TWI453029B - 去氧艾克特卡丁b(deoxyactagardine b), 包含其之醫藥組合物及其製造方法 - Google Patents

去氧艾克特卡丁b(deoxyactagardine b), 包含其之醫藥組合物及其製造方法 Download PDF

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Publication number
TWI453029B
TWI453029B TW099100713A TW99100713A TWI453029B TW I453029 B TWI453029 B TW I453029B TW 099100713 A TW099100713 A TW 099100713A TW 99100713 A TW99100713 A TW 99100713A TW I453029 B TWI453029 B TW I453029B
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TW
Taiwan
Prior art keywords
compound
compounds
pharmaceutical composition
treatment
pharmaceutically acceptable
Prior art date
Application number
TW099100713A
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English (en)
Chinese (zh)
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TW201029661A (en
Inventor
Sjoerd Nicolaas Wadman
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Novacta Biosystems Ltd
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Publication of TW201029661A publication Critical patent/TW201029661A/zh
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Publication of TWI453029B publication Critical patent/TWI453029B/zh

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/50—Cyclic peptides containing at least one abnormal peptide link
    • C07K7/54—Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/12—Cyclic peptides, e.g. bacitracins; Polymyxins; Gramicidins S, C; Tyrocidins A, B or C
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Engineering & Computer Science (AREA)
  • Communicable Diseases (AREA)
  • Epidemiology (AREA)
  • Oncology (AREA)
  • Immunology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Hydrogenated Pyridines (AREA)
  • Polysaccharides And Polysaccharide Derivatives (AREA)
  • Saccharide Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
TW099100713A 2009-01-14 2010-01-12 去氧艾克特卡丁b(deoxyactagardine b), 包含其之醫藥組合物及其製造方法 TWI453029B (zh)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US14449009P 2009-01-14 2009-01-14

Publications (2)

Publication Number Publication Date
TW201029661A TW201029661A (en) 2010-08-16
TWI453029B true TWI453029B (zh) 2014-09-21

Family

ID=42110329

Family Applications (1)

Application Number Title Priority Date Filing Date
TW099100713A TWI453029B (zh) 2009-01-14 2010-01-12 去氧艾克特卡丁b(deoxyactagardine b), 包含其之醫藥組合物及其製造方法

Country Status (22)

Country Link
US (2) US8283371B2 (enExample)
EP (1) EP2387580B1 (enExample)
JP (1) JP5719312B2 (enExample)
KR (1) KR20110119699A (enExample)
CN (1) CN102348718B (enExample)
AU (1) AU2010205472B2 (enExample)
CA (1) CA2749278A1 (enExample)
DK (1) DK2387580T3 (enExample)
EA (1) EA021683B1 (enExample)
ES (1) ES2520165T3 (enExample)
HR (1) HRP20141084T1 (enExample)
IL (1) IL213927A0 (enExample)
MX (1) MX2011007313A (enExample)
NZ (1) NZ594011A (enExample)
PL (1) PL2387580T3 (enExample)
PT (1) PT2387580E (enExample)
RS (1) RS53586B1 (enExample)
SG (1) SG172944A1 (enExample)
SI (1) SI2387580T1 (enExample)
TW (1) TWI453029B (enExample)
WO (1) WO2010082018A1 (enExample)
ZA (1) ZA201104991B (enExample)

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GB0714029D0 (en) * 2007-07-18 2007-08-29 Novacta Biosystems Ltd Lantibiotic-based compounds having antimicrobial activity
GB0714030D0 (en) * 2007-07-18 2007-08-29 Novacta Biosystems Ltd The use of type-B lantibiotic-based compounds having antimicrobial activity
NZ594011A (en) 2009-01-14 2013-12-20 Novacta Biosystems Ltd Deoxyactagardine derivatives
KR20110122139A (ko) 2009-02-04 2011-11-09 노박타 바이오시스템스 리미티드 액타가르딘 유도체
WO2011061748A1 (en) * 2009-11-19 2011-05-26 Strides Arcolab Limited Rifaximin premix
GB201001688D0 (en) 2010-02-02 2010-03-17 Novacta Biosystems Ltd Compounds
GB201013513D0 (en) * 2010-08-11 2010-09-22 Novacta Biosystems Ltd Formulations
GB201013507D0 (en) * 2010-08-11 2010-09-22 Novacta Biosystems Ltd Compounds
GB201013509D0 (en) * 2010-08-11 2010-09-22 Novacta Biosystems Ltd Compounds
GB201013508D0 (en) * 2010-08-11 2010-09-22 Novacta Biosystems Ltd Compounds
GB201213434D0 (en) 2012-07-27 2012-09-12 Novacta Biosystems Ltd The use of type-B lantibiotic-based compounds having antimicrobial activity

Citations (1)

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WO2007083112A2 (en) * 2006-01-17 2007-07-26 Novacta Biosystems Limited Lantibiotic biosynthetic gene clusters from a. garbadinensis and a. liguriae

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WO2007083112A2 (en) * 2006-01-17 2007-07-26 Novacta Biosystems Limited Lantibiotic biosynthetic gene clusters from a. garbadinensis and a. liguriae

Also Published As

Publication number Publication date
PT2387580E (pt) 2014-10-30
JP2012515195A (ja) 2012-07-05
SI2387580T1 (sl) 2014-11-28
CN102348718A (zh) 2012-02-08
KR20110119699A (ko) 2011-11-02
EP2387580A1 (en) 2011-11-23
ES2520165T3 (es) 2014-11-11
ZA201104991B (en) 2013-10-31
CN102348718B (zh) 2015-06-03
WO2010082018A1 (en) 2010-07-22
CA2749278A1 (en) 2010-07-22
US8741945B2 (en) 2014-06-03
MX2011007313A (es) 2011-08-04
TW201029661A (en) 2010-08-16
US20100179207A1 (en) 2010-07-15
DK2387580T3 (da) 2014-10-13
NZ594011A (en) 2013-12-20
EP2387580B1 (en) 2014-08-13
HRP20141084T1 (hr) 2015-02-13
US20120277145A1 (en) 2012-11-01
JP5719312B2 (ja) 2015-05-13
IL213927A0 (en) 2011-07-31
EA021683B1 (ru) 2015-08-31
EA201190071A1 (ru) 2012-06-29
SG172944A1 (en) 2011-08-29
AU2010205472B2 (en) 2013-03-14
US8283371B2 (en) 2012-10-09
AU2010205472A1 (en) 2011-07-28
RS53586B1 (sr) 2015-02-27
PL2387580T3 (pl) 2015-01-30

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