TNSN99007A1 - Composition de mesylate de trovafloxacine et procede pour sa preparation - Google Patents

Composition de mesylate de trovafloxacine et procede pour sa preparation

Info

Publication number
TNSN99007A1
TNSN99007A1 TNTNSN99007A TNSN99007A TNSN99007A1 TN SN99007 A1 TNSN99007 A1 TN SN99007A1 TN TNSN99007 A TNTNSN99007 A TN TNSN99007A TN SN99007 A TNSN99007 A TN SN99007A TN SN99007 A1 TNSN99007 A1 TN SN99007A1
Authority
TN
Tunisia
Prior art keywords
preparation
trovafloxacin mesylate
mesylate composition
composition
compositions
Prior art date
Application number
TNTNSN99007A
Other languages
English (en)
Inventor
Dale Johnson Alton
Michael Sinko Christopher
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of TNSN99007A1 publication Critical patent/TNSN99007A1/fr

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/286Polysaccharides, e.g. gums; Cyclodextrin
    • A61K9/2866Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4375Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a six-membered ring having nitrogen as a ring heteroatom, e.g. quinolizines, naphthyridines, berberine, vincamine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

L'INVENTION CONCERNE DES COMPOSITIONS, NOTAMMENT SOUS FORME DE COMPRIMES, CONTENANT LA FORME POLYMORPHE II DE MESYLATE DE TROVAFLOXACINE ET, EN OUTRE, UN LUBRIFIANT ET DE LA CELLULOSE MICROCRISTALLINE (CM) SERVANT DE DILUANT. ELLE CONCERNE EGALEMENT UN PROCEDE POUR LEUR PREPARATION. UTILISATION DE CES COMPOSITIONS POUR LE TRAITEMENT D'INFECTIONS BACTERIENNES.
TNTNSN99007A 1998-01-21 1999-01-20 Composition de mesylate de trovafloxacine et procede pour sa preparation TNSN99007A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US7201398P 1998-01-21 1998-01-21

Publications (1)

Publication Number Publication Date
TNSN99007A1 true TNSN99007A1 (fr) 2005-11-10

Family

ID=22105016

Family Applications (1)

Application Number Title Priority Date Filing Date
TNTNSN99007A TNSN99007A1 (fr) 1998-01-21 1999-01-20 Composition de mesylate de trovafloxacine et procede pour sa preparation

Country Status (34)

Country Link
US (1) US6187341B1 (fr)
EP (1) EP0930068A3 (fr)
JP (1) JPH11269072A (fr)
KR (1) KR100314977B1 (fr)
CN (1) CN1227743A (fr)
AP (1) AP1094A (fr)
AR (1) AR012780A1 (fr)
AU (1) AU758381B2 (fr)
BG (1) BG103106A (fr)
BR (1) BR9900116A (fr)
CA (1) CA2259698C (fr)
CO (1) CO4810225A1 (fr)
DZ (1) DZ2712A1 (fr)
EA (1) EA003247B1 (fr)
GT (1) GT199900004A (fr)
HR (1) HRP990023A2 (fr)
HU (1) HUP9900154A3 (fr)
ID (1) ID23735A (fr)
IL (1) IL128051A0 (fr)
IS (1) IS4947A (fr)
MA (1) MA24747A1 (fr)
NO (1) NO990243L (fr)
NZ (1) NZ333838A (fr)
OA (1) OA10958A (fr)
PA (1) PA8466701A1 (fr)
PE (1) PE20000169A1 (fr)
PL (1) PL330981A1 (fr)
SG (1) SG70666A1 (fr)
SK (1) SK4299A3 (fr)
TN (1) TNSN99007A1 (fr)
TR (1) TR199900089A2 (fr)
TW (1) TW518224B (fr)
YU (1) YU2399A (fr)
ZA (1) ZA99393B (fr)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL142642A0 (en) * 1998-11-10 2002-03-10 Bayer Ag Pharmaceutical moxifloxacin preparation
CA2382834A1 (fr) * 1999-09-20 2001-03-29 Alza Corporation Procede destine a reduire la transformation polymorphique d'un medicament
IL148820A0 (en) * 1999-10-08 2002-09-12 Smithkline Beecham Corp Fab i inhibitors
FR2808441B1 (fr) * 2000-05-04 2004-06-18 Oreal Utilisation de fibres dans une composition de soin ou de maquillage pour matifier la peau
DE10031043A1 (de) * 2000-06-26 2002-02-14 Bayer Ag Retardzubereitungen von Chinolonantibiotika und Verfahren zu ihrer Herstellung
WO2003088897A2 (fr) * 2001-04-06 2003-10-30 Affinium Pharmaceuticals, Inc. Inhibiteurs de fab i
EP1396263A1 (fr) * 2002-08-09 2004-03-10 Warner-Lambert Company Compositions d'enrobage pour tablettes et caplets
DK1575951T3 (da) * 2002-12-06 2014-09-15 Debiopharm Int Sa Heterocykliske forbindelser, fremgangsmåder til fremstilling deraf og deres anvendelse i terapi
CN100415284C (zh) * 2002-12-30 2008-09-03 毛友昌 六味木香片的制备方法
EP1608377B1 (fr) 2003-03-17 2008-10-01 Affinium Pharmaceuticals, Inc. Compositions comportant plusieurs agents antibiotiques, et leurs procedes de mise en oeuvre
ES2297067T3 (es) * 2003-03-19 2008-05-01 The Jordanian Pharmaceutical Manufacturing Co. Ltd. Composiciones farmaceuticas no higroscopicas que contienen acidos quinolinacarboxilicos de hidratados.
US8906413B2 (en) * 2003-05-12 2014-12-09 Supernus Pharmaceuticals, Inc. Drug formulations having reduced abuse potential
MXPA06000702A (es) * 2003-07-23 2006-04-11 Perrigo L Co Composicion que contiene fibra celulosica.
JP5087406B2 (ja) 2004-06-04 2012-12-05 アフィニウム ファーマシューティカルズ, インク. 治療薬ならびにその製造方法および使用方法
EP1809259B1 (fr) * 2004-10-15 2014-12-03 Supernus Pharmaceuticals, Inc. Preparations pharmaceutiques pour lesquelles le risque d'abus est reduit
JP2009518399A (ja) * 2005-12-05 2009-05-07 アフィニウム ファーマシューティカルズ, インク. Fabi阻害剤および抗菌剤としてのヘテロ環アクリルアミド化合物
WO2008009122A1 (fr) 2006-07-20 2008-01-24 Affinium Pharmaceuticals, Inc. Dérivés d'acrylamide en tant qu'inhibiteurs de fab i
WO2008098374A1 (fr) 2007-02-16 2008-08-21 Affinium Pharmaceuticals, Inc. Sels, promédicaments et polymorphes d'inhibiteurs de fab 1
DK2861608T3 (da) 2012-06-19 2019-06-24 Debiopharm Int Sa Prodrug-derivater af (e)-n-methyl-n-((3-methylbenzofuran-2-yl)methyl)-3-(7-oxo-5,6,7,8-tetrahydro-1,8-naphthyridin-3-yl)acrylamid
CN108778286A (zh) 2016-02-26 2018-11-09 德彪药业国际股份公司 用于治疗糖尿病足感染的药物

