EA201270256A1 - Производные т1-замещенного 5-фтор-2-оксопиримидинон-1 (2h) -карбоксамида - Google Patents

Производные т1-замещенного 5-фтор-2-оксопиримидинон-1 (2h) -карбоксамида

Info

Publication number
EA201270256A1
EA201270256A1 EA201270256A EA201270256A EA201270256A1 EA 201270256 A1 EA201270256 A1 EA 201270256A1 EA 201270256 A EA201270256 A EA 201270256A EA 201270256 A EA201270256 A EA 201270256A EA 201270256 A1 EA201270256 A1 EA 201270256A1
Authority
EA
Eurasian Patent Office
Prior art keywords
derivatives
substituted
oxopyrimidinon
karboxamid
fluor
Prior art date
Application number
EA201270256A
Other languages
English (en)
Other versions
EA020910B1 (ru
Inventor
Тимоти Бебель
Кристи Брайан
Бет Лорсбах
Тимоти Мартин
В. Оуэн
Марк Побанс
Скотт Торнберг
Джеффри Вебстер
Чэнлинь Яо
Original Assignee
ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43535294&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=EA201270256(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи filed Critical ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи
Publication of EA201270256A1 publication Critical patent/EA201270256A1/ru
Publication of EA020910B1 publication Critical patent/EA020910B1/ru

Links

Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/28—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N<
    • A01N47/38—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N< containing the group >N—CO—N< where at least one nitrogen atom is part of a heterocyclic ring; Thio analogues thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Abstract

Изобретение относится к N1-замещенным 5-фтор-2-оксопиримидинон-1-(2Н)-карбоксамидам и их производным, и к применению этих соединений в качестве фунгицидов.
EA201270256A 2009-08-07 2010-08-05 Производные n1-замещенного 5-фтор-2-оксопиримидинон-1(2h)-карбоксамида и их применение в качестве фунгицидов EA020910B1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US23224509P 2009-08-07 2009-08-07
PCT/US2010/044588 WO2011017545A1 (en) 2009-08-07 2010-08-05 N1-substituted-5-fluoro-2-oxopyrimidinone-1(2h)-carboxamide derivatives

Publications (2)

Publication Number Publication Date
EA201270256A1 true EA201270256A1 (ru) 2012-07-30
EA020910B1 EA020910B1 (ru) 2015-02-27

Family

ID=43535294

Family Applications (1)

Application Number Title Priority Date Filing Date
EA201270256A EA020910B1 (ru) 2009-08-07 2010-08-05 Производные n1-замещенного 5-фтор-2-оксопиримидинон-1(2h)-карбоксамида и их применение в качестве фунгицидов

Country Status (27)

Country Link
US (2) US8552020B2 (ru)
EP (1) EP2461686B1 (ru)
JP (1) JP5735510B2 (ru)
KR (1) KR101792284B1 (ru)
CN (1) CN102497781B (ru)
BR (1) BR112012002757B1 (ru)
CA (1) CA2769656C (ru)
CL (1) CL2012000312A1 (ru)
CO (1) CO6491115A2 (ru)
CR (1) CR20120032A (ru)
DK (1) DK2461686T3 (ru)
EA (1) EA020910B1 (ru)
EC (1) ECSP12011652A (ru)
ES (1) ES2552097T3 (ru)
HK (1) HK1171915A1 (ru)
HU (1) HUE027390T2 (ru)
IL (1) IL217950A (ru)
IN (1) IN2012DN00369A (ru)
MX (1) MX2012001617A (ru)
NI (1) NI201200021A (ru)
NZ (1) NZ597483A (ru)
PE (1) PE20120692A1 (ru)
PL (1) PL2461686T3 (ru)
PT (1) PT2461686E (ru)
UA (1) UA107671C2 (ru)
WO (1) WO2011017545A1 (ru)
ZA (1) ZA201200813B (ru)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UA107671C2 (en) * 2009-08-07 2015-02-10 Dow Agrosciences Llc N1-substityted-5-fluoro-2-oxopyrimidinone-1(2h)-carboxamide derivatives
WO2011017547A1 (en) * 2009-08-07 2011-02-10 Dow Agrosciences Llc N1-sulfonyl-5-fluoropyrimidinone derivatives
BR112012002677A2 (pt) 2009-08-07 2021-03-09 Dow Agrosciences Llc Moléculas de heteroaril-n-aril carbamatos, e composição pesticida
JP6324994B2 (ja) * 2012-12-28 2018-05-16 アダマ・マクテシム・リミテッド Ｎ−（置換）−５−フルオロ−４−イミノ−３−メチル−２−オキソ−３，４−ジヒドロピリミジン−１（２ｈ）−カルボキシレート誘導体
KR20150100869A (ko) * 2012-12-28 2015-09-02 다우 아그로사이언시즈 엘엘씨 N-(치환된)-5-플루오로-4-이미노-3-메틸-2-옥소-3,4-디히드로피리미딘-1(2h)-카르복스아미드 유도체
JP6336480B2 (ja) * 2012-12-28 2018-06-06 アダマ・マクテシム・リミテッド １−（置換ベンゾイル）−５−フルオロ−４−イミノ−３−メチル−３，４−ジヒドロピリミジン−２（１ｈ）−オンの誘導体
AU2013370494B2 (en) 2012-12-31 2017-08-17 Adama Makhteshim Ltd. 3-alkyl-5-fluoro-4-substituted-imino-3,4-dihydropyrimidin-2(1H)-one derivatives as fungicides
BR112016015157A2 (pt) 2013-12-31 2017-08-08 Adama Makhteshim Ltd Misturas fungicidas sinergísticas para controle de fungos em cereais
AU2014373959B2 (en) 2013-12-31 2017-10-26 Adama Makhteshim Ltd. 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1- (arylsulfonyl)-3,4-dihydropyrimidin-2(1H)-one and processes for their preparation
JP2020527563A (ja) 2017-07-17 2020-09-10 アダマ・マクテシム・リミテッド ５−フルオロ−４−イミノ−３−メチル−１−トシル−３，４−ジヒドロピリミジン−２−オンの多形体

