UA69438C2 - Morpholine benzamide salts - Google Patents
Morpholine benzamide salts Download PDFInfo
- Publication number
- UA69438C2 UA69438C2 UA2001085896A UA2001085896A UA69438C2 UA 69438 C2 UA69438 C2 UA 69438C2 UA 2001085896 A UA2001085896 A UA 2001085896A UA 2001085896 A UA2001085896 A UA 2001085896A UA 69438 C2 UA69438 C2 UA 69438C2
- Authority
- UA
- Ukraine
- Prior art keywords
- salt
- tetrahydro
- naphthyl
- disorders
- methyl
- Prior art date
Links
- PUDYSBKPGVXBNQ-UHFFFAOYSA-N benzamide;morpholine Chemical class C1COCCN1.NC(=O)C1=CC=CC=C1 PUDYSBKPGVXBNQ-UHFFFAOYSA-N 0.000 title 1
- 150000001875 compounds Chemical class 0.000 claims abstract description 75
- 150000003839 salts Chemical class 0.000 claims abstract description 62
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
- C07D295/14—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D295/155—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals with the ring nitrogen atoms and the carbon atoms with three bonds to hetero atoms separated by carbocyclic rings or by carbon chains interrupted by carbocyclic rings
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
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- A—HUMAN NECESSITIES
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Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Psychiatry (AREA)
- Addiction (AREA)
- Pain & Pain Management (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Psychology (AREA)
- Endocrinology (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Child & Adolescent Psychology (AREA)
- Hospice & Palliative Care (AREA)
- Rheumatology (AREA)
- Obesity (AREA)
- Reproductive Health (AREA)
- Urology & Nephrology (AREA)
- Nutrition Science (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| SE9900190A SE9900190D0 (sv) | 1999-01-22 | 1999-01-22 | New compounds |
| PCT/SE2000/000079 WO2000043378A1 (en) | 1999-01-22 | 2000-01-14 | New morpholinobenzamide salts |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| UA69438C2 true UA69438C2 (en) | 2004-09-15 |
Family
ID=20414186
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| UA2001085896A UA69438C2 (en) | 1999-01-22 | 2000-01-14 | Morpholine benzamide salts |
Country Status (28)
| Country | Link |
|---|---|
| US (1) | US6291458B1 (hu) |
| EP (1) | EP1149083A1 (hu) |
| JP (1) | JP2002535320A (hu) |
| KR (1) | KR20010101585A (hu) |
| CN (1) | CN1188405C (hu) |
| AR (1) | AR030145A1 (hu) |
| AU (1) | AU778674B2 (hu) |
| BR (1) | BR0007577A (hu) |
| CA (1) | CA2359105A1 (hu) |
| CZ (1) | CZ20012643A3 (hu) |
| DZ (1) | DZ3002A1 (hu) |
| EE (1) | EE200100381A (hu) |
| HU (1) | HUP0200412A3 (hu) |
| ID (1) | ID30556A (hu) |
| IL (1) | IL144444A0 (hu) |
| IS (1) | IS6007A (hu) |
| MY (1) | MY133438A (hu) |
| NO (1) | NO20013601L (hu) |
| NZ (1) | NZ512684A (hu) |
| PL (1) | PL349775A1 (hu) |
| RU (1) | RU2237668C2 (hu) |
| SE (1) | SE9900190D0 (hu) |
| SK (1) | SK10222001A3 (hu) |
| TN (1) | TNSN00015A1 (hu) |
| TR (1) | TR200102087T2 (hu) |
| UA (1) | UA69438C2 (hu) |
| WO (1) | WO2000043378A1 (hu) |
| ZA (1) | ZA200105491B (hu) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SE0002729D0 (sv) * | 2000-07-20 | 2000-07-20 | Astrazeneca Ab | Novel compound form |
| GT200600414A (es) | 2005-09-12 | 2007-09-20 | Sal de glucuranato de compuesto de piperazine | |
| TW200800306A (en) | 2005-09-12 | 2008-01-01 | Wyeth Corp | Sustained-release formulation and uses thereof |
| GT200600416A (es) * | 2005-09-12 | 2007-09-20 | Sales salicilato y gentisato de un compuesto de piperazina | |
| US20080033050A1 (en) * | 2006-08-04 | 2008-02-07 | Richards Patricia Allison Tewe | Method of treating thermoregulatory disfunction with paroxetine |
| RU2540464C2 (ru) * | 2012-05-28 | 2015-02-10 | Государственное бюджетное образовательное учреждение высшего профессионального образования "Волгоградский государственный медицинский университет" Министерства здравоохранения и социального развития Российской Федерации | Водорастворимое производное амида салициловой кислоты, обладающее транквилизирующей, ноотропной и анальгезирующей активностью |
