TW201728592A - Irak抑制劑及其用途 - Google Patents

Irak抑制劑及其用途 Download PDF

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Publication number
TW201728592A
TW201728592A TW106101765A TW106101765A TW201728592A TW 201728592 A TW201728592 A TW 201728592A TW 106101765 A TW106101765 A TW 106101765A TW 106101765 A TW106101765 A TW 106101765A TW 201728592 A TW201728592 A TW 201728592A
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Taiwan
Prior art keywords
compound
ring
group
formula
nitrogen
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TW106101765A
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English (en)
Chinese (zh)
Inventor
吉拉丹C 何瑞曼
羅納德T 威斯特
多納L 羅曼羅
梭尼斯 羅賓森
蜜 莎麗
馬修 大衛 瓦思勒
傑諾米 羅伯特 葛林梧
奎格E 瑪斯
林柏曼 羅撒納 坎培爾
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林伯士艾瑞斯公司
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Publication of TW201728592A publication Critical patent/TW201728592A/zh

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    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/53751,4-Oxazines, e.g. morpholine
    • A61K31/53771,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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    • A61K31/33Heterocyclic compounds
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    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4365Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system having sulfur as a ring hetero atom, e.g. ticlopidine
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    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
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    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

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TW106101765A 2012-01-10 2013-01-10 Irak抑制劑及其用途 TW201728592A (zh)

Applications Claiming Priority (5)

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