PT2461686E - Derivados de 5-fluoro-2-oxopirimidinona-1(2h)-carboxamida substituídos em n1 - Google Patents

Derivados de 5-fluoro-2-oxopirimidinona-1(2h)-carboxamida substituídos em n1 Download PDF

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Publication number
PT2461686E
PT2461686E PT108071754T PT10807175T PT2461686E PT 2461686 E PT2461686 E PT 2461686E PT 108071754 T PT108071754 T PT 108071754T PT 10807175 T PT10807175 T PT 10807175T PT 2461686 E PT2461686 E PT 2461686E
Authority
PT
Portugal
Prior art keywords
oxopyrimidinone
fluoro
substituted
carboxamide derivatives
carboxamide
Prior art date
Application number
PT108071754T
Other languages
English (en)
Portuguese (pt)
Inventor
Chenglin Yao
Timothy Boebel
Kristy Bryan
Beth Lorsbach
Timothy Martin
W Owen
Mark Pobanz
Scott Thornburgh
Jeffery Webster
Original Assignee
Dow Agrosciences Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43535294&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PT2461686(E) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Dow Agrosciences Llc filed Critical Dow Agrosciences Llc
Publication of PT2461686E publication Critical patent/PT2461686E/pt

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Classifications

    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/28Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N<
    • A01N47/38Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N< containing the group >N—CO—N< where at least one nitrogen atom is part of a heterocyclic ring; Thio analogues thereof
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
PT108071754T 2009-08-07 2010-08-05 Derivados de 5-fluoro-2-oxopirimidinona-1(2h)-carboxamida substituídos em n1 PT2461686E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US23224509P 2009-08-07 2009-08-07

Publications (1)

Publication Number Publication Date
PT2461686E true PT2461686E (pt) 2015-11-18

Family

ID=43535294

Family Applications (1)

Application Number Title Priority Date Filing Date
PT108071754T PT2461686E (pt) 2009-08-07 2010-08-05 Derivados de 5-fluoro-2-oxopirimidinona-1(2h)-carboxamida substituídos em n1

Country Status (27)

Country Link
US (2) US8552020B2 (ru)
EP (1) EP2461686B1 (ru)
JP (1) JP5735510B2 (ru)
KR (1) KR101792284B1 (ru)
CN (1) CN102497781B (ru)
BR (1) BR112012002757B1 (ru)
CA (1) CA2769656C (ru)
CL (1) CL2012000312A1 (ru)
CO (1) CO6491115A2 (ru)
CR (1) CR20120032A (ru)
DK (1) DK2461686T3 (ru)
EA (1) EA020910B1 (ru)
EC (1) ECSP12011652A (ru)
ES (1) ES2552097T3 (ru)
HK (1) HK1171915A1 (ru)
HU (1) HUE027390T2 (ru)
IL (1) IL217950A (ru)
IN (1) IN2012DN00369A (ru)
MX (1) MX2012001617A (ru)
NI (1) NI201200021A (ru)
NZ (1) NZ597483A (ru)
PE (1) PE20120692A1 (ru)
PL (1) PL2461686T3 (ru)
PT (1) PT2461686E (ru)
UA (1) UA107671C2 (ru)
WO (1) WO2011017545A1 (ru)
ZA (1) ZA201200813B (ru)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9006259B2 (en) * 2009-08-07 2015-04-14 Dow Agrosciences Llc N1-sulfonyl-5-fluoropyrimidinone derivatives
UA107671C2 (en) * 2009-08-07 2015-02-10 Dow Agrosciences Llc N1-substityted-5-fluoro-2-oxopyrimidinone-1(2h)-carboxamide derivatives
NZ597597A (en) 2009-08-07 2014-01-31 Dow Agrosciences Llc Pesticidal compositions containing heteroaryl-n-aryl carbamate compounds
MX2015008443A (es) * 2012-12-28 2015-09-23 Dow Agrosciences Llc Derivados de 1-(benzoilo-sustituido) -5-fluoro-4-imino-3-metil-3, 4-dihidropirimidin-2 (1h)-ona.
HUE047711T2 (hu) * 2012-12-28 2020-05-28 Adama Makhteshim Ltd N-(szubsztituált)-5-fluor-4-imino-3-metil-2-oxo-3,4-dihidropirimidin-1(2H)-karboxilát származékok
KR20150100869A (ko) * 2012-12-28 2015-09-02 다우 아그로사이언시즈 엘엘씨 N-(치환된)-5-플루오로-4-이미노-3-메틸-2-옥소-3,4-디히드로피리미딘-1(2h)-카르복스아미드 유도체
NZ708981A (en) 2012-12-31 2020-01-31 Adama Makhteshim Ltd 3-alkyl-5-fluoro-4-substituted-imino-3,4-dihydropyrimidin-2(1h)-one derivatives as fungicides
CN115380909A (zh) 2013-12-31 2022-11-25 阿达玛马克西姆股份有限公司 用防治谷类中真菌的协同杀真菌混合物
EP3862347A1 (en) 2013-12-31 2021-08-11 Adama Makhteshim Ltd. Processes for their preparation of 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1-(arylsulfonyl)- 3,4-dihydropyrimidin-2(1h)-one
IL271950B2 (en) 2017-07-17 2024-06-01 Adama Makhteshim Ltd Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-4,3-dihydropyrimidin-2-one

