TNSN99007A1 - Composition de mesylate de trovafloxacine et procede pour sa preparation - Google Patents
Composition de mesylate de trovafloxacine et procede pour sa preparationInfo
- Publication number
- TNSN99007A1 TNSN99007A1 TNTNSN99007A TNSN99007A TNSN99007A1 TN SN99007 A1 TNSN99007 A1 TN SN99007A1 TN TNSN99007 A TNTNSN99007 A TN TNSN99007A TN SN99007 A TNSN99007 A TN SN99007A TN SN99007 A1 TNSN99007 A1 TN SN99007A1
- Authority
- TN
- Tunisia
- Prior art keywords
- preparation
- trovafloxacin mesylate
- mesylate composition
- composition
- compositions
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/2833—Organic macromolecular compounds
- A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
- A61K9/2866—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/4375—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a six-membered ring having nitrogen as a ring heteroatom, e.g. quinolizines, naphthyridines, berberine, vincamine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
L'INVENTION CONCERNE DES COMPOSITIONS, NOTAMMENT SOUS FORME DE COMPRIMES, CONTENANT LA FORME POLYMORPHE II DE MESYLATE DE TROVAFLOXACINE ET, EN OUTRE, UN LUBRIFIANT ET DE LA CELLULOSE MICROCRISTALLINE (CM) SERVANT DE DILUANT. ELLE CONCERNE EGALEMENT UN PROCEDE POUR LEUR PREPARATION. UTILISATION DE CES COMPOSITIONS POUR LE TRAITEMENT D'INFECTIONS BACTERIENNES.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US7201398P | 1998-01-21 | 1998-01-21 |
Publications (1)
Publication Number | Publication Date |
---|---|
TNSN99007A1 true TNSN99007A1 (fr) | 2005-11-10 |
Family
ID=22105016
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
TNTNSN99007A TNSN99007A1 (fr) | 1998-01-21 | 1999-01-20 | Composition de mesylate de trovafloxacine et procede pour sa preparation |
Country Status (34)
Country | Link |
---|---|
US (1) | US6187341B1 (fr) |
EP (1) | EP0930068A3 (fr) |
JP (1) | JPH11269072A (fr) |
KR (1) | KR100314977B1 (fr) |
CN (1) | CN1227743A (fr) |
AP (1) | AP1094A (fr) |
AR (1) | AR012780A1 (fr) |
AU (1) | AU758381B2 (fr) |
BG (1) | BG103106A (fr) |
BR (1) | BR9900116A (fr) |
CA (1) | CA2259698C (fr) |
CO (1) | CO4810225A1 (fr) |
DZ (1) | DZ2712A1 (fr) |
EA (1) | EA003247B1 (fr) |
GT (1) | GT199900004A (fr) |
HR (1) | HRP990023A2 (fr) |
HU (1) | HUP9900154A3 (fr) |
ID (1) | ID23735A (fr) |
IL (1) | IL128051A0 (fr) |
IS (1) | IS4947A (fr) |
MA (1) | MA24747A1 (fr) |
NO (1) | NO990243L (fr) |
NZ (1) | NZ333838A (fr) |
OA (1) | OA10958A (fr) |
PA (1) | PA8466701A1 (fr) |
PE (1) | PE20000169A1 (fr) |
PL (1) | PL330981A1 (fr) |
SG (1) | SG70666A1 (fr) |
SK (1) | SK4299A3 (fr) |
TN (1) | TNSN99007A1 (fr) |
TR (1) | TR199900089A2 (fr) |
TW (1) | TW518224B (fr) |
YU (1) | YU2399A (fr) |
ZA (1) | ZA99393B (fr) |
Families Citing this family (20)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IL142642A0 (en) * | 1998-11-10 | 2002-03-10 | Bayer Ag | Pharmaceutical moxifloxacin preparation |
CA2382834A1 (fr) * | 1999-09-20 | 2001-03-29 | Alza Corporation | Procede destine a reduire la transformation polymorphique d'un medicament |
IL148820A0 (en) * | 1999-10-08 | 2002-09-12 | Smithkline Beecham Corp | Fab i inhibitors |
FR2808441B1 (fr) * | 2000-05-04 | 2004-06-18 | Oreal | Utilisation de fibres dans une composition de soin ou de maquillage pour matifier la peau |
DE10031043A1 (de) * | 2000-06-26 | 2002-02-14 | Bayer Ag | Retardzubereitungen von Chinolonantibiotika und Verfahren zu ihrer Herstellung |
WO2003088897A2 (fr) * | 2001-04-06 | 2003-10-30 | Affinium Pharmaceuticals, Inc. | Inhibiteurs de fab i |
EP1396263A1 (fr) * | 2002-08-09 | 2004-03-10 | Warner-Lambert Company | Compositions d'enrobage pour tablettes et caplets |
DK1575951T3 (da) * | 2002-12-06 | 2014-09-15 | Debiopharm Int Sa | Heterocykliske forbindelser, fremgangsmåder til fremstilling deraf og deres anvendelse i terapi |
CN100415284C (zh) * | 2002-12-30 | 2008-09-03 | 毛友昌 | 六味木香片的制备方法 |
EP1608377B1 (fr) | 2003-03-17 | 2008-10-01 | Affinium Pharmaceuticals, Inc. | Compositions comportant plusieurs agents antibiotiques, et leurs procedes de mise en oeuvre |
ES2297067T3 (es) * | 2003-03-19 | 2008-05-01 | The Jordanian Pharmaceutical Manufacturing Co. Ltd. | Composiciones farmaceuticas no higroscopicas que contienen acidos quinolinacarboxilicos de hidratados. |
