FR2930939B1 - Derives de pyrrole, leur preparation et leur application en therapeutique - Google Patents
Derives de pyrrole, leur preparation et leur application en therapeutiqueInfo
- Publication number
- FR2930939B1 FR2930939B1 FR0802552A FR0802552A FR2930939B1 FR 2930939 B1 FR2930939 B1 FR 2930939B1 FR 0802552 A FR0802552 A FR 0802552A FR 0802552 A FR0802552 A FR 0802552A FR 2930939 B1 FR2930939 B1 FR 2930939B1
- Authority
- FR
- France
- Prior art keywords
- preparation
- therapeutic application
- pyrrole derivatives
- pyrrole
- derivatives
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
- KAESVJOAVNADME-UHFFFAOYSA-N Pyrrole Chemical class C=1C=CNC=1 KAESVJOAVNADME-UHFFFAOYSA-N 0.000 title 1
- 230000001225 therapeutic effect Effects 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/12—Antidiarrhoeals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
Priority Applications (10)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0802552A FR2930939B1 (fr) | 2008-05-09 | 2008-05-09 | Derives de pyrrole, leur preparation et leur application en therapeutique |
PE2009000633A PE20091830A1 (es) | 2008-05-09 | 2009-05-07 | Derivados de pirrol como antagonistas de los receptores cannabinoides cb1 |
EP09750013A EP2283007A2 (fr) | 2008-05-09 | 2009-05-07 | Dérivés de 1,5-diphénylepyrrole-3-carboxamide, leur preparation et leur utilisation comme antagonistes des récepteurs cb1 des cannabinoïdes |
UY0001031814A UY31814A (es) | 2008-05-09 | 2009-05-07 | Derivados de pirrol, su preparación y su aplicación en terapéutica |
TW098115181A TW200951120A (en) | 2008-05-09 | 2009-05-07 | Pyrrole derivatives, their preparation and their therapeutic application |
JP2011507967A JP5611193B2 (ja) | 2008-05-09 | 2009-05-07 | 1,5−ジフェニルピロール−3−カルボキサミド誘導体、この調製、およびこのカンナビノイドcb1受容体拮抗薬としての利用 |
PA20098825701A PA8825701A1 (es) | 2008-05-09 | 2009-05-07 | Derivados de piro, su preparacion y su aplicacion en terapeutica |
PCT/FR2009/000535 WO2009141532A2 (fr) | 2008-05-09 | 2009-05-07 | Derives de pyrrole, leur preparation et leur application en therapeutique |
ARP090101646A AR071688A1 (es) | 2008-05-09 | 2009-05-07 | Derivados de pirrol, su preparacion y su aplicacion en terapeutica |
US12/942,780 US8680102B2 (en) | 2008-05-09 | 2010-11-09 | Pyrrole derivatives, their preparation and their therapeutic application |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0802552A FR2930939B1 (fr) | 2008-05-09 | 2008-05-09 | Derives de pyrrole, leur preparation et leur application en therapeutique |
Publications (2)
Publication Number | Publication Date |
---|---|
FR2930939A1 FR2930939A1 (fr) | 2009-11-13 |
FR2930939B1 true FR2930939B1 (fr) | 2010-07-30 |
Family
ID=39930534
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FR0802552A Expired - Fee Related FR2930939B1 (fr) | 2008-05-09 | 2008-05-09 | Derives de pyrrole, leur preparation et leur application en therapeutique |
Country Status (10)
Country | Link |
---|---|
US (1) | US8680102B2 (fr) |
EP (1) | EP2283007A2 (fr) |
JP (1) | JP5611193B2 (fr) |
AR (1) | AR071688A1 (fr) |
FR (1) | FR2930939B1 (fr) |
PA (1) | PA8825701A1 (fr) |
PE (1) | PE20091830A1 (fr) |
TW (1) | TW200951120A (fr) |
UY (1) | UY31814A (fr) |
