SV2003000705A - Inhibidores de espiropirimidin-2,4,6-triona metaloproteinasas pc11074/700021/bb - Google Patents

Inhibidores de espiropirimidin-2,4,6-triona metaloproteinasas pc11074/700021/bb

Info

Publication number
SV2003000705A
SV2003000705A SV2001000705A SV2001000705A SV2003000705A SV 2003000705 A SV2003000705 A SV 2003000705A SV 2001000705 A SV2001000705 A SV 2001000705A SV 2001000705 A SV2001000705 A SV 2001000705A SV 2003000705 A SV2003000705 A SV 2003000705A
Authority
SV
El Salvador
Prior art keywords
spiropirimidin
triona
metaloproteinases
inhibitors
formula
Prior art date
Application number
SV2001000705A
Other languages
English (en)
Spanish (es)
Inventor
Brian Scott Bronk
Mark Carl Noe
Martin James Wythes
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of SV2003000705A publication Critical patent/SV2003000705A/es

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    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/10Spiro-condensed systems
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    • C07DHETEROCYCLIC COMPOUNDS
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    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/10Spiro-condensed systems

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  • Pulmonology (AREA)
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  • Diabetes (AREA)
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SV2001000705A 2000-10-26 2001-10-25 Inhibidores de espiropirimidin-2,4,6-triona metaloproteinasas pc11074/700021/bb SV2003000705A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US24338900P 2000-10-26 2000-10-26

Publications (1)

Publication Number Publication Date
SV2003000705A true SV2003000705A (es) 2003-01-13

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SV2001000705A SV2003000705A (es) 2000-10-26 2001-10-25 Inhibidores de espiropirimidin-2,4,6-triona metaloproteinasas pc11074/700021/bb

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Country Link
EP (1) EP1332146A2 (hr)
JP (1) JP2004518635A (hr)
KR (1) KR20040004412A (hr)
CN (1) CN1501937A (hr)
AP (1) AP2001002318A0 (hr)
AR (1) AR035069A1 (hr)
AU (1) AU2002210813A1 (hr)
BG (1) BG107653A (hr)
BR (1) BR0114913A (hr)
CA (1) CA2425283A1 (hr)
CZ (1) CZ20031083A3 (hr)
EA (1) EA005762B1 (hr)
EC (1) ECSP034567A (hr)
EE (1) EE200300196A (hr)
GT (1) GT200100213A (hr)
HN (1) HN2001000244A (hr)
HR (1) HRP20030332A2 (hr)
HU (1) HUP0301577A3 (hr)
IL (1) IL154948A0 (hr)
IS (1) IS6762A (hr)
MA (1) MA26957A1 (hr)
MX (1) MXPA03003735A (hr)
NO (1) NO20031853L (hr)
OA (1) OA12529A (hr)
PA (1) PA8531401A1 (hr)
PE (1) PE20020589A1 (hr)
PL (1) PL366201A1 (hr)
SK (1) SK4972003A3 (hr)
SV (1) SV2003000705A (hr)
TN (1) TNSN01149A1 (hr)
WO (1) WO2002034753A2 (hr)
ZA (1) ZA200302190B (hr)

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DOP2002000332A (es) 2001-02-14 2002-08-30 Warner Lambert Co Inhibidores de piridina de metaloproteinasas de la matriz
DOP2002000333A (es) 2001-02-14 2002-09-30 Warner Lambert Co Derivados de acido isoftalico como inhibidores de metaloproteinasas de la matriz
EP1368323B1 (en) 2001-02-14 2010-06-30 Warner-Lambert Company LLC Pyrimidine matrix metalloproteinase inhibitors
PA8539501A1 (es) 2001-02-14 2002-09-30 Warner Lambert Co Compuestos triazolo como inhibidores de mmp
ES2231708T3 (es) 2001-02-14 2005-05-16 Warner-Lambert Company Llc Benzotiadicinas inhibidoras de metaloproteinasa de matriz.
US6924276B2 (en) 2001-09-10 2005-08-02 Warner-Lambert Company Diacid-substituted heteroaryl derivatives as matrix metalloproteinase inhibitors
WO2003032999A1 (en) 2001-10-12 2003-04-24 Warner-Lambert Company Llc Alkyne matrix metalloproteinase inhibitors
US6962922B2 (en) 2001-10-12 2005-11-08 Warner-Lambert Company Llc Alkynylated quinazoline compounds
US6894057B2 (en) 2002-03-08 2005-05-17 Warner-Lambert Company Oxo-azabicyclic compounds
WO2003091252A1 (en) * 2002-04-25 2003-11-06 Bristol-Myers Squibb Company Spirobarbituric acid derivatives useful as inhibitors of matrix metalloproteases
WO2003091258A1 (en) * 2002-04-26 2003-11-06 Pfizer Products Inc. N-substituted-heteroaryloxy-aryl-spiro-pyrimidine-2,4,6-trione metalloproteinase inhibitors
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