TWI231759B - Olopatadine formulations for topical administration - Google Patents

Olopatadine formulations for topical administration Download PDF

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Publication number
TWI231759B
TWI231759B TW091113234A TW91113234A TWI231759B TW I231759 B TWI231759 B TW I231759B TW 091113234 A TW091113234 A TW 091113234A TW 91113234 A TW91113234 A TW 91113234A TW I231759 B TWI231759 B TW I231759B
Authority
TW
Taiwan
Prior art keywords
solution
item
composition
acid
clarification
Prior art date
Application number
TW091113234A
Other languages
English (en)
Chinese (zh)
Inventor
Ernesto J Castillo
Wesley Wehsin Han
Huixiang Zhang
Hareshg Bhagat
Onkar N Singh
Original Assignee
Alcon Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=23162841&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=TWI231759(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Alcon Inc filed Critical Alcon Inc
Application granted granted Critical
Publication of TWI231759B publication Critical patent/TWI231759B/zh

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0043—Nose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/32—Macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. carbomers, poly(meth)acrylates, or polyvinyl pyrrolidone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0048—Eye, e.g. artificial tears
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/02—Nasal agents, e.g. decongestants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/14—Decongestants or antiallergics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Ophthalmology & Optometry (AREA)
  • Otolaryngology (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Inorganic Chemistry (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
TW091113234A 2001-06-27 2002-06-18 Olopatadine formulations for topical administration TWI231759B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US30131501P 2001-06-27 2001-06-27

Publications (1)

Publication Number Publication Date
TWI231759B true TWI231759B (en) 2005-05-01

Family

ID=23162841

Family Applications (1)

Application Number Title Priority Date Filing Date
TW091113234A TWI231759B (en) 2001-06-27 2002-06-18 Olopatadine formulations for topical administration

Country Status (20)

Country Link
US (2) US6995186B2 (cg-RX-API-DMAC7.html)
EP (1) EP1399127B1 (cg-RX-API-DMAC7.html)
JP (5) JP4827374B2 (cg-RX-API-DMAC7.html)
KR (1) KR100884711B1 (cg-RX-API-DMAC7.html)
CN (1) CN1211125C (cg-RX-API-DMAC7.html)
AR (1) AR034619A1 (cg-RX-API-DMAC7.html)
AT (1) ATE295149T1 (cg-RX-API-DMAC7.html)
AU (1) AU2002310461B2 (cg-RX-API-DMAC7.html)
BR (1) BRPI0210707B8 (cg-RX-API-DMAC7.html)
CA (1) CA2447924C (cg-RX-API-DMAC7.html)
DE (1) DE60204142T2 (cg-RX-API-DMAC7.html)
DK (1) DK1399127T3 (cg-RX-API-DMAC7.html)
ES (1) ES2238574T3 (cg-RX-API-DMAC7.html)
GC (1) GC0000397A (cg-RX-API-DMAC7.html)
MX (1) MXPA03011947A (cg-RX-API-DMAC7.html)
PL (1) PL205565B1 (cg-RX-API-DMAC7.html)
PT (1) PT1399127E (cg-RX-API-DMAC7.html)
TW (1) TWI231759B (cg-RX-API-DMAC7.html)
WO (1) WO2003002093A1 (cg-RX-API-DMAC7.html)
ZA (1) ZA200308771B (cg-RX-API-DMAC7.html)

Cited By (1)

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TWI427052B (zh) * 2005-09-30 2014-02-21 Johnson & Johnson Vision Care 穩定眼科組成物之方法

