UA77650C2 - Use of serotonin reuptake inhibitor in combination with deramcyclane - Google Patents
Use of serotonin reuptake inhibitor in combination with deramcyclane Download PDFInfo
- Publication number
- UA77650C2 UA77650C2 UA2002065005A UA2002065005A UA77650C2 UA 77650 C2 UA77650 C2 UA 77650C2 UA 2002065005 A UA2002065005 A UA 2002065005A UA 2002065005 A UA2002065005 A UA 2002065005A UA 77650 C2 UA77650 C2 UA 77650C2
- Authority
- UA
- Ukraine
- Prior art keywords
- serotonin reuptake
- reuptake inhibitor
- pharmaceutical composition
- citalopram
- disorder
- Prior art date
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- A61P25/20—Hypnotics; Sedatives
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- G—PHYSICS
- G01—MEASURING; TESTING
- G01N—INVESTIGATING OR ANALYSING MATERIALS BY DETERMINING THEIR CHEMICAL OR PHYSICAL PROPERTIES
- G01N33/00—Investigating or analysing materials by specific methods not covered by groups G01N1/00 - G01N31/00
- G01N33/48—Biological material, e.g. blood, urine; Haemocytometers
- G01N33/50—Chemical analysis of biological material, e.g. blood, urine; Testing involving biospecific ligand binding methods; Immunological testing
- G01N33/94—Chemical analysis of biological material, e.g. blood, urine; Testing involving biospecific ligand binding methods; Immunological testing involving narcotics or drugs or pharmaceuticals, neurotransmitters or associated receptors
- G01N33/9406—Neurotransmitters
- G01N33/9413—Dopamine
-
- G—PHYSICS
- G01—MEASURING; TESTING
- G01N—INVESTIGATING OR ANALYSING MATERIALS BY DETERMINING THEIR CHEMICAL OR PHYSICAL PROPERTIES
- G01N2500/00—Screening for compounds of potential therapeutic value
- G01N2500/04—Screening involving studying the effect of compounds C directly on molecule A (e.g. C are potential ligands for a receptor A, or potential substrates for an enzyme A)
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- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Engineering & Computer Science (AREA)
- Epidemiology (AREA)
- Biomedical Technology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Molecular Biology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Hematology (AREA)
- General Chemical & Material Sciences (AREA)
- Urology & Nephrology (AREA)
- Immunology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- General Physics & Mathematics (AREA)
- Cell Biology (AREA)
- Pathology (AREA)
- Biochemistry (AREA)
- Analytical Chemistry (AREA)
- Physics & Mathematics (AREA)
- Food Science & Technology (AREA)
- Microbiology (AREA)
- Biotechnology (AREA)
- Psychiatry (AREA)
- Inorganic Chemistry (AREA)
- Emergency Medicine (AREA)
- Addiction (AREA)
- Child & Adolescent Psychology (AREA)
- Pain & Pain Management (AREA)
- Obesity (AREA)
- Nutrition Science (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
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US16924599P | 1999-12-06 | 1999-12-06 | |
PCT/DK2000/000671 WO2001041701A2 (en) | 1999-12-06 | 2000-12-06 | The combination of a serotonin reuptake inhibitor and a 5-ht2c antagonist, inverse agonist or partial agonist |
Publications (1)
