UY27809A1 - Inhibidores de la transcriptasa inversa no nucleosidos - Google Patents

Inhibidores de la transcriptasa inversa no nucleosidos

Info

Publication number
UY27809A1
UY27809A1 UY27809A UY27809A UY27809A1 UY 27809 A1 UY27809 A1 UY 27809A1 UY 27809 A UY27809 A UY 27809A UY 27809 A UY27809 A UY 27809A UY 27809 A1 UY27809 A1 UY 27809A1
Authority
UY
Uruguay
Prior art keywords
nucleosid
inverse
inhibitors
transcript inhibitors
inverse transcript
Prior art date
Application number
UY27809A
Other languages
English (en)
Inventor
Bruno Simoneau
Serge Landry
Eric Malenfant
Julie Naud
Jeffrey O'meara
Bounkham Thavonekham
Christiane Yoakim
Original Assignee
Boehringer Ingelheim Int
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Int filed Critical Boehringer Ingelheim Int
Publication of UY27809A1 publication Critical patent/UY27809A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Virology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Molecular Biology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • AIDS & HIV (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Compuestos representados por la fórmula I: o una sal o un pro fármaco se proporcionan como inhibidores de transcriptasa inversa de VIH.
UY27809A 2002-05-16 2003-05-15 Inhibidores de la transcriptasa inversa no nucleosidos UY27809A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US38088602P 2002-05-16 2002-05-16

Publications (1)

Publication Number Publication Date
UY27809A1 true UY27809A1 (es) 2003-12-31

Family

ID=29550032

Family Applications (1)

Application Number Title Priority Date Filing Date
UY27809A UY27809A1 (es) 2002-05-16 2003-05-15 Inhibidores de la transcriptasa inversa no nucleosidos

Country Status (29)

Country Link
US (1) US6806265B2 (es)
EP (1) EP1506195B1 (es)
JP (1) JP4230448B2 (es)
KR (1) KR20050008716A (es)
CN (1) CN1318421C (es)
AR (1) AR040027A1 (es)
AT (1) ATE412653T1 (es)
AU (1) AU2003229186A1 (es)
BR (1) BR0310033A (es)
CA (1) CA2485916C (es)
DE (1) DE60324418D1 (es)
EA (1) EA009178B1 (es)
EC (1) ECSP045432A (es)
ES (1) ES2315492T3 (es)
HK (1) HK1080849A1 (es)
HR (1) HRP20041065A2 (es)
IL (1) IL163753A0 (es)
MX (1) MXPA04010409A (es)
MY (1) MY134646A (es)
NO (1) NO20044104L (es)
NZ (1) NZ536736A (es)
PE (1) PE20040365A1 (es)
PL (1) PL371663A1 (es)
RS (1) RS98004A (es)
TW (1) TW200404071A (es)
UA (1) UA79285C2 (es)
UY (1) UY27809A1 (es)
WO (1) WO2003097644A2 (es)
ZA (1) ZA200406912B (es)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2004087169A1 (en) * 2003-03-27 2004-10-14 Boehringer Ingelheim International Gmbh Antiviral combination of nevirapine and a further antiretroviral compound
US7348338B2 (en) 2003-07-17 2008-03-25 Plexxikon, Inc. PPAR active compounds
JP4845730B2 (ja) 2003-07-17 2011-12-28 プレキシコン,インコーポレーテッド Ppar活性化合物
DE102004051277A1 (de) * 2004-10-21 2006-04-27 Merck Patent Gmbh Heterocyclische Carbonylverbindungen
US7531568B2 (en) * 2004-11-30 2009-05-12 Plexxikon, Inc. PPAR active compounds
US20070072904A1 (en) * 2005-09-07 2007-03-29 Jack Lin PPAR active compounds
TW200800872A (en) * 2005-09-07 2008-01-01 Plexxikon Inc PPAR active compounds
US20080234349A1 (en) * 2005-09-07 2008-09-25 Jack Lin PPAR active compounds
US8492428B2 (en) 2005-09-20 2013-07-23 Mayo Foundation For Medical Education And Research Small-molecule botulinum toxin inhibitors
PE20090159A1 (es) * 2007-03-08 2009-02-21 Plexxikon Inc COMPUESTOS DERIVADOS DE ACIDO INDOL-PROPIONICO COMO MODULADORES PPARs
WO2016083276A1 (de) 2014-11-25 2016-06-02 Bayer Pharma Aktiengesellschaft Substituierte pyridobenzodiazepinon-derivate und ihre verwendung
CN115745910A (zh) 2017-07-21 2023-03-07 安塔比奥公司 化学化合物
MA54133B1 (fr) 2018-03-08 2022-01-31 Incyte Corp Composés d'aminopyrazine diol utilisés comme inhibiteurs de pi3k-y
WO2020010003A1 (en) 2018-07-02 2020-01-09 Incyte Corporation AMINOPYRAZINE DERIVATIVES AS PI3K-γ INHIBITORS