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5286754A (en) 1986-01-21 1994-02-15 Bayer Aktiengesellschaft Pharmaceutical formulations of ciprofloxacin
DE3601566A1 (de) * 1986-01-21 1987-07-23 Bayer Ag Pharmazeutische zubereitungen von ciprofloxacin
US4957554A (en) 1989-08-16 1990-09-18 Minnesota Mining And Manufacturing Company Dimensionally-controlled ceramics
DE4120646A1 (de) 1991-06-22 1992-12-24 Bayer Ag 7-isoindolinyl-chinolon- und naphthyridoncarbonsaeure-derivate
CA2229786C (fr) * 1995-08-29 2002-02-19 David Bruning Joseph Formes zwitterioniques de trovafloxacine

Also Published As

Publication number Publication date
EA003247B1 (ru) 2003-02-27
ID23735A (id) 2000-05-11
KR19990068014A (ko) 1999-08-25
PL330981A1 (en) 1999-08-02
IL128051A0 (en) 1999-11-30
ZA99393B (en) 2000-07-21
CA2259698A1 (fr) 1999-07-21
MA24747A1 (fr) 1999-10-01
HUP9900154A3 (en) 2000-12-28
EP0930068A3 (fr) 1999-12-22
BG103106A (en) 1999-08-31
DZ2712A1 (fr) 2003-09-01
CO4810225A1 (es) 1999-06-30
AP1094A (en) 2002-08-19
PA8466701A1 (es) 2000-09-29
AU1217399A (en) 1999-08-12
AP9901443A0 (en) 1999-03-31
OA10958A (en) 2001-10-31
SK4299A3 (en) 2000-06-12
HUP9900154A2 (hu) 1999-09-28
US6187341B1 (en) 2001-02-13
SG70666A1 (en) 2000-02-22
YU2399A (sh) 2002-06-19
GT199900004A (es) 2000-07-08
TR199900089A3 (tr) 1999-10-21
NO990243D0 (no) 1999-01-20
TW518224B (en) 2003-01-21
NZ333838A (en) 2000-03-27
IS4947A (is) 1999-07-22
HU9900154D0 (en) 1999-03-29
EA199900046A3 (ru) 1999-12-29
EP0930068A2 (fr) 1999-07-21
KR100314977B1 (ko) 2001-11-24
PE20000169A1 (es) 2000-03-10
NO990243L (no) 1999-07-22
AU758381B2 (en) 2003-03-20
JPH11269072A (ja) 1999-10-05
HRP990023A2 (en) 1999-08-31
TR199900089A2 (xx) 1999-10-21
AR012780A1 (es) 2000-11-08
BR9900116A (pt) 2000-05-02
CN1227743A (zh) 1999-09-08
CA2259698C (fr) 2003-04-15
EA199900046A2 (ru) 1999-08-26

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