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TWI231759B (en) * 2001-06-27 2005-05-01 Alcon Inc Olopatadine formulations for topical administration
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ZA200610350B (en) * 2004-06-28 2008-12-31 Alcon Inc Topical formulations for treating allergic diseases
PL1814538T3 (pl) * 2004-11-24 2010-02-26 Alcon Inc Sposób dostarczania donosowego sprayu
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PT2453872E (pt) * 2009-07-17 2013-10-30 Alcon Res Ltd Regime de pulverização nasal de olopatadina para crianças
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KR20120091037A (ko) * 2009-10-01 2012-08-17 알콘 리서치, 리미티드 올로파타딘 조성물 및 그의 용도
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CA2812164A1 (en) * 2010-11-08 2012-05-18 Healor Ltd. Buffered ophthalmic compositions and methods of use thereof
TWI544922B (zh) * 2011-05-19 2016-08-11 愛爾康研究有限公司 高濃度歐羅派特錠（ｏｌｏｐａｔａｄｉｎｅ）眼用組成物
CN102885767A (zh) * 2012-11-02 2013-01-23 江苏吉贝尔药业有限公司 一种新的盐酸奥洛他定滴眼液及其制备方法
MA47418A (fr) 2017-02-01 2021-06-02 Takeda Pharmaceuticals Co Composés et compositions pour le traitement de troubles ophtalmiques
WO2018235935A1 (ja) * 2017-06-23 2018-12-27 参天製薬株式会社 水溶性粘稠化剤を含有する医薬組成物
JP7037349B2 (ja) * 2017-06-23 2022-03-16 参天製薬株式会社 水溶性粘稠化剤を含有する医薬組成物
AU2020398812A1 (en) * 2019-12-06 2022-06-30 Toko Yakuhin Kogyo Co., Ltd. Rhinenchysis composition containing olopatadine
EP4129341A4 (en) * 2020-03-31 2024-04-24 Santen Pharmaceutical Co., Ltd. AQUEOUS OPHTHALMIC COMPOSITION CONTAINING A SILVER SALT BY MEANS OF WHICH A RESIN CONTAINER IS FILLED
CN111700860A (zh) * 2020-07-09 2020-09-25 浙江尖峰药业有限公司 盐酸奥洛他定滴眼液及其制备方法
CN119318630B (zh) * 2024-10-16 2025-08-22 苏州欧康维视生物科技有限公司 一种阿托品药物组合物

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Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI427052B (zh) * 2005-09-30 2014-02-21 Johnson & Johnson Vision Care 穩定眼科組成物之方法

Also Published As

Publication number Publication date
ATE295149T1 (de) 2005-05-15
US6995186B2 (en) 2006-02-07
AU2002310461B2 (en) 2006-05-18
CN1211125C (zh) 2005-07-20
PL367780A1 (en) 2005-03-07
DK1399127T3 (da) 2005-06-13
BR0210707A (pt) 2004-07-20
US7402609B2 (en) 2008-07-22
CA2447924A1 (en) 2003-01-09
BRPI0210707B8 (pt) 2021-05-25
ES2238574T3 (es) 2005-09-01
WO2003002093A1 (en) 2003-01-09
DE60204142T2 (de) 2005-10-06
JP2013127005A (ja) 2013-06-27
JP4827374B2 (ja) 2011-11-30
HK1059573A1 (en) 2004-07-09
AR034619A1 (es) 2004-03-03
DE60204142D1 (de) 2005-06-16
MXPA03011947A (es) 2004-03-26
KR20040025919A (ko) 2004-03-26
CA2447924C (en) 2009-11-03
JP2009114213A (ja) 2009-05-28
PT1399127E (pt) 2005-07-29
JP2004536096A (ja) 2004-12-02
KR100884711B1 (ko) 2009-02-19
JP2010150292A (ja) 2010-07-08
EP1399127B1 (en) 2005-05-11
JP5328947B2 (ja) 2013-10-30
US20030055102A1 (en) 2003-03-20
CN1525849A (zh) 2004-09-01
US20050158387A1 (en) 2005-07-21
EP1399127A1 (en) 2004-03-24
JP2012107046A (ja) 2012-06-07
GC0000397A (en) 2007-03-31
BRPI0210707B1 (pt) 2015-08-04
PL205565B1 (pl) 2010-05-31
ZA200308771B (en) 2005-01-26

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