TNSN05244A1 - Novel diphenyl azetidinone with improved physiological characteristics, corresponding production method, medicaments containing said compound and use of the latter - Google Patents

Novel diphenyl azetidinone with improved physiological characteristics, corresponding production method, medicaments containing said compound and use of the latter

Info

Publication number
TNSN05244A1
TNSN05244A1 TNP2005000244A TNSN05244A TNSN05244A1 TN SN05244 A1 TNSN05244 A1 TN SN05244A1 TN P2005000244 A TNP2005000244 A TN P2005000244A TN SN05244 A TNSN05244 A TN SN05244A TN SN05244 A1 TNSN05244 A1 TN SN05244A1
Authority
TN
Tunisia
Prior art keywords
compound
production method
medicaments containing
physiological characteristics
corresponding production
Prior art date
Application number
TNP2005000244A
Other languages
English (en)
Inventor
Gerhard Jaehne
Wendelin Frick
Andreas Lindenschmidt
Stefanie Flohr
Hubert Heuer
Hans-Ludwig Schaefer
Werner Kramer
Eric Galia
Heiner Glombik
Original Assignee
Aventis Pharma Deutschland Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma Deutschland Gmbh filed Critical Aventis Pharma Deutschland Gmbh
Publication of TNSN05244A1 publication Critical patent/TNSN05244A1/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C233/00—Carboxylic acid amides
    • C07C233/01—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C233/16—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms
    • C07C233/17—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom
    • C07C233/18—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom having the carbon atom of the carboxamide group bound to a hydrogen atom or to a carbon atom of an acyclic saturated carbon skeleton
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/397—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having four-membered rings, e.g. azetidine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D205/08—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Diabetes (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
TNP2005000244A 2003-04-01 2005-09-30 Novel diphenyl azetidinone with improved physiological characteristics, corresponding production method, medicaments containing said compound and use of the latter TNSN05244A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10314610A DE10314610A1 (de) 2003-04-01 2003-04-01 Neues Diphenylazetidinon mit verbesserten physiologischen Eigenschaften, Verfahren zu dessen Herstellung, diese Verbindungen enthaltende Arzneimittel und dessen Verwendung
PCT/EP2004/002690 WO2004087655A1 (de) 2003-04-01 2004-03-16 Neues diphenylazetidinon mit verbesserten physiologischen eigenschaften, verfahren zu dessen herstellung, diese verbindungen enthaltende arzneimittel und dessen verwendung

Publications (1)

Publication Number Publication Date
TNSN05244A1 true TNSN05244A1 (en) 2007-06-11

Family

ID=33103147

Family Applications (1)

Application Number Title Priority Date Filing Date
TNP2005000244A TNSN05244A1 (en) 2003-04-01 2005-09-30 Novel diphenyl azetidinone with improved physiological characteristics, corresponding production method, medicaments containing said compound and use of the latter

Country Status (44)

Country Link
US (2) US7205290B2 (ar)
EP (2) EP1613589B1 (ar)
JP (1) JP2006522040A (ar)
KR (1) KR20050119180A (ar)
CN (2) CN100361970C (ar)
AR (1) AR043783A1 (ar)
AT (2) ATE386020T1 (ar)
AU (1) AU2004226287B2 (ar)
BR (1) BRPI0408920A (ar)
CA (1) CA2520689A1 (ar)
CL (1) CL43489B (ar)
CR (1) CR7995A (ar)
CY (2) CY1107398T1 (ar)
DE (3) DE10314610A1 (ar)
DK (2) DK1613589T3 (ar)
EC (1) ECSP056071A (ar)
ES (2) ES2298731T3 (ar)
GT (1) GT200400058A (ar)
HK (1) HK1087697A1 (ar)
HN (1) HN2004000109A (ar)
HR (1) HRP20050870A2 (ar)
JO (1) JO2493B1 (ar)
MA (1) MA27753A1 (ar)
ME (1) MEP41408A (ar)
MX (1) MXPA05010128A (ar)
MY (1) MY136269A (ar)
NI (1) NI200500164A (ar)
NO (1) NO20055001L (ar)
NZ (1) NZ542751A (ar)
PA (1) PA8599401A1 (ar)
PE (1) PE20050011A1 (ar)
PL (2) PL1613589T3 (ar)
PT (2) PT1613589E (ar)
RS (1) RS51146B (ar)
RU (1) RU2334737C2 (ar)
SA (1) SA04250154B1 (ar)
SI (2) SI1862455T1 (ar)
SV (1) SV2004001756A (ar)
TN (1) TNSN05244A1 (ar)
TW (1) TW200504009A (ar)
UA (1) UA80754C2 (ar)
UY (1) UY28253A1 (ar)
WO (1) WO2004087655A1 (ar)
ZA (1) ZA200506708B (ar)

