UY31548A1 - Derivados de azetidinas, su preparacion y su aplicacion en terapéutica - Google Patents

Derivados de azetidinas, su preparacion y su aplicacion en terapéutica

Info

Publication number
UY31548A1
UY31548A1 UY31548A UY31548A UY31548A1 UY 31548 A1 UY31548 A1 UY 31548A1 UY 31548 A UY31548 A UY 31548A UY 31548 A UY31548 A UY 31548A UY 31548 A1 UY31548 A1 UY 31548A1
Authority
UY
Uruguay
Prior art keywords
azetidines
preparation
therapeutics
derivatives
application
Prior art date
Application number
UY31548A
Other languages
English (en)
Inventor
Sabuco Jean-Francois
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=40935338&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UY31548(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from FR0708830A external-priority patent/FR2925051B1/fr
Priority claimed from FR0802492A external-priority patent/FR2930941B1/fr
Application filed filed Critical
Publication of UY31548A1 publication Critical patent/UY31548A1/es

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    • C—CHEMISTRY; METALLURGY
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/04—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
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    • C—CHEMISTRY; METALLURGY
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

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  • Health & Medical Sciences (AREA)
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  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Biomedical Technology (AREA)
  • Neurology (AREA)
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  • Diabetes (AREA)
  • Cardiology (AREA)
  • Hematology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Psychiatry (AREA)
  • Addiction (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Pulmonology (AREA)
  • Obesity (AREA)
  • Rheumatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Endocrinology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Immunology (AREA)
  • Pain & Pain Management (AREA)
  • Hospice & Palliative Care (AREA)
  • Reproductive Health (AREA)
  • Ophthalmology & Optometry (AREA)
  • Vascular Medicine (AREA)
  • Child & Adolescent Psychology (AREA)

Abstract

Se divulgan compuestos derivados de azetidinas que responden a la formula (I), en el estado de base o de sal de adicion o una base, en la que los sustituyentes e índices son tales como los especificados en la memoria descriptiva y en las reivindicaciones. Se divulgan los procedimientos de preparacion de (I), sus intermediarios y la aplicaciones ene. tratamiento o la prevencion de enfermedades que implican a los receptores de los cannabinoides CB1.
UY31548A 2007-12-18 2008-12-18 Derivados de azetidinas, su preparacion y su aplicacion en terapéutica UY31548A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0708830A FR2925051B1 (fr) 2007-12-18 2007-12-18 Derives d'azetidines,leur preparation et leur application en therapeutique
FR0802492A FR2930941B1 (fr) 2008-05-06 2008-05-06 Derives d'azetidines, leur preparation et leur application en therapeutique

Publications (1)

Publication Number Publication Date
UY31548A1 true UY31548A1 (es) 2009-08-03

Family

ID=40935338

Family Applications (1)

Application Number Title Priority Date Filing Date
UY31548A UY31548A1 (es) 2007-12-18 2008-12-18 Derivados de azetidinas, su preparacion y su aplicacion en terapéutica

Country Status (27)

Country Link
US (2) US8445478B2 (es)
EP (1) EP2234966B1 (es)
JP (1) JP5460614B2 (es)
KR (1) KR20100098563A (es)
CN (1) CN101945852B (es)
AR (1) AR069700A1 (es)
AU (1) AU2008351943B2 (es)
BR (1) BRPI0822054A2 (es)
CA (1) CA2709863A1 (es)
CL (1) CL2008003780A1 (es)
CO (1) CO6290755A2 (es)
CY (1) CY1114991T1 (es)
DK (1) DK2234966T3 (es)
EA (1) EA019315B1 (es)
ES (1) ES2439258T3 (es)
HK (1) HK1152038A1 (es)
HR (1) HRP20131168T1 (es)
IL (1) IL206420A (es)
MA (1) MA32019B1 (es)
PA (1) PA8808101A1 (es)
PE (1) PE20091270A1 (es)
PL (1) PL2234966T3 (es)
PT (1) PT2234966E (es)
SI (1) SI2234966T1 (es)
TW (1) TW200930360A (es)
UY (1) UY31548A1 (es)
WO (1) WO2009106708A2 (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UA103319C2 (en) 2008-05-06 2013-10-10 Глаксосмитклайн Ллк Thiazole- and oxazole-benzene sulfonamide compounds
FR2946650B1 (fr) * 2009-06-16 2011-08-19 Sanofi Aventis Esters derives d'azetidines, leur preparation et leur application en therapeutique.
EP2611788B1 (en) 2010-09-03 2017-04-12 University of Florida Research Foundation, Incorporated Nicotine compounds and analogs thereof, synthetic methods of making compounds, and methods of use
GB201321601D0 (en) * 2013-12-06 2014-01-22 Canbex Therapeutics Ltd Modulator
US11003343B2 (en) * 2014-01-06 2021-05-11 Lett.rs LLC Electronic personal signature generation and distribution for personal communication