Publication Number | Publication Date |
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UA77650C2 true UA77650C2 (en) | 2007-01-15 |
Family
ID=22614803
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
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UA2002065005A UA77650C2 (en) | 1999-12-06 | 2000-06-12 | Use of serotonin reuptake inhibitor in combination with deramcyclane |
Country Status (33)
Country | Link |
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US (4) | US20020103249A1 (de) |
EP (2) | EP1237553B1 (de) |
JP (1) | JP2003516326A (de) |
KR (1) | KR100832026B1 (de) |
CN (2) | CN1433313A (de) |
AT (1) | ATE314849T1 (de) |
AU (2) | AU1850801A (de) |
BG (1) | BG106895A (de) |
BR (1) | BR0016385A (de) |
CA (1) | CA2393470A1 (de) |
CO (1) | CO5251409A1 (de) |
CY (1) | CY1105014T1 (de) |
CZ (1) | CZ20021961A3 (de) |
DE (1) | DE60025398T2 (de) |
DK (1) | DK1237553T3 (de) |
EA (1) | EA006391B1 (de) |
ES (1) | ES2255519T3 (de) |
HR (1) | HRP20020527A2 (de) |
HU (1) | HUP0203586A3 (de) |
IL (2) | IL149994A0 (de) |
IS (1) | IS2227B (de) |
ME (1) | MEP6208A (de) |
MX (1) | MXPA02005613A (de) |
NO (1) | NO20022657L (de) |
NZ (1) | NZ545907A (de) |
PL (1) | PL356402A1 (de) |
PT (1) | PT1237553E (de) |
SK (1) | SK7962002A3 (de) |
TR (1) | TR200201512T2 (de) |
UA (1) | UA77650C2 (de) |
WO (2) | WO2001041766A1 (de) |
YU (1) | YU41902A (de) |
ZA (1) | ZA200204391B (de) |
Families Citing this family (37)
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AR021155A1 (es) * | 1999-07-08 | 2002-06-12 | Lundbeck & Co As H | Tratamiento de desordenes neuroticos |
GB0005477D0 (en) | 2000-03-07 | 2000-04-26 | Resolution Chemicals Limited | Process for the preparation of citalopram |
US6589996B2 (en) | 2000-03-17 | 2003-07-08 | Orion Corporation | Treatment of disorders relating to the serotonergic system |
US6335372B1 (en) * | 2000-11-28 | 2002-01-01 | Orion Corporation | Treatment of obsessive compulsive disorder |
US6335371B1 (en) * | 2000-11-28 | 2002-01-01 | Orion Corporation | Method for inducing cognition enhancement |
AU2002218338A1 (en) * | 2000-11-28 | 2002-06-11 | Orion Corporation | Treatment of psychiatric disorders with trimethyl-bicyclo(2.2.1)heptane derivatives |
FI20002612A0 (fi) * | 2000-11-28 | 2000-11-28 | Orion Yhtymae Oyj | Yhdistelmäterapia serotoniinivälityksen häiriöiden hoitamiseksi |
MXPA03008777A (es) * | 2001-05-01 | 2004-02-12 | Lundbeck & Co As H | El uso de escitalopram enantiomericamente puro. |
GB0118892D0 (en) * | 2001-08-02 | 2001-09-26 | Vernalis Res Ltd | Method of treatment |
SE0201544D0 (sv) * | 2002-05-17 | 2002-05-17 | Biovitrum Ab | Novel compounds and thier use |
MXPA05012493A (es) * | 2003-05-27 | 2006-05-25 | Forest Laboratories | Combinacion de un antagonista del receptor de nmda y un inhibidor selectivo de reabsorcion de serotonina para el tratamiento de depresion y otros trastornos de estado de animo. |
US20050234093A1 (en) * | 2003-06-25 | 2005-10-20 | H. Lundbeck A/S | Treatment of depression and other affective disorders |
AR047553A1 (es) * | 2003-07-04 | 2006-01-25 | Lundbeck & Co As H | La combinacion de un inhibidor de reabsorcion de serotonina y agomelatina |