WO (1) | WO2009141532A2 (fr) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP2017531011A (ja) | 2014-10-16 | 2017-10-19 | ザ ボード オブ トラスティーズ オブ ザ リーランド スタンフォード ジュニア ユニバーシティ | 麻酔のための新規の方法、化合物および組成物 |
ES2910071T3 (es) | 2018-03-08 | 2022-05-11 | Incyte Corp | Compuestos de aminopirazina diol como inhibidores de PI3K-Y |
WO2020010003A1 (fr) | 2018-07-02 | 2020-01-09 | Incyte Corporation | DÉRIVÉS D'AMINOPYRAZINE UTILISÉS EN TANT QU'INHIBITEURS DE PI3K-γ |
WO2023089612A1 (fr) * | 2021-11-19 | 2023-05-25 | Yissum Research Development Company Of The Hebrew University Of Jerusalem Ltd. | Antagonistes périphériques du récepteur cb1 pour le traitement de symptômes du bas appareil urinaire (luts) |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US7271176B2 (en) | 1998-09-04 | 2007-09-18 | Millennium Pharmaceuticals, Inc. | Chemokine receptor antagonists and methods of use thereof |
JP2005532982A (ja) * | 2001-09-24 | 2005-11-04 | バイエル・フアーマシユーチカルズ・コーポレーシヨン | 肥満の処置のためのピロール誘導体の製造及び使用 |
GB0230088D0 (en) * | 2002-12-24 | 2003-01-29 | Astrazeneca Ab | Therapeutic agents |
GB0403780D0 (en) * | 2004-02-20 | 2004-03-24 | Astrazeneca Ab | Therapeutic agents |
FR2874012B1 (fr) | 2004-08-09 | 2008-08-22 | Sanofi Synthelabo | Derives de pyrrole, leur preparation et leur utlisation en therapeutique |
FR2882054B1 (fr) * | 2005-02-17 | 2007-04-13 | Sanofi Aventis Sa | Derives de 1,5-diarylpyrrole, leur preparation et leur application en therapeutique |
FR2887548B1 (fr) * | 2005-06-27 | 2007-09-21 | Sanofi Aventis Sa | Derives de 4,5-diarylpyrrole, leur preparation et leur application en therapeutique |
WO2008002974A1 (fr) * | 2006-06-27 | 2008-01-03 | Abbott Laboratories | Dérivés de pyrrole et leurs procédés d'utilisation |
FR2908766B1 (fr) * | 2006-11-20 | 2009-01-09 | Sanofi Aventis Sa | Derives de pyrrole,leur preparation et leur utilisation en therapeutique. |
-
2008
- 2008-05-09 FR FR0802552A patent/FR2930939B1/fr not_active Expired - Fee Related
-
2009
- 2009-05-07 JP JP2011507967A patent/JP5611193B2/ja not_active Expired - Fee Related
- 2009-05-07 AR ARP090101646A patent/AR071688A1/es unknown
- 2009-05-07 UY UY0001031814A patent/UY31814A/es not_active Application Discontinuation
- 2009-05-07 TW TW098115181A patent/TW200951120A/zh unknown
- 2009-05-07 WO PCT/FR2009/000535 patent/WO2009141532A2/fr active Application Filing
- 2009-05-07 PA PA20098825701A patent/PA8825701A1/es unknown
- 2009-05-07 EP EP09750013A patent/EP2283007A2/fr not_active Withdrawn
- 2009-05-07 PE PE2009000633A patent/PE20091830A1/es not_active Application Discontinuation
-
2010
- 2010-11-09 US US12/942,780 patent/US8680102B2/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
JP5611193B2 (ja) | 2014-10-22 |
PA8825701A1 (es) | 2009-12-16 |
AR071688A1 (es) | 2010-07-07 |
JP2011519905A (ja) | 2011-07-14 |
US8680102B2 (en) | 2014-03-25 |
EP2283007A2 (fr) | 2011-02-16 |
PE20091830A1 (es) | 2009-12-21 |
UY31814A (es) | 2010-01-05 |
FR2930939A1 (fr) | 2009-11-13 |
WO2009141532A3 (fr) | 2010-02-11 |
TW200951120A (en) | 2009-12-16 |
WO2009141532A2 (fr) | 2009-11-26 |
US20110152320A1 (en) | 2011-06-23 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
FR2933700B1 (fr) | Derives de pyridino-pyridinones, leur preparation et leur application en therapeutique | |
