo[4,3-a]pyrazines as ion channel modulators |
CN111138325B (zh) * | 2019-12-20 | 2021-11-30 | 台州学院 | 一种(Z)-β-磺酰基烯胺类化合物的制备方法 |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP2001139575A (ja) * | 1999-11-15 | 2001-05-22 | Fujisawa Pharmaceut Co Ltd | 新規ピラゾロピリジン誘導体 |
FR2906250B1 (fr) * | 2006-09-22 | 2008-10-31 | Sanofi Aventis Sa | Derives de 2-aryl-6phenyl-imidazo(1,2-a) pyridines, leur preparation et leur application en therapeutique |
CA2672213C (en) * | 2006-12-22 | 2016-02-16 | Astex Therapeutics Limited | Bicyclic amine derivatives as protein tyrosine kinase inhibitors |
FR2928923B1 (fr) * | 2008-03-21 | 2010-04-23 | Sanofi Aventis | Derives polysubstitues de 2-heteroaryl-6-phenyl-imidazo °1,2-a!pyridines, leur preparation et leur application en therapeutiques |
FR2928924B1 (fr) * | 2008-03-21 | 2010-04-23 | Sanofi Aventis | Derives polysubstitues de 6-heteroaryle-imidazo°1,2-a! pyridines, leur preparation et leur application en therapeutique |
FR2928921B1 (fr) * | 2008-03-21 | 2010-04-23 | Sanofi Aventis | Derives polysubstitues de 2-aryl-6-phenyl-imidazo°1,2-a!pyridines, leur preparation et leur application en therapeutique |
US8198449B2 (en) * | 2008-09-11 | 2012-06-12 | Bristol-Myers Squibb Company | Compounds for the treatment of hepatitis C |
FR2950344B1 (fr) * | 2009-09-18 | 2011-11-25 | Sanofi Aventis | Derives de 5-phenyl-pyrazolopyridine, leur preparation et leur aplication en therapeutique. |
-
2009
- 2009-12-04 FR FR0958651A patent/FR2953520B1/fr not_active Expired - Fee Related
-
2010
- 2010-12-02 JO JOP/2010/0430A patent/JO3098B1/ar active
- 2010-12-03 EA EA201290520A patent/EA020652B1/ru not_active IP Right Cessation
- 2010-12-03 UY UY33079A patent/UY33079A/es not_active Application Discontinuation
- 2010-12-03 KR KR1020127017287A patent/KR101696959B1/ko active IP Right Grant
- 2010-12-03 BR BR112012013511A patent/BR112012013511A2/pt not_active IP Right Cessation
- 2010-12-03 MX MX2012006421A patent/MX2012006421A/es active IP Right Grant
- 2010-12-03 MA MA35024A patent/MA33893B1/fr unknown
- 2010-12-03 MY MYPI2012002449A patent/MY157676A/en unknown
- 2010-12-03 SG SG2012039749A patent/SG181138A1/en unknown
- 2010-12-03 CA CA2782704A patent/CA2782704C/fr not_active Expired - Fee Related
- 2010-12-03 CN CN201080062600.0A patent/CN102762559B/zh not_active Expired - Fee Related
- 2010-12-03 JP JP2012541567A patent/JP5738310B2/ja not_active Expired - Fee Related
- 2010-12-03 WO PCT/FR2010/052605 patent/WO2011067544A1/fr active Application Filing
- 2010-12-03 EP EP10801625.4A patent/EP2507238B1/fr not_active Not-in-force
- 2010-12-03 NZ NZ600368A patent/NZ600368A/en not_active IP Right Cessation
- 2010-12-03 AR ARP100104462A patent/AR079250A1/es unknown
- 2010-12-03 AU AU2010326429A patent/AU2010326429B2/en not_active Ceased
- 2010-12-03 TW TW099142230A patent/TWI481606B/zh not_active IP Right Cessation
- 2010-12-03 US US13/513,497 patent/US8680096B2/en not_active Expired - Fee Related
-
2012
- 2012-05-30 IL IL220060A patent/IL220060A/en not_active IP Right Cessation
- 2012-06-04 CO CO12093017A patent/CO6551713A2/es active IP Right Grant
- 2012-06-04 CL CL2012001461A patent/CL2012001461A1/es unknown
- 2012-10-22 HK HK12110468.8A patent/HK1169984A1/xx not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
CN102762559B (zh) | 2014-11-05 |
JP5738310B2 (ja) | 2015-06-24 |
MY157676A (en) | 2016-07-15 |
EP2507238B1 (fr) | 2013-07-31 |
SG181138A1 (en) | 2012-07-30 |
US20120245164A1 (en) | 2012-09-27 |
CN102762559A (zh) | 2012-10-31 |
TW201129564A (en) | 2011-09-01 |
MX2012006421A (es) | 2012-10-09 |
IL220060A (en) | 2015-05-31 |
BR112012013511A2 (pt) | 2016-06-07 |
JO3098B1 (ar) | 2017-03-15 |
CA2782704A1 (fr) | 2011-06-09 |
JP2013512884A (ja) | 2013-04-18 |
MA33893B1 (fr) | 2013-01-02 |
EP2507238A1 (fr) | 2012-10-10 |
NZ600368A (en) | 2013-12-20 |
CL2012001461A1 (es) | 2012-10-12 |
HK1169984A1 (en) | 2013-02-15 |
WO2011067544A1 (fr) | 2011-06-09 |
US8680096B2 (en) | 2014-03-25 |
AU2010326429A1 (en) | 2012-06-21 |
KR20120103672A (ko) | 2012-09-19 |
FR2953520A1 (fr) | 2011-06-10 |
KR101696959B1 (ko) | 2017-01-16 |
AR079250A1 (es) | 2012-01-04 |
AU2010326429B2 (en) | 2016-07-14 |
CA2782704C (fr) | 2018-01-02 |
EA201290520A1 (ru) | 2013-01-30 |
FR2953520B1 (fr) | 2011-11-25 |
TWI481606B (zh) | 2015-04-21 |
CO6551713A2 (es) | 2012-10-31 |
EA020652B1 (ru) | 2014-12-30 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
109 | Application deemed to be withdrawn |
Effective date: 20181127 |