EP1500391A1 (de) * | 2003-07-24 | 2005-01-26 | Neuro3D | Medizinische Verwendung von Bicycloheptan-Derivaten |
ES2319539T3 (es) | 2003-09-17 | 2009-05-08 | Janssen Pharmaceutica Nv | Compuestos heterociclicos condensados como moduladores del receptor de serotonina. |
EP1708790B1 (de) * | 2003-12-02 | 2010-04-21 | PharmaNeuroBoost N.V. | Verwendung von pipamperon und einem d2-rezeptor antagonisten oder einem serotonin/dopamin antagonisten zur behandlung von psychotischen störungen |
US7855195B2 (en) | 2003-12-02 | 2010-12-21 | Pharmaneuroboost N.V. | Method of treating mental disorders using D4 and 5-HT2A antagonists, inverse agonists or partial agonists |
US20050203130A1 (en) * | 2003-12-02 | 2005-09-15 | Erik Buntinx | Use of D4 and 5-HT2A antagonists, inverse agonists or partial agonists |
US7884096B2 (en) | 2003-12-02 | 2011-02-08 | Pharmaneuroboost N.V. | Method of treating mental disorders using of D4 and 5-HT2A antagonists, inverse agonists or partial agonists |
WO2005053703A1 (en) * | 2003-12-02 | 2005-06-16 | Leslie James Sheldon | Combination therapy for dementia, depression and apathy |
US20050241110A1 (en) * | 2004-04-09 | 2005-11-03 | Bruce Baker | Ergonomic handles, especially for garden tools |
US7598255B2 (en) | 2005-08-04 | 2009-10-06 | Janssen Pharmaceutica Nv | Pyrimidine compounds as serotonin receptor modulators |
JP2009538117A (ja) * | 2006-03-22 | 2009-11-05 | ハー・ルンドベック・アクチエゼルスカベット | うつ病を処置するための化合物を同定する方法 |
BRPI0713425A2 (pt) | 2006-06-16 | 2012-03-13 | H. Lundbeck A/S | composto, composição farmacêutica, método para tratar uma doença, uso de um composto, e processos para a preparação de um composto, e para a fabricação de um composto |
US20080081067A1 (en) * | 2006-10-03 | 2008-04-03 | Gupta Manishkumar | Sustained release pharmaceutical compositions of venlafaxine and process for preparation thereof |
JP5460594B2 (ja) * | 2007-08-03 | 2014-04-02 | リチュテル・ゲデオン・ヴェジェーセティ・ジャール・ニュイルヴァーノシャン・ミューコェデー・レースヴェーニュタールシャシャーグ | ドーパミン受容体リガンドを含有する医薬組成物およびドーパミン受容体リガンドを用いる処置方法 |
WO2009082268A2 (ru) | 2007-12-21 | 2009-07-02 | Alla Chem, Llc | ЛИГАНДЫ α-АДРЕНОЦЕПТОРОВ, ДОПАМИНОВЫХ, ГИСТАМИНОВЫХ, ИМИДАЗОЛИНОВЫХ И СЕРОТОНИНОВЫХ РЕЦЕПТОРОВ И ИХ ПРИМЕНЕНИЕ |
WO2010006231A1 (en) * | 2008-07-10 | 2010-01-14 | Ore Pharmaceuticals Inc. | Treating inflammation and related conditions with irindalone |
WO2012008528A1 (ja) | 2010-07-15 | 2012-01-19 | 大日本住友製薬株式会社 | ピラゾール化合物 |
WO2012054815A1 (en) | 2010-10-22 | 2012-04-26 | Duke University | Slow-release formulations of 5-hydroxytryptophan as an adjunct to pro-serotonergic therapies |
WO2013119800A1 (en) | 2012-02-07 | 2013-08-15 | Massachusetts Institute Of Technology | Use of antagonists of ghrelin or ghrelin receptor to prevent or treat stress-sensitive psychiatric illness |
WO2014046544A1 (en) | 2012-09-21 | 2014-03-27 | Aapa B.V. | Substituted 3-heteroaryloxy-3-(hetero)aryl-propylamines as serotonin transporter and serotonin ht2c receptor modulators |
WO2014144231A1 (en) | 2013-03-15 | 2014-09-18 | Massachusetts Institute Of Technology | Use of antagonists of growth hormone or growth hormone receptor to prevent or treat stress-sensitive psychiatric illness |
