UY30232A1 - Nuevas formas cristalinas - Google Patents

Nuevas formas cristalinas

Info

Publication number
UY30232A1
UY30232A1 UY30232A UY30232A UY30232A1 UY 30232 A1 UY30232 A1 UY 30232A1 UY 30232 A UY30232 A UY 30232A UY 30232 A UY30232 A UY 30232A UY 30232 A1 UY30232 A1 UY 30232A1
Authority
UY
Uruguay
Prior art keywords
salt
acid
crystal forms
new crystal
phosphoric
Prior art date
Application number
UY30232A
Other languages
English (en)
Inventor
Martin Bohlin
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of UY30232A1 publication Critical patent/UY30232A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/06—Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • C07D235/08—Radicals containing only hydrogen and carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4184—1,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system

Abstract

Una sal de un compuestos N-(2-terc-butil-1-((4,4-difluorociclohexil)metil)-1h-benzimidazol-5-il)etanosulfonamida, que es una sal de ácido etanosulfonico, una sal de ácido sulfurico, una sal de ácido etanodisulfonico, una sal de ácido clorhídrico, una sal de ácido bromhídrico, una sal de ácido fosforico, una sal de ácido acético, una sal de ácido fosforico, una sal de ácido acético, una sal de ácido fumárico, una sal de ácido maleico, una sal de ácido tartárico, una sal de ácido cítrico, una sal de ácido metanosulfonico, o una sal de ácido p-toluensulfonico de dicho compuesto.
UY30232A 2006-03-23 2007-03-22 Nuevas formas cristalinas UY30232A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US78532606P 2006-03-23 2006-03-23

Publications (1)

Publication Number Publication Date
UY30232A1 true UY30232A1 (es) 2007-10-31

Family

ID=38522716

Family Applications (1)

Application Number Title Priority Date Filing Date
UY30232A UY30232A1 (es) 2006-03-23 2007-03-22 Nuevas formas cristalinas

Country Status (18)

Country Link
US (2) US7566788B2 (es)
EP (1) EP2001856A4 (es)
JP (1) JP2009530373A (es)
KR (1) KR20080105098A (es)
CN (1) CN101454293A (es)
AR (1) AR060065A1 (es)
AU (1) AU2007227811A1 (es)
BR (1) BRPI0709631A2 (es)
CA (1) CA2648829A1 (es)
EC (1) ECSP088714A (es)
IL (1) IL193671A0 (es)
MX (1) MX2008012015A (es)
NO (1) NO20084353L (es)
RU (1) RU2008136556A (es)
TW (1) TW200745049A (es)
UY (1) UY30232A1 (es)
WO (1) WO2007108754A1 (es)
ZA (1) ZA200807598B (es)

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* Cited by examiner, † Cited by third party
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SE0302573D0 (sv) 2003-09-26 2003-09-26 Astrazeneca Ab Benzimidazole derivatives, compositions containing them, preparation thereof and uses thereof
BRPI0515897A (pt) * 2004-09-24 2008-08-12 Astrazeneca Ab composto, uso do mesmo, composição farmacêutica, e, método para a terapia de dor em um animal de sangue quente, e para a preparação de um composto
TW200808769A (en) * 2006-04-18 2008-02-16 Astrazeneca Ab Therapeutic compounds
US20110086853A1 (en) * 2009-10-08 2011-04-14 William Brown Therapeutic Compounds
CN101758337B (zh) 2009-12-03 2012-02-15 湖南阿斯达生化科技有限公司 一种助焊剂用非卤素活性剂
GB202019335D0 (en) * 2020-12-09 2021-01-20 Artelo Biosciences Ltd Pharmaceutical compositions

Family Cites Families (43)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1604908A (en) 1965-06-24 1971-05-15 Substd benzimidazoles - with anthelmintic,fungicidal activity and some with antiviral and antibacterial activity
FR5354M (es) 1965-09-10 1967-09-11
US5387600A (en) 1992-07-30 1995-02-07 Fuji Photo Film Co., Ltd. Treating arteriosclerosis using benzimidazole compositions
DE4237617A1 (de) 1992-11-06 1994-05-11 Bayer Ag Verwendung von substituierten Benzimidazolen
DE4237597A1 (de) 1992-11-06 1994-05-11 Bayer Ag Substituierte Benzimidazole
DE4237557A1 (de) 1992-11-06 1994-05-11 Bayer Ag Substituierte Benzimidazole
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US6720317B1 (en) 1999-09-17 2004-04-13 Millennium Pharmaceuticals, Inc. Inhibitors of factor Xa
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Also Published As

Publication number Publication date
WO2007108754A1 (en) 2007-09-27
AR060065A1 (es) 2008-05-21
MX2008012015A (es) 2008-10-01
US7566788B2 (en) 2009-07-28
EP2001856A4 (en) 2011-02-16
TW200745049A (en) 2007-12-16
AU2007227811A1 (en) 2007-09-27
CN101454293A (zh) 2009-06-10
US20100022610A1 (en) 2010-01-28
KR20080105098A (ko) 2008-12-03
BRPI0709631A2 (pt) 2011-07-19
CA2648829A1 (en) 2007-09-27
EP2001856A1 (en) 2008-12-17
US20070225346A1 (en) 2007-09-27
NO20084353L (no) 2008-10-16
JP2009530373A (ja) 2009-08-27
ECSP088714A (es) 2008-10-31
IL193671A0 (en) 2009-05-04
RU2008136556A (ru) 2010-04-27
ZA200807598B (en) 2010-02-24

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