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5366972A (en) 1989-04-20 1994-11-22 Boehringer Ingelheim Pharmaceuticals, Inc. 5,11-dihydro-6H-dipyrido(3,2-B:2',3'-E)(1,4)diazepines and their use in the prevention or treatment of HIV infection
US5705499A (en) * 1995-10-06 1998-01-06 Boehringer Ingelheim Pharmaceuticals, Inc. 8-arylalkyl- and 8-arylheteroalkyl-5,11-dihydro-6H-dipyrido 3,2-B:2',3'-e! 1!diazepines and their use in the treatment of HIV-1 infection
TWI270547B (en) * 2000-06-16 2007-01-11 Boehringer Ingelheim Ca Ltd Non-nucleoside reverse transcriptase inhibitors
US6716836B2 (en) 2001-03-22 2004-04-06 Boehringer Ingelheim (Canada) Ltd. Non-nucleoside reverse transcriptase inhibitors
US6673791B2 (en) 2001-07-30 2004-01-06 Boehringer Ingelheim (Canada) Ltd. Non-nucleoside reverse transcriptase inhibitors

Also Published As

Publication number Publication date
CA2485916A1 (en) 2003-11-27
HK1080849A1 (en) 2006-05-04
IL163753A0 (en) 2005-12-18
EA009178B1 (ru) 2007-12-28
ECSP045432A (es) 2005-01-03
BR0310033A (pt) 2005-02-15
EP1506195B1 (en) 2008-10-29
WO2003097644A2 (en) 2003-11-27
ATE412653T1 (de) 2008-11-15
UA79285C2 (en) 2007-06-11
TW200404071A (en) 2004-03-16
NO20044104L (no) 2004-12-01
KR20050008716A (ko) 2005-01-21
CN1318421C (zh) 2007-05-30
AU2003229186A1 (en) 2003-12-02
CN1653066A (zh) 2005-08-10
MY134646A (en) 2007-12-31
PL371663A1 (en) 2005-06-27
CA2485916C (en) 2009-12-08
WO2003097644A3 (en) 2004-02-05
MXPA04010409A (es) 2005-02-17
AR040027A1 (es) 2005-03-09
JP4230448B2 (ja) 2009-02-25
PE20040365A1 (es) 2004-07-22
EA200401482A1 (ru) 2005-06-30
DE60324418D1 (de) 2008-12-11
ZA200406912B (en) 2006-06-28
JP2005526851A (ja) 2005-09-08
NZ536736A (en) 2006-11-30
HRP20041065A2 (en) 2005-04-30
RS98004A (en) 2006-12-15
ES2315492T3 (es) 2009-04-01
US6806265B2 (en) 2004-10-19
US20040006071A1 (en) 2004-01-08
EP1506195A2 (en) 2005-02-16

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Legal Events

Date Code Title Description
109 Application deemed to be withdrawn

Effective date: 20150126