UA112061C2 - Активуючі ampk гетероциклічні сполуки і способи їх використання - Google Patents
Активуючі ampk гетероциклічні сполуки і способи їх використанняInfo
- Publication number
- UA112061C2 UA112061C2 UAA201302459A UAA201302459A UA112061C2 UA 112061 C2 UA112061 C2 UA 112061C2 UA A201302459 A UAA201302459 A UA A201302459A UA A201302459 A UAA201302459 A UA A201302459A UA 112061 C2 UA112061 C2 UA 112061C2
- Authority
- UA
- Ukraine
- Prior art keywords
- methods
- heterocyclic compounds
- ampk activating
- activating heterocyclic
- ampk
- Prior art date
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Abstract
Розкриті заміщені піридинові сполуки, а також фармацевтичні композиції і способи використання. Один варіант здійснення являє собою сполуку, яка характеризується структурою,де значення Е, J, Т, позначеної "В" кільцевої системи, Т, R, R, w і х описані в даному документі. Відповідно до визначених варіантів здійснення, розкрита в даному документі сполука активує метаболічний шлях АМРК і може бути використана для лікування пов'язаних з метаболізмом порушень і станів.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
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US36892810P | 2010-07-29 | 2010-07-29 | |
PCT/US2011/046019 WO2012016217A1 (en) | 2010-07-29 | 2011-07-29 | Ampk-activating heterocyclic compounds and methods for using the same |
Publications (1)
Publication Number | Publication Date |
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UA112061C2 true UA112061C2 (uk) | 2016-07-25 |
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Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
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UAA201302459A UA112061C2 (uk) | 2010-07-29 | 2011-07-29 | Активуючі ampk гетероциклічні сполуки і способи їх використання |
Country Status (24)
Country | Link |
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US (8) | US8791136B2 (uk) |
EP (1) | EP2598483B1 (uk) |
JP (1) | JP5889895B2 (uk) |
KR (1) | KR101764952B1 (uk) |
CN (1) | CN103201267B (uk) |
AU (1) | AU2011283684B2 (uk) |
BR (1) | BR112013002112B1 (uk) |
CA (1) | CA2806341C (uk) |
CL (1) | CL2013000261A1 (uk) |
DK (1) | DK2598483T3 (uk) |
EA (1) | EA025611B1 (uk) |
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