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2399791A1 (en) * 2000-02-11 2001-08-16 Bristol-Myers Squibb Company Cannabinoid receptor modulators, their processes of preparation, and use of cannabinoid receptor modulators in treating respiratory and non-respiratory diseases
FR2805817B1 (fr) * 2000-03-03 2002-04-26 Aventis Pharma Sa Compositions pharmaceutiques contenant des derives d'azetidine, les nouveaux derives d'azetidine et leur preparation
FR2814678B1 (fr) * 2000-10-04 2002-12-20 Aventis Pharma Sa Association d'un antagoniste du recepteur cb1 et de sibutramine, les compositions pharmaceutiques les contenant et leur utilisation pour la traitement de l'obesite
RU2304580C2 (ru) * 2002-07-29 2007-08-20 Ф.Хоффманн-Ля Рош Аг Новые бензодиоксолы
ATE453620T1 (de) * 2003-05-01 2010-01-15 Vernalis Res Ltd Azetidincarboxamid-derivate zur verwendung zur behandlung von cb1-rezeptor-vermittelten krankheiten
PE20071092A1 (es) * 2005-12-08 2007-12-10 Aventis Pharma Inc Composicion farmaceutica que comprende un antagonista de cb1 y un agente antisicotico
EP1993560B1 (en) * 2006-03-10 2011-12-28 Jenrin Discovery Cannabinoid receptor antagonists/inverse agonists useful for treating obesity

Also Published As

Publication number Publication date
HRP20131168T1 (hr) 2014-01-03
PT2234966E (pt) 2013-12-19
PE20091270A1 (es) 2009-09-23
MA32019B1 (fr) 2011-01-03
JP5460614B2 (ja) 2014-04-02
EA019315B1 (ru) 2014-02-28
IL206420A0 (en) 2010-12-30
CY1114991T1 (el) 2016-12-14
PL2234966T3 (pl) 2014-02-28
JP2011506583A (ja) 2011-03-03
US8445478B2 (en) 2013-05-21
ES2439258T3 (es) 2014-01-22
CN101945852A (zh) 2011-01-12
DK2234966T3 (da) 2014-01-06
KR20100098563A (ko) 2010-09-07
EP2234966A2 (fr) 2010-10-06
SI2234966T1 (sl) 2014-01-31
WO2009106708A2 (fr) 2009-09-03
PA8808101A1 (es) 2009-07-23
AU2008351943A1 (en) 2009-09-03
HK1152038A1 (en) 2012-02-17
AR069700A1 (es) 2010-02-10
CA2709863A1 (fr) 2009-09-03
CO6290755A2 (es) 2011-06-20
IL206420A (en) 2015-01-29
US20110009377A1 (en) 2011-01-13
WO2009106708A3 (fr) 2009-12-30
TW200930360A (en) 2009-07-16
AU2008351943B2 (en) 2013-12-19
CL2008003780A1 (es) 2010-04-09
US20130237513A1 (en) 2013-09-12
EA201070758A1 (ru) 2011-02-28
EP2234966B1 (fr) 2013-09-11
CN101945852B (zh) 2014-05-07
BRPI0822054A2 (pt) 2015-06-23

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