TWI688566B - ６,７-二氫吡唑並[１,５-α]吡-４(５Ｈ)-酮化合物及其作為ＭＧＬＵＲ２受體的負性別構調節物之用途 - Google Patents

６,７-二氫吡唑並[１,５-α]吡-４(５Ｈ)-酮化合物及其作為ＭＧＬＵＲ２受體的負性別構調節物之用途 Download PDF

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TWI688566B
TWI688566B TW104124698A TW104124698A TWI688566B TW I688566 B TWI688566 B TW I688566B TW 104124698 A TW104124698 A TW 104124698A TW 104124698 A TW104124698 A TW 104124698A TW I688566 B TWI688566 B TW I688566B
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alkyl
group
disorders
pyridine
compound
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TW104124698A
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TW201625630A (zh
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塞吉奧阿爾瓦 阿隆索地亞哥
麥克 范高
瑪麗亞 馬丁馬汀
蘇珊娜 寇迪塞德
荷西 安德烈斯吉爾
奧斯卡 德爾加多岡薩雷斯
蓋瑞 特雷薩德恩
安德烈斯 特瑞巴克蘇亞雷斯
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比利時商健生藥品公司
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/50—Pyridazines; Hydrogenated pyridazines
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
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  • Hospice & Palliative Care (AREA)
  • Addiction (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
TW104124698A 2014-08-01 2015-07-30 ６,７-二氫吡唑並[１,５-α]吡-４(５Ｈ)-酮化合物及其作為ＭＧＬＵＲ２受體的負性別構調節物之用途 TWI688566B (zh)

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EP14179600.3 2014-08-01
EP14179600 2014-08-01
EP14196083 2014-12-03
EP14196083.1 2014-12-03

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TWI688566B true TWI688566B (zh) 2020-03-21

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