TW200927118A - Treatment of vasomotor symptoms - Google Patents
Treatment of vasomotor symptoms Download PDFInfo
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- TW200927118A TW200927118A TW097134893A TW97134893A TW200927118A TW 200927118 A TW200927118 A TW 200927118A TW 097134893 A TW097134893 A TW 097134893A TW 97134893 A TW97134893 A TW 97134893A TW 200927118 A TW200927118 A TW 200927118A
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- acid
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- vascular
- motility
- menopause
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- 229940124597 therapeutic agent Drugs 0.000 description 1
- 238000002560 therapeutic procedure Methods 0.000 description 1
- QORWJWZARLRLPR-UHFFFAOYSA-H tricalcium bis(phosphate) Chemical compound [Ca+2].[Ca+2].[Ca+2].[O-]P([O-])([O-])=O.[O-]P([O-])([O-])=O QORWJWZARLRLPR-UHFFFAOYSA-H 0.000 description 1
- JEJAMASKDTUEBZ-UHFFFAOYSA-N tris(1,1,3-tribromo-2,2-dimethylpropyl) phosphate Chemical compound BrCC(C)(C)C(Br)(Br)OP(=O)(OC(Br)(Br)C(C)(C)CBr)OC(Br)(Br)C(C)(C)CBr JEJAMASKDTUEBZ-UHFFFAOYSA-N 0.000 description 1
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Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/12—Drugs for genital or sexual disorders; Contraceptives for climacteric disorders
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
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| US97160507P | 2007-09-12 | 2007-09-12 |
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| TW200927118A true TW200927118A (en) | 2009-07-01 |
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| TW097134893A TW200927118A (en) | 2007-09-12 | 2008-09-11 | Treatment of vasomotor symptoms |
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| MA (1) | MA31757B1 (enExample) |
| MX (1) | MX2010002032A (enExample) |
| NZ (1) | NZ584183A (enExample) |
| PE (1) | PE20091188A1 (enExample) |
| TN (1) | TN2010000108A1 (enExample) |
| TW (1) | TW200927118A (enExample) |
| UY (1) | UY31335A1 (enExample) |
| WO (1) | WO2009034111A1 (enExample) |
| ZA (1) | ZA201000384B (enExample) |
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| US10675280B2 (en) | 2001-10-20 | 2020-06-09 | Sprout Pharmaceuticals, Inc. | Treating sexual desire disorders with flibanserin |
| UA78974C2 (en) | 2001-10-20 | 2007-05-10 | Boehringer Ingelheim Pharma | Use of flibanserin for treating disorders of sexual desire |
| JP2009503020A (ja) | 2005-08-03 | 2009-01-29 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | 肥満症の治療におけるフリバンセリンの使用 |
| ATE524446T1 (de) * | 2006-12-20 | 2011-09-15 | Boehringer Ingelheim Int | Sulfatierte benzimidazolon-derivate mit gemischter serotonin-rezeptor-affinität |
| UY31335A1 (es) * | 2007-09-12 | 2009-04-30 | Tratamiento de sintomas vasomotores | |
| WO2017133337A1 (zh) * | 2016-02-02 | 2017-08-10 | 深圳市塔吉瑞生物医药有限公司 | 一种取代的苯并咪唑酮化合物及包含该化合物的组合物 |
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| CA2599721A1 (en) | 2005-03-04 | 2006-09-14 | Boehringer Ingelheim International Gmbh | Pharmaceutical compositions for the treatment and/or prevention of depression |
| WO2006096439A2 (en) * | 2005-03-04 | 2006-09-14 | Boehringer Ingelheim International Gmbh | Pharmaceutical compositions for the treatment and/or prevention of schizophrenia and related diseases |