| WO2020183011A1 (en) | 2019-03-14 | 2020-09-17 | Institut Curie | Htr1d inhibitors and uses thereof in the treatment of cancer |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3919624A1 (de) | 1989-06-15 | 1990-12-20 | Boehringer Ingelheim Kg | Neue 2,5-diaminotetraline, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel |
| GB9119920D0 (en) | 1991-09-18 | 1991-10-30 | Glaxo Group Ltd | Chemical compounds |
| ES2162792T3 (es) | 1991-09-18 | 2002-01-16 | Glaxo Group Ltd | Derivados de benzanilida como antagonistas de 5-ht1d. |
| GB9119932D0 (en) | 1991-09-18 | 1991-10-30 | Glaxo Group Ltd | Chemical compounds |
| DK148392D0 (da) | 1992-12-09 | 1992-12-09 | Lundbeck & Co As H | Heterocykliske forbindelser |
| GB2273930A (en) | 1992-12-30 | 1994-07-06 | Glaxo Group Ltd | Benzanilide derivatives |
| DK0689536T3 (da) * | 1993-03-16 | 2001-07-30 | Pfizer | Naphthalenderivater |
| EP0724580A1 (en) | 1993-10-19 | 1996-08-07 | Smithkline Beecham Plc | Benzanilide derivatives as 5ht-1d receptor antagonists |
| SE9601110D0 (sv) * | 1996-03-22 | 1996-03-22 | Astra Ab | Substituted 1,2,3,4-tetrahydronaphthalene derivatives |
| SE9702799D0 (sv) * | 1997-07-25 | 1997-07-25 | Astra Ab | New compounds |
-
1999
- 1999-01-22 SE SE9900190A patent/SE9900190D0/xx unknown
-
2000
- 2000-01-09 DZ DZ000004A patent/DZ3002A1/xx active
- 2000-01-14 TR TR2001/02087T patent/TR200102087T2/xx unknown
- 2000-01-14 EP EP00902246A patent/EP1149083A1/en not_active Withdrawn
- 2000-01-14 KR KR1020017009056A patent/KR20010101585A/ko not_active Application Discontinuation
- 2000-01-14 WO PCT/SE2000/000079 patent/WO2000043378A1/en not_active Application Discontinuation
- 2000-01-14 BR BR0007577-9A patent/BR0007577A/pt not_active IP Right Cessation
- 2000-01-14 SK SK1022-2001A patent/SK10222001A3/sk unknown
- 2000-01-14 CA CA002359105A patent/CA2359105A1/en not_active Abandoned
- 2000-01-14 EE EEP200100381A patent/EE200100381A/xx unknown
- 2000-01-14 ID IDW00200101578A patent/ID30556A/id unknown
- 2000-01-14 UA UA2001085896A patent/UA69438C2/uk unknown
- 2000-01-14 RU RU2001123433A patent/RU2237668C2/ru not_active IP Right Cessation
- 2000-01-14 AU AU23374/00A patent/AU778674B2/en not_active Ceased
- 2000-01-14 CZ CZ20012643A patent/CZ20012643A3/cs unknown
- 2000-01-14 PL PL00349775A patent/PL349775A1/xx not_active Application Discontinuation
- 2000-01-14 CN CNB008030103A patent/CN1188405C/zh not_active Expired - Fee Related
- 2000-01-14 HU HU0200412A patent/HUP0200412A3/hu unknown
- 2000-01-14 IL IL14444400A patent/IL144444A0/xx unknown
- 2000-01-14 NZ NZ512684A patent/NZ512684A/xx unknown
- 2000-01-14 JP JP2000594794A patent/JP2002535320A/ja active Pending
- 2000-01-18 AR ARP000100215A patent/AR030145A1/es unknown
- 2000-01-20 TN TNTNSN00015A patent/TNSN00015A1/fr unknown
- 2000-01-20 MY MYPI20000180A patent/MY133438A/en unknown
- 2000-07-21 US US09/621,387 patent/US6291458B1/en not_active Expired - Fee Related
-
2001
- 2001-07-03 ZA ZA200105491A patent/ZA200105491B/en unknown
- 2001-07-17 IS IS6007A patent/IS6007A/is unknown
- 2001-07-20 NO NO20013601A patent/NO20013601L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| IS6007A (is) | 2001-07-17 |
| NO20013601L (no) | 2001-09-11 |
| ID30556A (id) | 2001-12-20 |
| IL144444A0 (en) | 2002-05-23 |
| WO2000043378A1 (en) | 2000-07-27 |
| TR200102087T2 (tr) | 2001-12-21 |
| PL349775A1 (en) | 2002-09-09 |
| JP2002535320A (ja) | 2002-10-22 |
| AR030145A1 (es) | 2003-08-13 |
| EE200100381A (et) | 2002-12-16 |
| NZ512684A (en) | 2003-06-30 |
| CN1188405C (zh) | 2005-02-09 |
| RU2237668C2 (ru) | 2004-10-10 |
| KR20010101585A (ko) | 2001-11-14 |
| SK10222001A3 (sk) | 2002-03-05 |
| HUP0200412A3 (en) | 2002-11-28 |
| CN1337956A (zh) | 2002-02-27 |
| AU778674B2 (en) | 2004-12-16 |
| HUP0200412A2 (en) | 2002-06-29 |
| DZ3002A1 (fr) | 2004-03-27 |
| CZ20012643A3 (cs) | 2002-01-16 |
| EP1149083A1 (en) | 2001-10-31 |
| SE9900190D0 (sv) | 1999-01-22 |
| NO20013601D0 (no) | 2001-07-20 |
| TNSN00015A1 (fr) | 2005-11-10 |
| US6291458B1 (en) | 2001-09-18 |
| AU2337400A (en) | 2000-08-07 |
| CA2359105A1 (en) | 2000-07-27 |
| MY133438A (en) | 2007-11-30 |
| BR0007577A (pt) | 2001-10-23 |
| ZA200105491B (en) | 2002-10-03 |
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