US10317418B2 (en) | 2015-02-24 | 2019-06-11 | Massachusetts Institute Of Technology | Use of ghrelin or functional ghrelin receptor agonists to prevent and treat stress-sensitive psychiatric illness |
WO2016205631A1 (en) * | 2015-06-17 | 2016-12-22 | Massachusetts Institute Of Technology | Serotonin 2c receptor antagonists to prevent and treat stress-related trauma disorders |
CN107556206A (zh) * | 2016-06-30 | 2018-01-09 | 陕西合成药业股份有限公司 | 一种新型5‑羟色胺再摄取抑制剂类化合物及其制备方法和在医学上的应用 |
US11478467B2 (en) | 2017-05-04 | 2022-10-25 | Sreenivasarao Vepachedu | Targeted drug rescue with novel compositions, combinations, and methods thereof |
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GB8814057D0 (en) * | 1988-06-14 | 1988-07-20 | Lundbeck & Co As H | New enantiomers & their isolation |
US5155218A (en) * | 1990-05-08 | 1992-10-13 | Neurogenetic Corporation | Dna encoding human 5-ht1d receptors |
WO1994004533A1 (en) | 1992-08-20 | 1994-03-03 | Smithkline Beecham Plc | Condensed indole derivatives as 5ht2c and 5ht2b antagonists |
WO1994014801A1 (en) | 1992-12-29 | 1994-07-07 | Smithkline Beecham Plc | Heterocyclic urea derivatives as 5ht2c and 5ht2b antagonists |
ATE187448T1 (de) * | 1993-02-10 | 1999-12-15 | Yamanouchi Pharma Co Ltd | Morpholinderivate |
GB9313913D0 (en) | 1993-07-06 | 1993-08-18 | Smithkline Beecham Plc | Novel compounds |
CA2134038C (en) * | 1994-06-16 | 1997-06-03 | David Taiwai Wong | Potentiation of drug response |
MX9700693A (es) * | 1994-07-26 | 1997-04-30 | Pfizer | Derivados del 4-indol. |
US5597826A (en) | 1994-09-14 | 1997-01-28 | Pfizer Inc. | Compositions containing sertraline and a 5-HT1D receptor agonist or antagonist |
GB9420999D0 (en) | 1994-10-18 | 1994-12-07 | Smithkline Beecham Plc | Novel compounds |
EP0714663A3 (de) * | 1994-11-28 | 1997-01-15 | Lilly Co Eli | Potenzierung von Wirkstoffresponz durch Serotonin 1A Rezeptor Antagonisten |
EP0807104A2 (de) | 1995-02-02 | 1997-11-19 | Smithkline Beecham Plc | Heterozyklische verbindungen mit 5ht2c rezeptor antagonismus |
SE9501567D0 (sv) * | 1995-04-27 | 1995-04-27 | Astra Ab | A new combination |
GB9511355D0 (en) | 1995-06-06 | 1995-08-02 | Fujisawa Pharmaceutical Co | Urea derivatives |
GB9514384D0 (en) * | 1995-07-13 | 1995-09-13 | American Home Prod | Medical treatment |
GB9517559D0 (en) | 1995-08-26 | 1995-10-25 | Smithkline Beecham Plc | Novel compounds |
FR2744449B1 (fr) | 1996-02-02 | 1998-04-24 | Pf Medicament | Nouvelles piperazines aromatiques derivees de cycloazanes substitues, ainsi que leur procede de preparation, les compositions pharmaceutiques et leur utilisation comme medicaments |
GB9607219D0 (en) | 1996-04-04 | 1996-06-12 | Smithkline Beecham Plc | Novel compounds |
ES2182064T3 (es) | 1996-04-12 | 2003-03-01 | Janssen Pharmaceutica Nv | Derivados de isoxazolidina. |
EP0813873B1 (de) * | 1996-06-19 | 2002-02-13 | Akzo Nobel N.V. | Pharmazeutische Zusammensetzungen mit Mirtazapin und einem oder mehreren selektiven Serotonin-Aufnahme Inhibitoren |
US5958429A (en) * | 1996-08-16 | 1999-09-28 | Eli Lilly And Company | Potentiation of serotonin response |