| CA2608249A1 (en) * | 2005-05-06 | 2006-11-16 | Boehringer Ingelheim International Gmbh | Method for the treatment of drug abuse with flibanserin |
| US20060258640A1 (en) * | 2005-05-13 | 2006-11-16 | Boehringer Ingelheim International Gmbh | Use of Flibanserin in the treatment of chronic pain |
| JP2008540672A (ja) * | 2005-05-19 | 2008-11-20 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | 病状に起因する性的機能不全の治療方法 |
| US20060264511A1 (en) * | 2005-05-19 | 2006-11-23 | Boehringer Ingelheim International Gmbh | Method for the treatment of drug-induced sexual dysfunction |
| EP2502621A1 (en) | 2005-06-27 | 2012-09-26 | Valeant International (Barbados) SRL | Crystalline forms of bupropion HBr |
| JP2009503020A (ja) * | 2005-08-03 | 2009-01-29 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | 肥満症の治療におけるフリバンセリンの使用 |
| HU227490B1 (en) | 2005-08-26 | 2011-07-28 | Egis Gyogyszergyar Nyilvanosan Muekoedoe Reszvenytarsasag | Sustained release pharmaceutical preparation containing carvedilol |
| JP2009513604A (ja) * | 2005-10-29 | 2009-04-02 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | 月経前障害及び他の女性の性的障害治療用のベンゾイミダゾロン誘導体 |
| US20070123540A1 (en) * | 2005-10-29 | 2007-05-31 | Angelo Ceci | Sexual desire enhancing medicaments comprising benzimidazolone derivatives |
| US20070105869A1 (en) * | 2005-11-08 | 2007-05-10 | Stephane Pollentier | Use of flibanserin for the treatment of pre-menopausal sexual desire disorders |
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| CA2641917A1 (en) * | 2006-02-18 | 2007-08-23 | Boehringer Ingelheim International Gmbh | Pharmaceutical compositions for the treatment of attention deficit hyperactivity disorder comprising flibanserin |
| CA2642101A1 (en) * | 2006-02-20 | 2007-08-30 | Boehringer Ingelheim International Gmbh | Benzimidazolone derivatives for the treatment of urinary incontinence |
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| WO2008000760A1 (en) * | 2006-06-30 | 2008-01-03 | Boehringer Ingelheim International Gmbh | Flibanserin for the treatment of urinary incontinence and related diseases |
| JP2009543839A (ja) | 2006-07-14 | 2009-12-10 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | 女性の性的障害を治療するためのフリバンセリンの使用 |
| WO2008006839A2 (en) * | 2006-07-14 | 2008-01-17 | Boehringer Ingelheim International Gmbh | Combinations of flibanserin with caffeine, process for their preparation and use thereof as medicaments |
| CL2007002214A1 (es) * | 2006-08-14 | 2008-03-07 | Boehringer Ingelheim Int | Composicion farmaceutica en la forma de comprimido, donde al menos la longitud del comprimido en el estado anterior de la aplicacion es al menos 7/12 del diametro pilorico del paciente y despues de ingerirlo en estado alimentado, la longitud del comp |
| AU2007286288A1 (en) * | 2006-08-14 | 2008-02-21 | Boehringer Ingelheim International Gmbh | Formulations of flibanserin and method for manufacturing the same |
| EP2056797A2 (en) | 2006-08-25 | 2009-05-13 | Boehringer Ingelheim International GmbH | Controlled release system and method for manufacturing the same |
| ATE524446T1 (de) | 2006-12-20 | 2011-09-15 | Boehringer Ingelheim Int | Sulfatierte benzimidazolon-derivate mit gemischter serotonin-rezeptor-affinität |
| US20100093754A1 (en) | 2007-03-28 | 2010-04-15 | Boehringer Ingelheim International Gmbh | Pharmaceutical Compositions Comprising Flibanserin and a Further Agent in the Treatment of Sexual Disorders |
