TNSN01149A1 - Spiro-pyrimidine-2,4,6-triones inhibitrices de metalloproteinases, et compositions les contenant. - Google Patents

Spiro-pyrimidine-2,4,6-triones inhibitrices de metalloproteinases, et compositions les contenant.

Info

Publication number
TNSN01149A1
TNSN01149A1 TNTNSN01149A TNSN01149A TNSN01149A1 TN SN01149 A1 TNSN01149 A1 TN SN01149A1 TN TNSN01149 A TNTNSN01149 A TN TNSN01149A TN SN01149 A TNSN01149 A TN SN01149A TN SN01149 A1 TNSN01149 A1 TN SN01149A1
Authority
TN
Tunisia
Prior art keywords
compositions containing
inhibitors
triones
metalloproteinases
spiro
Prior art date
Application number
TNTNSN01149A
Other languages
English (en)
French (fr)
Inventor
Scott Bronk Brian
Carl Noe Mark
James Wythes Martin
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of TNSN01149A1 publication Critical patent/TNSN01149A1/fr

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/10Spiro-condensed systems
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    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/10Spiro-condensed systems

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  • Pulmonology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Diabetes (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Ophthalmology & Optometry (AREA)
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TNTNSN01149A 2000-10-26 2001-10-25 Spiro-pyrimidine-2,4,6-triones inhibitrices de metalloproteinases, et compositions les contenant. TNSN01149A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US24338900P 2000-10-26 2000-10-26

Publications (1)

Publication Number Publication Date
TNSN01149A1 true TNSN01149A1 (fr) 2005-11-10

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Application Number Title Priority Date Filing Date
TNTNSN01149A TNSN01149A1 (fr) 2000-10-26 2001-10-25 Spiro-pyrimidine-2,4,6-triones inhibitrices de metalloproteinases, et compositions les contenant.

Country Status (32)

Country Link
EP (1) EP1332146A2 (hr)
JP (1) JP2004518635A (hr)
KR (1) KR20040004412A (hr)
CN (1) CN1501937A (hr)
AP (1) AP2001002318A0 (hr)
AR (1) AR035069A1 (hr)
AU (1) AU2002210813A1 (hr)
BG (1) BG107653A (hr)
BR (1) BR0114913A (hr)
CA (1) CA2425283A1 (hr)
CZ (1) CZ20031083A3 (hr)
EA (1) EA005762B1 (hr)
EC (1) ECSP034567A (hr)
EE (1) EE200300196A (hr)
GT (1) GT200100213A (hr)
HN (1) HN2001000244A (hr)
HR (1) HRP20030332A2 (hr)
HU (1) HUP0301577A3 (hr)
IL (1) IL154948A0 (hr)
IS (1) IS6762A (hr)
MA (1) MA26957A1 (hr)
MX (1) MXPA03003735A (hr)
NO (1) NO20031853L (hr)
OA (1) OA12529A (hr)
PA (1) PA8531401A1 (hr)
PE (1) PE20020589A1 (hr)
PL (1) PL366201A1 (hr)
SK (1) SK4972003A3 (hr)
SV (1) SV2003000705A (hr)
TN (1) TNSN01149A1 (hr)
WO (1) WO2002034753A2 (hr)
ZA (1) ZA200302190B (hr)

Families Citing this family (36)

* Cited by examiner, † Cited by third party
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DOP2002000332A (es) 2001-02-14 2002-08-30 Warner Lambert Co Inhibidores de piridina de metaloproteinasas de la matriz
DOP2002000333A (es) 2001-02-14 2002-09-30 Warner Lambert Co Derivados de acido isoftalico como inhibidores de metaloproteinasas de la matriz
EP1368323B1 (en) 2001-02-14 2010-06-30 Warner-Lambert Company LLC Pyrimidine matrix metalloproteinase inhibitors
PA8539501A1 (es) 2001-02-14 2002-09-30 Warner Lambert Co Compuestos triazolo como inhibidores de mmp
ES2231708T3 (es) 2001-02-14 2005-05-16 Warner-Lambert Company Llc Benzotiadicinas inhibidoras de metaloproteinasa de matriz.
US6924276B2 (en) 2001-09-10 2005-08-02 Warner-Lambert Company Diacid-substituted heteroaryl derivatives as matrix metalloproteinase inhibitors
WO2003032999A1 (en) 2001-10-12 2003-04-24 Warner-Lambert Company Llc Alkyne matrix metalloproteinase inhibitors
US6962922B2 (en) 2001-10-12 2005-11-08 Warner-Lambert Company Llc Alkynylated quinazoline compounds
US6894057B2 (en) 2002-03-08 2005-05-17 Warner-Lambert Company Oxo-azabicyclic compounds
WO2003091252A1 (en) * 2002-04-25 2003-11-06 Bristol-Myers Squibb Company Spirobarbituric acid derivatives useful as inhibitors of matrix metalloproteases
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