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US3368938A (en) 1966-01-13 1968-02-13 Hoffmann La Roche Controlling fungi with 5-fluorocytosine
US3868373A (en) 1970-01-27 1975-02-25 Hoffmann La Roche 4-Amino-5-fluoro-2-tri(lower alkyl) silyloxypyrimidines
CH579057A5 (ru) 1973-09-07 1976-08-31 Hoffmann La Roche
FR2530636A1 (fr) 1982-07-23 1984-01-27 Rhone Poulenc Agrochimie Nouveaux derives de la tetrahydro-2,3,6,7 5h-thiazolo (3,2-a) pyrimidine, leur preparation et leur utilisation comme herbicides
GR80171B (en) 1983-08-29 1985-01-02 Ciba Geigy Ag N-(2-nitrophenyl)-4-aminopyrimidine derivatives process for the preparation thereof and use
JPS60123486A (ja) 1983-12-09 1985-07-02 Asahi Glass Co Ltd フルオロブラストサイジンｓおよびその製法
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JP3109012B2 (ja) 1992-06-18 2000-11-13 クミアイ化学工業株式会社 チアゾロ［５，４−ｄ］ピリミジン誘導体及び農園芸用殺菌剤
JP3217191B2 (ja) 1992-07-16 2001-10-09 ビーエーエスエフ アクチェンゲゼルシャフト ヘテロ芳香族化合物およびこれを含有する植物保護剤
JP4010563B2 (ja) * 1995-07-05 2007-11-21 イー・アイ・デユポン・ドウ・ヌムール・アンド・カンパニー 殺菌・殺カビ性のピリミジノン類
PT888359E (pt) 1996-03-11 2002-10-31 Syngenta Participations Ag Derivados de pirimidin-4-ona como pesticida
HRP970239B1 (en) 1997-05-09 2004-04-30 Inst Ru Er Bouekovic Process for the preparation of sulfonyl-pyrimidine derivatives with antitumor activity
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WO2003018051A1 (en) 2001-08-27 2003-03-06 Vic Jira Anti-fungal composition
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EP2044086A2 (en) 2006-06-30 2009-04-08 Janssen Pharmaceutica N.V. Thiazolopyrimidine modulators of trpv1
EP2562165A1 (en) 2008-01-22 2013-02-27 Dow AgroSciences LLC 5-fluoro pyrimidine derivatives as fungicides
MX2011001091A (es) * 2008-08-01 2011-03-15 Dow Agrosciences Llc Uso de 5-fluorocitosina como un fungicida.
USRE46144E1 (en) * 2009-01-23 2016-09-13 Purdue Pharmaceutical Products L.P. Hydroxamic acid derivatives
UA107671C2 (en) * 2009-08-07 2015-02-10 Dow Agrosciences Llc N1-substityted-5-fluoro-2-oxopyrimidinone-1(2h)-carboxamide derivatives
WO2011017547A1 (en) 2009-08-07 2011-02-10 Dow Agrosciences Llc N1-sulfonyl-5-fluoropyrimidinone derivatives

Also Published As

Publication number Publication date
CN102497781B (zh) 2014-12-10
KR101792284B1 (ko) 2017-10-31
PT2461686E (pt) 2015-11-18
PL2461686T3 (pl) 2016-04-29
MX2012001617A (es) 2012-04-11
EA020910B1 (ru) 2015-02-27
AU2010279409A1 (en) 2012-02-02
JP2013501727A (ja) 2013-01-17
US9000002B2 (en) 2015-04-07
HUE027390T2 (en) 2016-10-28
EP2461686A4 (en) 2013-02-13
BR112012002757B1 (pt) 2020-10-06
HK1171915A1 (en) 2013-04-12
ECSP12011652A (es) 2012-03-30
DK2461686T3 (en) 2016-01-18
CA2769656A1 (en) 2011-02-10
WO2011017545A1 (en) 2011-02-10
CN102497781A (zh) 2012-06-13
CA2769656C (en) 2018-05-15
ES2552097T3 (es) 2015-11-25
KR20120052281A (ko) 2012-05-23
ZA201200813B (en) 2013-05-29
UA107671C2 (en) 2015-02-10
EP2461686A1 (en) 2012-06-13
US20140011824A1 (en) 2014-01-09
EP2461686B1 (en) 2015-10-07
BR112012002757A2 (pt) 2019-12-17
US20110034492A1 (en) 2011-02-10
US8552020B2 (en) 2013-10-08
JP5735510B2 (ja) 2015-06-17
PE20120692A1 (es) 2012-06-08
CL2012000312A1 (es) 2012-10-05
NI201200021A (es) 2012-05-22
IL217950A0 (en) 2012-03-29
CO6491115A2 (es) 2012-07-31
IL217950A (en) 2015-04-30
NZ597483A (en) 2014-02-28
CR20120032A (es) 2012-03-22
IN2012DN00369A (ru) 2015-08-21

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Legal Events

Date Code Title Description
MM4A Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s)

Designated state(s): AM AZ KG MD TJ TM

PC4A Registration of transfer of a eurasian patent by assignment
MM4A Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s)

Designated state(s): BY KZ RU