SE9703375D0 (sv) | 1997-09-18 | 1997-09-18 | Astra Ab | A new combination |
US6960577B2 (en) * | 1998-05-22 | 2005-11-01 | Eli Lilly And Company | Combination therapy for treatment of refractory depression |
BR9911049A (pt) * | 1998-05-22 | 2001-02-06 | Lilly Co Eli | Terapia combinada para tratamento de depressão resistente |
CZ20004280A3 (cs) * | 1998-05-29 | 2001-09-12 | Eli Lilly And Company | Lék pro léčbu bipolárních poruch a farmaceutický prostředek |
DE19827750C1 (de) * | 1998-06-22 | 1999-07-29 | Centeon Pharma Gmbh | Verfahren zum Abtrennen von HIV aus einer Flüssigkeit |
DE19900673A1 (de) * | 1999-01-11 | 2000-07-13 | Basf Ag | Verwendung von Bindungspartnern für 5-HT5-Rezeptoren zur Behandlung neurodegenerativer und neuropsychiatrischer Störungen |
US20070259952A1 (en) * | 2006-05-02 | 2007-11-08 | H. Lundbeck A/S | Uses of escitalopram |
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2000
- 2000-06-12 UA UA2002065005A patent/UA77650C2/uk unknown
- 2000-12-04 AU AU18508/01A patent/AU1850801A/en not_active Abandoned
- 2000-12-04 WO PCT/DK2000/000667 patent/WO2001041766A1/en active Application Filing
- 2000-12-05 CO CO00092734A patent/CO5251409A1/es unknown
- 2000-12-06 TR TR2002/01512T patent/TR200201512T2/xx unknown
- 2000-12-06 PL PL00356402A patent/PL356402A1/xx not_active Application Discontinuation
- 2000-12-06 JP JP2001542871A patent/JP2003516326A/ja not_active Withdrawn
- 2000-12-06 PT PT00981174T patent/PT1237553E/pt unknown
- 2000-12-06 BR BR0016385-6A patent/BR0016385A/pt not_active Application Discontinuation
- 2000-12-06 CZ CZ20021961A patent/CZ20021961A3/cs unknown
- 2000-12-06 MX MXPA02005613A patent/MXPA02005613A/es not_active Application Discontinuation
- 2000-12-06 KR KR1020027007231A patent/KR100832026B1/ko not_active IP Right Cessation
- 2000-12-06 YU YU41902A patent/YU41902A/sh unknown
- 2000-12-06 CA CA002393470A patent/CA2393470A1/en not_active Abandoned
- 2000-12-06 EP EP00981174A patent/EP1237553B1/de not_active Expired - Lifetime
- 2000-12-06 DK DK00981174T patent/DK1237553T3/da active
- 2000-12-06 DE DE60025398T patent/DE60025398T2/de not_active Expired - Fee Related
- 2000-12-06 AT AT00981174T patent/ATE314849T1/de not_active IP Right Cessation
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- 2000-12-06 US US09/731,411 patent/US20020103249A1/en not_active Abandoned
- 2000-12-06 NZ NZ545907A patent/NZ545907A/en unknown
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- 2000-12-06 ME MEP-62/08A patent/MEP6208A/xx unknown
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- 2000-12-06 EP EP08021043A patent/EP2036564A1/de not_active Withdrawn
- 2000-12-06 EA EA200200649A patent/EA006391B1/ru not_active IP Right Cessation
- 2000-12-06 HU HU0203586A patent/HUP0203586A3/hu unknown
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2002
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2006
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- 2006-10-05 US US11/539,100 patent/US20070105843A1/en not_active Abandoned
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2009
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