| UY31335A1 (es) * | 2007-09-12 | 2009-04-30 | Tratamiento de sintomas vasomotores |
-
2008
- 2008-09-10 UY UY31335A patent/UY31335A1/es not_active Application Discontinuation
- 2008-09-10 PE PE2008001580A patent/PE20091188A1/es not_active Application Discontinuation
- 2008-09-10 CL CL2008002693A patent/CL2008002693A1/es unknown
- 2008-09-11 BR BRPI0816791A patent/BRPI0816791A2/pt not_active IP Right Cessation
- 2008-09-11 WO PCT/EP2008/062011 patent/WO2009034111A1/en not_active Ceased
- 2008-09-11 TW TW097134893A patent/TW200927118A/zh unknown
- 2008-09-11 MX MX2010002032A patent/MX2010002032A/es not_active Application Discontinuation
- 2008-09-11 JP JP2010524478A patent/JP2010539130A/ja active Pending
- 2008-09-11 US US12/675,231 patent/US20110136825A1/en not_active Abandoned
- 2008-09-11 ES ES08803978.9T patent/ES2444707T3/es active Active
- 2008-09-11 CN CN2008801069327A patent/CN101801380B/zh not_active Expired - Fee Related
- 2008-09-11 AU AU2008297104A patent/AU2008297104A1/en not_active Abandoned
- 2008-09-11 AR ARP080103952A patent/AR068416A1/es unknown
- 2008-09-11 EA EA201000433A patent/EA201000433A1/ru unknown
- 2008-09-11 KR KR1020107005191A patent/KR20100059848A/ko not_active Withdrawn
- 2008-09-11 EP EP08803978.9A patent/EP2200614B1/en active Active
- 2008-09-11 CA CA2699414A patent/CA2699414C/en not_active Expired - Fee Related
- 2008-09-11 NZ NZ584183A patent/NZ584183A/en not_active IP Right Cessation
-
2010
- 2010-01-19 ZA ZA201000384A patent/ZA201000384B/xx unknown
- 2010-03-11 TN TNP2010000108A patent/TN2010000108A1/fr unknown
- 2010-03-12 CO CO10029659A patent/CO6260073A2/es not_active Application Discontinuation
- 2010-04-08 MA MA32746A patent/MA31757B1/fr unknown
-
2013
- 2013-03-20 US US13/847,683 patent/US20140005203A1/en not_active Abandoned
-
2014
- 2014-12-26 US US14/583,275 patent/US10166230B2/en active Active
-
2017
- 2017-08-25 US US15/686,665 patent/US9949969B2/en not_active Expired - Fee Related
-
2018
- 2018-11-26 US US16/200,004 patent/US10596170B2/en not_active Expired - Fee Related
-
2020
- 2020-03-05 US US16/810,273 patent/US20200253962A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| US20150250783A1 (en) | 2015-09-10 |
| AR068416A1 (es) | 2009-11-18 |
| US10596170B2 (en) | 2020-03-24 |
| US20110136825A1 (en) | 2011-06-09 |
| MX2010002032A (es) | 2010-03-15 |
| US9949969B2 (en) | 2018-04-24 |
| US20190091219A1 (en) | 2019-03-28 |
| US20140005203A1 (en) | 2014-01-02 |
| US20200253962A1 (en) | 2020-08-13 |
| CL2008002693A1 (es) | 2009-10-16 |
| EA201000433A1 (ru) | 2010-10-29 |
| CN101801380A (zh) | 2010-08-11 |
| WO2009034111A1 (en) | 2009-03-19 |
| UY31335A1 (es) | 2009-04-30 |
| CO6260073A2 (es) | 2011-03-22 |
| TN2010000108A1 (fr) | 2011-09-26 |
| PE20091188A1 (es) | 2009-08-31 |
| NZ584183A (en) | 2012-05-25 |
| MA31757B1 (fr) | 2010-10-01 |
| KR20100059848A (ko) | 2010-06-04 |
| ZA201000384B (en) | 2010-09-29 |
| CN101801380B (zh) | 2013-05-08 |
| CA2699414C (en) | 2016-04-05 |
| US10166230B2 (en) | 2019-01-01 |
| AU2008297104A1 (en) | 2009-03-19 |
| JP2010539130A (ja) | 2010-12-16 |
| EP2200614B1 (en) | 2013-11-27 |
| BRPI0816791A2 (pt) | 2019-09-24 |
| US20180071283A1 (en) | 2018-03-15 |
| CA2699414A1 (en) | 2009-03-19 |
| ES2444707T3 (es) | 2014-02-26 |
| EP2200614A1 (en) | 2010-06-30 |
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