MX2009005366A - Derivados de pirrol, su preparacion y su utilizacion en terapeutica. - Google Patents

Derivados de pirrol, su preparacion y su utilizacion en terapeutica.

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Publication number
MX2009005366A
MX2009005366A MX2009005366A MX2009005366A MX2009005366A MX 2009005366 A MX2009005366 A MX 2009005366A MX 2009005366 A MX2009005366 A MX 2009005366A MX 2009005366 A MX2009005366 A MX 2009005366A MX 2009005366 A MX2009005366 A MX 2009005366A
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MX
Mexico
Prior art keywords
substituted
group
therapy
preparation
0pyrrol
Prior art date
Application number
MX2009005366A
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English (en)
Inventor
Francis Barth
Murielle Rinaldi-Carmona
Christian Congy
Laurent Hortala
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Sanofi Aventis
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Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38521242&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX2009005366(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Sanofi Aventis filed Critical Sanofi Aventis
Publication of MX2009005366A publication Critical patent/MX2009005366A/es

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    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
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Abstract

La invención se refiere a compuestos que tienen la fórmula (I), en donde A representa; un grupo alquileno (C1-C6) sustituido o no sustituido, un grupo de Fórmula (II) que tiene m= 0, 1 o 2 y p=0 o 1; R1 representa hidrógeno o un alquilo (C1-C2); R2 representa un grupo alquilo (C3-C10) sustituido o no sustituido, un radical carbocíclico no aromático (C3-C12) sustituido o no sustituido, un radical heterocíclico sustituido o no sustituido, un grupo alquileno (C1-C3) sustituido, un grupo NR10 R11; R9 representa un grupo funcional o un radical heterocíclico. Método de preparación y uso en terapia.
MX2009005366A 2006-11-20 2007-11-19 Derivados de pirrol, su preparacion y su utilizacion en terapeutica. MX2009005366A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0610202A FR2908766B1 (fr) 2006-11-20 2006-11-20 Derives de pyrrole,leur preparation et leur utilisation en therapeutique.
PCT/FR2007/001888 WO2008068423A2 (fr) 2006-11-20 2007-11-19 Derives de pyrrole, leur preparation et leur utilisation en therapeutique.

Publications (1)

Publication Number Publication Date
MX2009005366A true MX2009005366A (es) 2009-06-08

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MX2009005366A MX2009005366A (es) 2006-11-20 2007-11-19 Derivados de pirrol, su preparacion y su utilizacion en terapeutica.

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US (1) US8044072B2 (es)
EP (1) EP2094656B1 (es)
JP (1) JP5210320B2 (es)
KR (1) KR20090080992A (es)
CN (1) CN101535250A (es)
AR (1) AR064596A1 (es)
AT (1) ATE520654T1 (es)
AU (1) AU2007330651A1 (es)
BR (1) BRPI0718962A2 (es)
CA (1) CA2669996A1 (es)
CL (1) CL2007003318A1 (es)
CR (1) CR10772A (es)
DO (1) DOP2009000105A (es)
EA (1) EA200970497A1 (es)
EC (1) ECSP099339A (es)
FR (1) FR2908766B1 (es)
IL (1) IL198481A0 (es)
MA (1) MA30996B1 (es)
MX (1) MX2009005366A (es)
NO (1) NO20092066L (es)
PE (1) PE20081495A1 (es)
SV (1) SV2009003265A (es)
TN (1) TN2009000166A1 (es)
TW (1) TW200829565A (es)
UY (1) UY30729A1 (es)
WO (1) WO2008068423A2 (es)
ZA (1) ZA200903865B (es)

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Publication number Priority date Publication date Assignee Title
FR2930940B1 (fr) * 2008-05-09 2011-02-11 Sanofi Aventis Derives de pyrrole, leur preparation et leur application en therapeutique
FR2930939B1 (fr) * 2008-05-09 2010-07-30 Sanofi Aventis Derives de pyrrole, leur preparation et leur application en therapeutique
CN102964304B (zh) * 2012-09-28 2015-06-17 苏州大学 含吡唑烷酮结构的手性氨基氰化物的制备方法
KR102200264B1 (ko) * 2016-07-12 2021-01-11 광둥 레이노벤트 바이오테크 컴퍼니 리미티드 Ppar 작용제인 피롤리딘 유도체
US11396493B2 (en) 2017-12-21 2022-07-26 Guangdong Raynovent Biotech Co., Ltd. Amorphous pyrrolidine derivative as PPAR agonist and preparation method thereof
WO2020113094A1 (en) 2018-11-30 2020-06-04 Nuvation Bio Inc. Pyrrole and pyrazole compounds and methods of use thereof

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AU2002319627A1 (en) * 2001-07-20 2003-03-03 Merck And Co., Inc. Substituted imidazoles as cannabinoid receptor modulators
FR2856683A1 (fr) * 2003-06-25 2004-12-31 Sanofi Synthelabo Derives de 4-cyanopyrazole-3-carboxamide, leur preparation et leur application en therapeutique
BRPI0510564A (pt) * 2004-05-28 2007-11-20 Solvay Pharm Bv compostos e tautÈmeros, estereoisÈmeros, e sais farmacologicamente aceitáveis dos mesmos, composições farmacêuticas, método para preparar composições farmacêuticas, e, uso de um composto
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FR2881744B1 (fr) * 2005-02-09 2007-04-27 Sanofi Aventis Sa Derives de n-[(4,5-diphenyl-2-thienyl)methyl]amine, leur preparation et leur application en therapeutique
AU2006215567B2 (en) * 2005-02-16 2011-05-12 Abbott Healthcare Products B.V. 1H-imidazole derivatives as cannabinoid CB2 receptor modulators

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WO2008068423A3 (fr) 2008-07-31
NO20092066L (no) 2009-08-11
US8044072B2 (en) 2011-10-25
AR064596A1 (es) 2009-04-15
CR10772A (es) 2009-07-23
ZA200903865B (en) 2010-08-25
FR2908766A1 (fr) 2008-05-23
IL198481A0 (en) 2010-02-17
AU2007330651A1 (en) 2008-06-12
TN2009000166A1 (fr) 2010-10-18
EA200970497A1 (ru) 2009-10-30
UY30729A1 (es) 2008-07-03
EP2094656A2 (fr) 2009-09-02
CA2669996A1 (fr) 2008-06-12
MA30996B1 (fr) 2009-12-01
FR2908766B1 (fr) 2009-01-09
ATE520654T1 (de) 2011-09-15
TW200829565A (en) 2008-07-16
KR20090080992A (ko) 2009-07-27
US20090281116A1 (en) 2009-11-12
BRPI0718962A2 (pt) 2013-12-17
SV2009003265A (es) 2010-02-05
DOP2009000105A (es) 2009-05-31
CL2007003318A1 (es) 2008-07-04
JP5210320B2 (ja) 2013-06-12
JP2010510198A (ja) 2010-04-02
EP2094656B1 (fr) 2011-08-17
ECSP099339A (es) 2009-06-30

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