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RU2009108280A (ru) 2006-08-08 2010-09-20 Санофи-Авентис (Fr) Ариламиноарилалкилзамещенные имидазолидин-2,4-дионы, способы их получения, содержащие эти соединения лекарственные средства и их применение
DE102007029612A1 (de) * 2007-06-27 2009-01-08 Sanofi-Aventis Deutschland Gmbh Verfahren zur Herstellung von Pentahydroxyhexylcarbamoylundekan- säurebenzylester
US20080319221A1 (en) * 2007-06-22 2008-12-25 Bernd Junker Esters of Pentahydroxyhexylcarbamoyl Alkanoic Acids
US20080319218A1 (en) * 2007-06-22 2008-12-25 Andreas Haubrich Processes for Making and Using Benzyl Pentahydroxyhexylcarbamoylundecanoate
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WO2009112203A1 (de) * 2008-03-14 2009-09-17 Sanofi-Aventis Deutschland Gmbh Verfahren zur herstellung eines diphenylazetidinons
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WO2012120058A1 (de) 2011-03-08 2012-09-13 Sanofi Mit benzyl- oder heteromethylengruppen substituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung
US8828995B2 (en) 2011-03-08 2014-09-09 Sanofi Branched oxathiazine derivatives, method for the production thereof, use thereof as medicine and drug containing said derivatives and use thereof
EP2683700B1 (de) 2011-03-08 2015-02-18 Sanofi Tetrasubstituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung
EP2683699B1 (de) 2011-03-08 2015-06-24 Sanofi Di- und trisubstituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung
EP2683702B1 (de) 2011-03-08 2014-12-24 Sanofi Neue substituierte phenyl-oxathiazinderivate, verfahren zu deren herstellung, diese verbindungen enthaltende arzneimittel und deren verwendung
US8901114B2 (en) 2011-03-08 2014-12-02 Sanofi Oxathiazine derivatives substituted with carbocycles or heterocycles, method for producing same, drugs containing said compounds, and use thereof
EP2567959B1 (en) 2011-09-12 2014-04-16 Sanofi 6-(4-hydroxy-phenyl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
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Also Published As

Publication number Publication date
NO20055001L (no) 2005-10-27
HRP20050870A2 (en) 2006-10-31
CN101139306A (zh) 2008-03-12
GT200400058A (es) 2004-11-10
ECSP056071A (es) 2006-01-27
CA2520689A1 (en) 2004-10-14
PT1613589E (pt) 2008-03-27
SI1862455T1 (sl) 2009-06-30
UA80754C2 (en) 2007-10-25
JP2006522040A (ja) 2006-09-28
WO2004087655A1 (de) 2004-10-14
AU2004226287B2 (en) 2010-03-18
CY1109055T1 (el) 2014-07-02
NI200500164A (es) 2006-01-11
KR20050119180A (ko) 2005-12-20
DE10314610A1 (de) 2004-11-04
BRPI0408920A (pt) 2006-03-28
EP1862455A3 (de) 2007-12-12
RS20050719A (en) 2008-04-04
PT1862455E (pt) 2009-04-23
PL1613589T3 (pl) 2008-07-31
RU2005133631A (ru) 2006-03-10
HK1087697A1 (en) 2006-10-20
UY28253A1 (es) 2004-11-08
EP1862455A2 (de) 2007-12-05
RS51146B (sr) 2010-10-31
CL43489B (es) 2005-01-21
MY136269A (en) 2008-09-30
PE20050011A1 (es) 2005-02-28
DE502004006195D1 (de) 2008-03-27
AU2004226287A1 (en) 2004-10-14
MEP41408A (en) 2011-02-10
MA27753A1 (fr) 2006-02-01
US7772429B2 (en) 2010-08-10
EP1613589A1 (de) 2006-01-11
CN1768034A (zh) 2006-05-03
SI1613589T1 (sl) 2008-06-30
DK1862455T3 (da) 2009-06-02
AR043783A1 (es) 2005-08-10
US20070197498A1 (en) 2007-08-23
EP1862455B1 (de) 2009-02-25
ATE423766T1 (de) 2009-03-15
NZ542751A (en) 2007-05-31
DK1613589T3 (da) 2008-06-09
US7205290B2 (en) 2007-04-17
EP1613589B1 (de) 2008-02-13
ES2298731T3 (es) 2008-05-16
CR7995A (es) 2006-09-22
US20050020563A1 (en) 2005-01-27
SV2004001756A (es) 2004-11-18
SA04250154B1 (ar) 2007-10-29
CY1107398T1 (el) 2012-12-19
JO2493B1 (ar) 2009-10-05
PL1862455T3 (pl) 2009-07-31
ZA200506708B (en) 2007-01-31
PA8599401A1 (es) 2004-10-08
ATE386020T1 (de) 2008-03-15
HN2004000109A (es) 2008-02-21
MXPA05010128A (es) 2005-11-16
RU2334737C2 (ru) 2008-09-27
ES2322876T3 (es) 2009-06-30
CN100361970C (zh) 2008-01-16
TW200504009A (en) 2005-02-01
DE502004009059D1 (de) 2009-04-09

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