TW201400494A - 寡糖化合物之製造方法 - Google Patents

寡糖化合物之製造方法 Download PDF

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Publication number
TW201400494A
TW201400494A TW102110255A TW102110255A TW201400494A TW 201400494 A TW201400494 A TW 201400494A TW 102110255 A TW102110255 A TW 102110255A TW 102110255 A TW102110255 A TW 102110255A TW 201400494 A TW201400494 A TW 201400494A
Authority
TW
Taiwan
Prior art keywords
group
haloalkyl
alkyl
alkoxycarbonyl
sugar
Prior art date
Application number
TW102110255A
Other languages
English (en)
Chinese (zh)
Inventor
Fumitaka Goto
Takahiro Tomoyasu
Hiroki Okazaki
Hiroaki Yuasa
Hirofumi Ochiai
Hiroshi Akagi
Yuta Sato
Koichi Sorajo
Original Assignee
Otsuka Pharma Co Ltd
Otsuka Chemical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Otsuka Pharma Co Ltd, Otsuka Chemical Co Ltd filed Critical Otsuka Pharma Co Ltd
Publication of TW201400494A publication Critical patent/TW201400494A/zh

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/02—Acyclic radicals, not substituted by cyclic structures
    • C07H15/12—Acyclic radicals, not substituted by cyclic structures attached to a nitrogen atom of the saccharide radical
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Biotechnology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Crystallography & Structural Chemistry (AREA)
  • Saccharide Compounds (AREA)
  • Polysaccharides And Polysaccharide Derivatives (AREA)
TW102110255A 2012-03-22 2013-03-22 寡糖化合物之製造方法 TW201400494A (zh)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2012066433 2012-03-22

Publications (1)

Publication Number Publication Date
TW201400494A true TW201400494A (zh) 2014-01-01

Family

ID=49222799

Family Applications (1)

Application Number Title Priority Date Filing Date
TW102110255A TW201400494A (zh) 2012-03-22 2013-03-22 寡糖化合物之製造方法

Country Status (3)

Country Link
JP (1) JP6273199B2 (ja)
TW (1) TW201400494A (ja)
WO (1) WO2013141350A1 (ja)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN109096348A (zh) * 2018-09-12 2018-12-28 江苏美迪克化学品有限公司 一种磺达肝癸钠单糖中间体的制备方法

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2014047155A (ja) * 2012-08-30 2014-03-17 Tottori Univ 保護硫酸化オリゴ糖化合物及びその製造方法
JP7401882B2 (ja) * 2016-03-09 2023-12-20 株式会社糖鎖工学研究所 硫酸基を有する糖の製造方法
CN110862422B (zh) * 2019-11-11 2023-03-10 三峡大学 β-半乳烯糖氮苷的合成方法及其在制药中的应用

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH06795B2 (ja) * 1985-04-02 1994-01-05 理化学研究所 アシアロガングリオシド関連化合物の製造方法
JPH0631288B2 (ja) * 1985-12-02 1994-04-27 理化学研究所 ヒト絨毛膜性生殖腺刺激ホルモンの糖鎖関連多糖性ハプテンおよびその製造法
JPS62138497A (ja) * 1985-12-10 1987-06-22 Rikagaku Kenkyusho ラクト−ガングリオ系列スフインゴ糖脂質およびその製造法
DK39886D0 (da) * 1986-01-27 1986-01-27 Hans Goeran Magnusson Hydroxybeskyttelsesgrupper
JPS6341493A (ja) * 1986-08-06 1988-02-22 Rikagaku Kenkyusho ガングリオシドｇｍ↓２関連化合物及びその製造方法
JPS63221104A (ja) * 1987-03-09 1988-09-14 Rikagaku Kenkyusho ガングリオシド関連化合物及びその製造法
JPS63218692A (ja) * 1987-03-09 1988-09-12 Rikagaku Kenkyusho ガングリオシド関連化合物及びその製造法
JPH02300196A (ja) * 1989-05-15 1990-12-12 Mect Corp ガングリオシドＧＭ↓１↓ｂ関連化合物
AU7153991A (en) * 1989-12-13 1991-07-18 Glycomed Incorporated Synthesis of rotavirus receptor saccharides
US5466681A (en) * 1990-02-23 1995-11-14 Microcarb, Inc. Receptor conjugates for targeting penicillin antibiotics to bacteria
JPH05310770A (ja) * 1992-04-30 1993-11-22 Nisshin Oil Mills Ltd:The ガングリオシドＧＭ１ｂ類縁体
WO1999052922A1 (en) * 1998-04-10 1999-10-21 Helix Biopharma Corp. ANTIMICROBIAL βGalNAc(1→4)βGal DERIVATIVES AND METHODS OF USE
GB0602352D0 (en) * 2006-02-06 2006-03-15 Glycoform Ltd Glycoconjugation
BRPI1007325A2 (pt) * 2009-02-02 2019-09-24 Otsuka Pharma Co Ltd "baixo peso molecular de polissulfatados derivados de ácido hialurônico e medicamentos que contenham o mesmo."
JP2012046511A (ja) * 2010-07-30 2012-03-08 Otsuka Chem Co Ltd 低分子量多硫酸化ヒアルロン酸誘導体を含有する医薬

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN109096348A (zh) * 2018-09-12 2018-12-28 江苏美迪克化学品有限公司 一种磺达肝癸钠单糖中间体的制备方法
CN109096348B (zh) * 2018-09-12 2020-06-16 江苏美迪克化学品有限公司 一种磺达肝癸钠单糖中间体的制备方法

Also Published As

Publication number Publication date
JP6273199B2 (ja) 2018-01-31
WO2013141350A1 (ja) 2013-09-26
JPWO2013141350A1 (ja) 2015-08-03

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