Family Cites Families (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3309359A (en) 1965-10-22 1967-03-14 Hoffmann La Roche N-mono-acyl-5-fluorocytosine derivatives and process
US3368938A (en) 1966-01-13 1968-02-13 Hoffmann La Roche Controlling fungi with 5-fluorocytosine
US3868373A (en) 1970-01-27 1975-02-25 Hoffmann La Roche 4-Amino-5-fluoro-2-tri(lower alkyl) silyloxypyrimidines
CH579057A5 (ru) 1973-09-07 1976-08-31 Hoffmann La Roche
FR2530636A1 (fr) 1982-07-23 1984-01-27 Rhone Poulenc Agrochimie Nouveaux derives de la tetrahydro-2,3,6,7 5h-thiazolo (3,2-a) pyrimidine, leur preparation et leur utilisation comme herbicides
EP0139613A1 (de) 1983-08-29 1985-05-02 Ciba-Geigy Ag N-(2-Nitrophenyl)-4-aminopyrimidin-Derivate, deren Herstellung und Verwendung
JPS60123486A (ja) 1983-12-09 1985-07-02 Asahi Glass Co Ltd フルオロブラストサイジンsおよびその製法
US4845081A (en) 1984-10-18 1989-07-04 University Of Florida Aminomethyl derivatives of biologically active substances, and enhanced delivery thereof across topical membranes
ATE109776T1 (de) 1988-03-09 1994-08-15 Ciba Geigy Ag Mittel zum schutz von pflanzen gegen krankheiten.
DE3821711A1 (de) 1988-06-28 1990-02-08 Bayer Ag Thiazolopyrimidin-derivate, verfahren zu ihrer herstellung und ihre verwendung als schaedlingsbekaempfungsmittel
JP3109012B2 (ja) 1992-06-18 2000-11-13 クミアイ化学工業株式会社 チアゾロ[5,4−d]ピリミジン誘導体及び農園芸用殺菌剤
JP3217191B2 (ja) 1992-07-16 2001-10-09 ビーエーエスエフ アクチェンゲゼルシャフト ヘテロ芳香族化合物およびこれを含有する植物保護剤
MX9800136A (es) * 1995-07-05 1998-03-29 Du Pont Pirimidinonas fungicidas.
AU716248B2 (en) 1996-03-11 2000-02-24 Novartis Ag Pyrimidin-4-one derivatives as pesticide
HRP970239B1 (en) 1997-05-09 2004-04-30 Inst Ru Er Bouekovic Process for the preparation of sulfonyl-pyrimidine derivatives with antitumor activity
GT199900185A (es) 1998-11-06 2001-04-18 Novedosa pirimidin-4-enamina como fungicida.
WO2003018051A1 (en) 2001-08-27 2003-03-06 Vic Jira Anti-fungal composition
JPWO2005095419A1 (ja) 2004-04-01 2008-02-21 武田薬品工業株式会社 チアゾロピリミジン誘導体
US20080004253A1 (en) 2006-06-30 2008-01-03 Bryan James Branstetter Thiazolopyrimidine modulators of TRPV1
DK2562166T3 (en) 2008-01-22 2015-11-23 Dow Agrosciences Llc 5-fluoro-pyrimidine derivatives as fungicides
CN104521977A (zh) * 2008-08-01 2015-04-22 陶氏益农公司 5-氟胞嘧啶作为杀真菌剂的用途
EP2389375B1 (en) * 2009-01-23 2015-05-20 Euro-Celtique S.A. Hydroxamic acid derivatives
UA107671C2 (en) * 2009-08-07 2015-02-10 Dow Agrosciences Llc N1-substityted-5-fluoro-2-oxopyrimidinone-1(2h)-carboxamide derivatives
US9006259B2 (en) 2009-08-07 2015-04-14 Dow Agrosciences Llc N1-sulfonyl-5-fluoropyrimidinone derivatives

Also Published As

Publication number Publication date
EP2461686A4 (en) 2013-02-13
BR112012002757B1 (pt) 2020-10-06
IN2012DN00369A (ru) 2015-08-21
KR101792284B1 (ko) 2017-10-31
NI201200021A (es) 2012-05-22
MX2012001617A (es) 2012-04-11
CN102497781B (zh) 2014-12-10
ES2552097T3 (es) 2015-11-25
AU2010279409A1 (en) 2012-02-02
US20110034492A1 (en) 2011-02-10
EA201270256A1 (ru) 2012-07-30
IL217950A (en) 2015-04-30
JP5735510B2 (ja) 2015-06-17
CL2012000312A1 (es) 2012-10-05
US20140011824A1 (en) 2014-01-09
US8552020B2 (en) 2013-10-08
ZA201200813B (en) 2013-05-29
CA2769656A1 (en) 2011-02-10
HUE027390T2 (en) 2016-10-28
HK1171915A1 (en) 2013-04-12
CA2769656C (en) 2018-05-15
KR20120052281A (ko) 2012-05-23
EP2461686A1 (en) 2012-06-13
CR20120032A (es) 2012-03-22
PL2461686T3 (pl) 2016-04-29
NZ597483A (en) 2014-02-28
DK2461686T3 (en) 2016-01-18
IL217950A0 (en) 2012-03-29
JP2013501727A (ja) 2013-01-17
EA020910B1 (ru) 2015-02-27
CO6491115A2 (es) 2012-07-31
ECSP12011652A (es) 2012-03-30
WO2011017545A1 (en) 2011-02-10
US9000002B2 (en) 2015-04-07
BR112012002757A2 (pt) 2019-12-17
EP2461686B1 (en) 2015-10-07
PE20120692A1 (es) 2012-06-08
UA107671C2 (en) 2015-02-10
CN102497781A (zh) 2012-06-13

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