UY30729A1 - Derivados de pirrol, su preparacion y su utilizacion en terapéutica - Google Patents

Derivados de pirrol, su preparacion y su utilizacion en terapéutica

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Publication number
UY30729A1
UY30729A1 UY30729A UY30729A UY30729A1 UY 30729 A1 UY30729 A1 UY 30729A1 UY 30729 A UY30729 A UY 30729A UY 30729 A UY30729 A UY 30729A UY 30729 A1 UY30729 A1 UY 30729A1
Authority
UY
Uruguay
Prior art keywords
therapeutics
derivatives
preparation
pirrol
diphenylpyrrol
Prior art date
Application number
UY30729A
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English (en)
Inventor
Francis Barth
Christian Congy
Laurent Hortala
Rinaldi Carmona Murilelle
Original Assignee
Sanofi Aventis
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Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38521242&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UY30729(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Sanofi Aventis filed Critical Sanofi Aventis
Publication of UY30729A1 publication Critical patent/UY30729A1/es

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    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
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Abstract

La presente invencion se refiere a derivados de 4,5-difenipirrol-2-carboxamida, compuestos que responden a la formula (I): en la que los sustituyentes y radicales son tales como se especifican en la memoria descriptiva y en las reivindicaciones: Se refiere además a procedimiento de preparacion y aplicacion en terapéutica para el tratamiento o la prevencion de enfermedades en las que están implicados los receptores CB1
UY30729A 2006-11-20 2007-11-20 Derivados de pirrol, su preparacion y su utilizacion en terapéutica UY30729A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0610202A FR2908766B1 (fr) 2006-11-20 2006-11-20 Derives de pyrrole,leur preparation et leur utilisation en therapeutique.

Publications (1)

Publication Number Publication Date
UY30729A1 true UY30729A1 (es) 2008-07-03

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UY30729A UY30729A1 (es) 2006-11-20 2007-11-20 Derivados de pirrol, su preparacion y su utilizacion en terapéutica

Country Status (27)

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US (1) US8044072B2 (es)
EP (1) EP2094656B1 (es)
JP (1) JP5210320B2 (es)
KR (1) KR20090080992A (es)
CN (1) CN101535250A (es)
AR (1) AR064596A1 (es)
AT (1) ATE520654T1 (es)
AU (1) AU2007330651A1 (es)
BR (1) BRPI0718962A2 (es)
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FR2930939B1 (fr) * 2008-05-09 2010-07-30 Sanofi Aventis Derives de pyrrole, leur preparation et leur application en therapeutique
FR2930940B1 (fr) * 2008-05-09 2011-02-11 Sanofi Aventis Derives de pyrrole, leur preparation et leur application en therapeutique
CN102964304B (zh) * 2012-09-28 2015-06-17 苏州大学 含吡唑烷酮结构的手性氨基氰化物的制备方法
US10526320B2 (en) 2016-07-12 2020-01-07 Guangdong Raynovent Biotech Co., Ltd. Pyrrolidine derivatives as PPAR agonists
CN111356676B (zh) 2017-12-21 2022-09-27 广东众生睿创生物科技有限公司 作为ppar激动剂的吡咯烷衍生物的无定形及其制备方法
WO2020113094A1 (en) 2018-11-30 2020-06-04 Nuvation Bio Inc. Pyrrole and pyrazole compounds and methods of use thereof

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EP1756066B1 (en) * 2004-05-28 2008-08-20 Solvay Pharmaceuticals B.V. Tetrasubstituted imidazole derivatives as cannabinoid cb1 receptor modulators with a high cb1/cb2 receptor subtype selectivity
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CR10772A (es) 2009-07-23
FR2908766B1 (fr) 2009-01-09
TW200829565A (en) 2008-07-16
US20090281116A1 (en) 2009-11-12
CN101535250A (zh) 2009-09-16
BRPI0718962A2 (pt) 2013-12-17
WO2008068423A2 (fr) 2008-06-12
MX2009005366A (es) 2009-06-08
EP2094656B1 (fr) 2011-08-17
JP5210320B2 (ja) 2013-06-12
ATE520654T1 (de) 2011-09-15
DOP2009000105A (es) 2009-05-31
CA2669996A1 (fr) 2008-06-12
AR064596A1 (es) 2009-04-15
MA30996B1 (fr) 2009-12-01
CL2007003318A1 (es) 2008-07-04
JP2010510198A (ja) 2010-04-02
EP2094656A2 (fr) 2009-09-02
ECSP099339A (es) 2009-06-30
NO20092066L (no) 2009-08-11
FR2908766A1 (fr) 2008-05-23
ZA200903865B (en) 2010-08-25
IL198481A0 (en) 2010-02-17
EA200970497A1 (ru) 2009-10-30
WO2008068423A3 (fr) 2008-07-31
US8044072B2 (en) 2011-10-25
KR20090080992A (ko) 2009-07-27
AU2007330651A1 (en) 2008-06-12
PE20081495A1 (es) 2008-12-31
SV2009003265A (es) 2010-02-05
TN2009000166A1 (fr) 2010-10-18

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