TW202005970A - β－內醯胺化合物及丙磺舒之組合及其用途 - Google Patents

β－內醯胺化合物及丙磺舒之組合及其用途 Download PDF

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TW202005970A
TW202005970A TW108119817A TW108119817A TW202005970A TW 202005970 A TW202005970 A TW 202005970A TW 108119817 A TW108119817 A TW 108119817A TW 108119817 A TW108119817 A TW 108119817A TW 202005970 A TW202005970 A TW 202005970A
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pharmaceutically acceptable
acceptable salt
administration
probenecid
lactam compound
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TW108119817A
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English (en)
Chinese (zh)
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麥可 鄧恩
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愛爾蘭商伊泰倫醫療國際有限公司
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/429—Thiazoles condensed with heterocyclic ring systems
    • A61K31/43—Compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula, e.g. penicillins, penems
    • A61K31/431—Compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula, e.g. penicillins, penems containing further heterocyclic rings, e.g. ticarcillin, azlocillin, oxacillin
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TW108119817A 2018-06-07 2019-06-06 β－內醯胺化合物及丙磺舒之組合及其用途 TW202005970A (zh)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US201862682116P 2018-06-07 2018-06-07
US62/682,116 2018-06-07
US201962804970P 2019-02-13 2019-02-13
US62/804,970 2019-02-13

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US (3) US11554112B2 (https=)
EP (1) EP3801486A1 (https=)
JP (2) JP2021525787A (https=)
CN (2) CN112739338A (https=)
AU (1) AU2019281018B2 (https=)
BR (1) BR112020024498A2 (https=)
TW (1) TW202005970A (https=)
WO (1) WO2019234240A1 (https=)

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US11554112B2 (en) 2018-06-07 2023-01-17 Herum Therapeutics International Limited Combinations of β-lactam compounds and probenecid and uses thereof
MX2021009755A (es) 2019-02-13 2021-11-17 Iterum Therapeutics International Ltd Combinaciones de compuestos beta-lactámicos y probenecid, y usos de los mismos.
CA3169900A1 (en) * 2020-03-11 2021-09-16 Iterum Therapeutics International Limited Combinations of beta-lactam compounds, probenecid, and valproic acid and uses thereof
WO2021207606A1 (en) * 2020-04-10 2021-10-14 University Of Georgia Research Foundation, Inc. Methods for treatment of coronavirus infections
US11116737B1 (en) 2020-04-10 2021-09-14 University Of Georgia Research Foundation, Inc. Methods of using probenecid for treatment of coronavirus infections
CN111840236B (zh) * 2020-08-07 2022-09-02 安徽康正康仁药业有限公司 一种注射用美罗培南丙磺舒钠复方冻干制剂
CN111821462A (zh) * 2020-08-07 2020-10-27 安徽康正康仁药业有限公司 青霉素类钠盐与丙磺舒钠组成的复方冻干制剂
CN112076161B (zh) * 2020-08-07 2022-10-18 安徽康正康仁药业有限公司 一种头孢菌素类钠盐与丙磺舒钠组成的复方冻干制剂

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MX2021009755A (es) 2019-02-13 2021-11-17 Iterum Therapeutics International Ltd Combinaciones de compuestos beta-lactámicos y probenecid, y usos de los mismos.
CA3169900A1 (en) 2020-03-11 2021-09-16 Iterum Therapeutics International Limited Combinations of beta-lactam compounds, probenecid, and valproic acid and uses thereof

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JP2021525787A (ja) 2021-09-27
BR112020024498A2 (pt) 2021-03-02
US20230218588A1 (en) 2023-07-13
JP2024107004A (ja) 2024-08-08
CN118903120A (zh) 2024-11-08
US20190374516A1 (en) 2019-12-12
AU2019281018B2 (en) 2025-01-30
CN112739338A (zh) 2021-04-30
AU2019281018A1 (en) 2020-12-10
EP3801486A1 (en) 2021-04-14
US12109197B2 (en) 2024-10-08
US20250127764A1 (en) 2025-04-24
WO2019234240A1 (en) 2019-12-12

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