FR2945534B1 (fr) | DERIVES DE CYCLOPENTAL[c]PYRROLE-2-CARBOXYLATES, LEUR PREPARATION ET LEUR APPLICATION EN THERAPEUTIQUE | |
FR2911604B1 (fr) | Derives de n-(heteroaryl-1h-indole-2-carboxamides, leur preparation et leur application en therapeutique | |
FR2953520B1 (fr) | Derives de diphenyl-pyrazolopyridines, leur preparation et leur application en therapeutique | |
FR2949470B1 (fr) | Derives anticancereux, leur preparation et leur application therapeutique | |
FR2915198B1 (fr) | Derives de triazolopyridine-carboxamides et triazolopyridine -carboxamides, leur preparation et leur application en therapeutique. | |
FR2926556B1 (fr) | Derives de carboxamides n-azabicycliques, leur preparation et leur application en therapeutique | |
FR2915199B1 (fr) | Derives de triazolopyridine-carboxamides et triazolopyrimidine-carboxamides, leur preparation et leur application en therapeutique. | |
FR2910473B1 (fr) | Derives de n-(amino-heteroaryl)-1h-pyrrolopyridine-2- carboxamides, leur preparation et leur application en therapeutique. | |
FR2952934B1 (fr) | Derives de pyridino-pyridinones, leur preparation et leur application en therapeutique | |
FR2903985B1 (fr) | Derives de n-(amino-heteroaryl)-1h-indole-2-carboxamides, leur preparation et leur application en therapeutique | |
FR2943669B1 (fr) | Derives de nicotinamide,leur preparation et leur application en therapeutique | |
FR2891825B1 (fr) | Derives de la 1-amino-isoquinoline, leur preparation et leur application en therapeutique | |
FR2917413B1 (fr) | Derives de 7-alkynyl-1,8-naphthyridones, leur preparation et leur application en therapeutique | |
FR2927625B1 (fr) | Nouveaux derives de 3-aminoalkyl-1,3-dihydro-2h-indol-2-one, leur preparation et leur application en therapeutique | |
FR2915197B1 (fr) | Derives de triazolopyridine-carboxamides, leur preparation et leur application therapeutique. | |
FR2930249B1 (fr) | Nouveaux derives de 3-aminoalkyl-1,3-dihydro-2h-indol-2-one, leur preparation et leur application en therapeutique. | |
FR2947546B1 (fr) | Derives de pyrazoles, leur preparation et leur application en therapeutique | |
FR2940284B1 (fr) | Derives de 6-cycloamino-2,3-di-pyridinyl-imidazo°1,2-b!- pyridazine,leur preparation et leur application en therapeutique | |
FR2896246B1 (fr) | Derives de pyrido-pyrimidone, leur preparation, leur application en therapeutique. | |
FR2892416B1 (fr) | Derives de 6-heteroarylpyridoindolone, leur preparation et leur application en therapeutique | |
FR2925901B1 (fr) | DERIVES DE N-HETEROCYCLIQUE-IMIDAZO°1,2-a!PYRIDINE-2- CARBOXAMIDES, LEUR PREPARATION ET LEUR APPLICATION EN THERAPEUTIQUE | |
FR2932481B1 (fr) | Derives de 4-{2-°4-phenyl-3,6-dihydro-2h-pyridin-1-yl!-2- oxo-alkyl}-1-piperazin-2-one, leur preparation et leur application en therapeutique. | |
FR2930939B1 (fr) | Derives de pyrrole, leur preparation et leur application en therapeutique | |
FR2911605B1 (fr) | Derives de pyrrolopyridine-2-carbowamides, leur preparation et leur application en therapeutique |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
PLFP | Fee payment |
Year of fee payment: 8 |
|
ST | Notification of lapse |
Effective date: 20170131 |