US8906413B2 (en) * | 2003-05-12 | 2014-12-09 | Supernus Pharmaceuticals, Inc. | Drug formulations having reduced abuse potential |
MXPA06000702A (es) * | 2003-07-23 | 2006-04-11 | Perrigo L Co | Composicion que contiene fibra celulosica. |
JP5087406B2 (ja) | 2004-06-04 | 2012-12-05 | アフィニウム ファーマシューティカルズ, インク. | 治療薬ならびにその製造方法および使用方法 |
EP1809259B1 (fr) * | 2004-10-15 | 2014-12-03 | Supernus Pharmaceuticals, Inc. | Preparations pharmaceutiques pour lesquelles le risque d'abus est reduit |
JP2009518399A (ja) * | 2005-12-05 | 2009-05-07 | アフィニウム ファーマシューティカルズ, インク. | Fabi阻害剤および抗菌剤としてのヘテロ環アクリルアミド化合物 |
WO2008009122A1 (fr) | 2006-07-20 | 2008-01-24 | Affinium Pharmaceuticals, Inc. | Dérivés d'acrylamide en tant qu'inhibiteurs de fab i |
WO2008098374A1 (fr) | 2007-02-16 | 2008-08-21 | Affinium Pharmaceuticals, Inc. | Sels, promédicaments et polymorphes d'inhibiteurs de fab 1 |
DK2861608T3 (da) | 2012-06-19 | 2019-06-24 | Debiopharm Int Sa | Prodrug-derivater af (e)-n-methyl-n-((3-methylbenzofuran-2-yl)methyl)-3-(7-oxo-5,6,7,8-tetrahydro-1,8-naphthyridin-3-yl)acrylamid |
CN108778286A (zh) | 2016-02-26 | 2018-11-09 | 德彪药业国际股份公司 | 用于治疗糖尿病足感染的药物 |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5286754A (en) | 1986-01-21 | 1994-02-15 | Bayer Aktiengesellschaft | Pharmaceutical formulations of ciprofloxacin |
DE3601566A1 (de) * | 1986-01-21 | 1987-07-23 | Bayer Ag | Pharmazeutische zubereitungen von ciprofloxacin |
US4957554A (en) | 1989-08-16 | 1990-09-18 | Minnesota Mining And Manufacturing Company | Dimensionally-controlled ceramics |
DE4120646A1 (de) | 1991-06-22 | 1992-12-24 | Bayer Ag | 7-isoindolinyl-chinolon- und naphthyridoncarbonsaeure-derivate |
CA2229786C (fr) * | 1995-08-29 | 2002-02-19 | David Bruning Joseph | Formes zwitterioniques de trovafloxacine |
-
1999
- 1999-01-11 PA PA19998466701A patent/PA8466701A1/es unknown
- 1999-01-13 EP EP99300258A patent/EP0930068A3/fr not_active Withdrawn
- 1999-01-14 AP APAP/P/1999/001443A patent/AP1094A/en active
- 1999-01-14 IL IL12805199A patent/IL128051A0/xx unknown
- 1999-01-14 TR TR1999/00089A patent/TR199900089A2/xx unknown
- 1999-01-14 SK SK42-99A patent/SK4299A3/sk unknown
- 1999-01-15 ID IDP990036D patent/ID23735A/id unknown
- 1999-01-15 GT GT199900004A patent/GT199900004A/es unknown
- 1999-01-15 MA MA25433A patent/MA24747A1/fr unknown
- 1999-01-15 OA OA9900009A patent/OA10958A/en unknown
- 1999-01-15 PE PE1999000036A patent/PE20000169A1/es not_active Application Discontinuation
- 1999-01-19 CA CA002259698A patent/CA2259698C/fr not_active Expired - Fee Related
- 1999-01-19 IS IS4947A patent/IS4947A/is unknown
- 1999-01-19 JP JP11010298A patent/JPH11269072A/ja active Pending
- 1999-01-19 AR ARP990100191A patent/AR012780A1/es not_active Application Discontinuation
- 1999-01-19 BR BR9900116-0A patent/BR9900116A/pt not_active IP Right Cessation
- 1999-01-20 US US09/233,823 patent/US6187341B1/en not_active Expired - Fee Related
- 1999-01-20 SG SG1999000117A patent/SG70666A1/en unknown
- 1999-01-20 DZ DZ990013A patent/DZ2712A1/fr active
- 1999-01-20 ZA ZA9900393A patent/ZA99393B/xx unknown
- 1999-01-20 AU AU12173/99A patent/AU758381B2/en not_active Ceased
- 1999-01-20 NZ NZ333838A patent/NZ333838A/xx unknown
- 1999-01-20 KR KR1019990001589A patent/KR100314977B1/ko not_active IP Right Cessation
- 1999-01-20 CN CN99101232A patent/CN1227743A/zh active Pending
- 1999-01-20 TN TNTNSN99007A patent/TNSN99007A1/fr unknown
- 1999-01-20 PL PL99330981A patent/PL330981A1/xx unknown
- 1999-01-20 HU HU9900154A patent/HUP9900154A3/hu unknown
- 1999-01-20 NO NO990243A patent/NO990243L/no not_active Application Discontinuation
- 1999-01-20 YU YU2399A patent/YU2399A/sh unknown
- 1999-01-21 HR HR60/072,013A patent/HRP990023A2/hr not_active Application Discontinuation
- 1999-01-21 CO CO99003190A patent/CO4810225A1/es unknown
- 1999-01-21 TW TW088100897A patent/TW518224B/zh not_active IP Right Cessation
- 1999-01-21 EA EA199900046A patent/EA003247B1/ru not_active IP Right Cessation
- 1999-01-21 BG BG103106A patent/BG103106A/xx unknown
Also Published As
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