SU1301317A3 - Способ получени 3-кето- @ -стероидов,замещенных в положении 7 - Google Patents

Способ получени 3-кето- @ -стероидов,замещенных в положении 7 Download PDF

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Publication number
SU1301317A3
SU1301317A3 SU813366202A SU3366202A SU1301317A3 SU 1301317 A3 SU1301317 A3 SU 1301317A3 SU 813366202 A SU813366202 A SU 813366202A SU 3366202 A SU3366202 A SU 3366202A SU 1301317 A3 SU1301317 A3 SU 1301317A3
Authority
SU
USSR - Soviet Union
Prior art keywords
product
group
free
alkali metal
solution
Prior art date
Application number
SU813366202A
Other languages
English (en)
Russian (ru)
Inventor
Неделек Люсьен
Торелли Весперто
Филиберт Даниэль
Original Assignee
Руссель Юклаф (Фирма)
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Руссель Юклаф (Фирма) filed Critical Руссель Юклаф (Фирма)
Application granted granted Critical
Publication of SU1301317A3 publication Critical patent/SU1301317A3/ru

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/0088—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 containing unsubstituted amino radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/10—Antioedematous agents; Diuretics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0003—Androstane derivatives
    • C07J1/0033—Androstane derivatives substituted in position 17 alfa and 17 beta
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0051—Estrane derivatives
    • C07J1/0081—Substituted in position 17 alfa and 17 beta
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J21/00—Normal steroids containing carbon, hydrogen, halogen or oxygen having an oxygen-containing hetero ring spiro-condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J21/001—Lactones
    • C07J21/003—Lactones at position 17
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J51/00—Normal steroids with unmodified cyclopenta(a)hydrophenanthrene skeleton not provided for in groups C07J1/00 - C07J43/00

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Superconductors And Manufacturing Methods Therefor (AREA)
SU813366202A 1980-12-23 1981-12-17 Способ получени 3-кето- @ -стероидов,замещенных в положении 7 SU1301317A3 (ru)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8027272A FR2496669A1 (fr) 1980-12-23 1980-12-23 Nouveaux derives steroides 3-ceto4 ou1-4 substitues en position 7, leur procede de preparation et leur application comme medicaments

Publications (1)

Publication Number Publication Date
SU1301317A3 true SU1301317A3 (ru) 1987-03-30

Family

ID=9249374

Family Applications (1)

Application Number Title Priority Date Filing Date
SU813366202A SU1301317A3 (ru) 1980-12-23 1981-12-17 Способ получени 3-кето- @ -стероидов,замещенных в положении 7

Country Status (19)

Country Link
US (1) US4396614A ( )
EP (1) EP0055170B1 ( )
JP (1) JPS57163399A ( )
KR (1) KR870001937B1 ( )
AT (1) ATE10004T1 ( )
AU (1) AU549260B2 ( )
CA (1) CA1196910A ( )
DE (1) DE3166872D1 ( )
DK (1) DK569281A ( )
ES (2) ES8401989A1 ( )
FI (1) FI77463C ( )
FR (1) FR2496669A1 ( )
GR (1) GR77629B ( )
HU (1) HU184974B ( )
IE (1) IE52462B1 ( )
IL (1) IL64503A0 ( )
PT (1) PT74184B ( )
SU (1) SU1301317A3 ( )
ZA (1) ZA818673B ( )

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4501695A (en) * 1983-05-16 1985-02-26 The Upjohn Company Spironalactone process
FR2596395B1 (fr) * 1986-03-26 1989-05-26 Roussel Uclaf Nouveaux steroides comportant un cycle spirannique en position 17, leur procede de preparation, leur application comme medicaments et les compositions les renfermant
US5276023A (en) * 1989-08-08 1994-01-04 Roussel Uclaf 19-nor-steroid esters
WO2008137038A1 (en) 2007-05-03 2008-11-13 Yale University Locally active 'soft' antiandrogens

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3053840A (en) * 1960-06-23 1962-09-11 Searle & Co 11-oxygenated polydehydro 17-carboxyethyl-9-halo-17-hydroxyandrostan-3-one lactones
BE787940A (fr) * 1971-08-25 1973-02-26 Searle & Co Nouveaux medicaments diuretiques et hypotenseurs et procede de leur preparation
US3845041A (en) * 1973-12-26 1974-10-29 Searle & Co 7-halomethyl-17-hydroxy-3-oxo-17alpha-pregn-4-ene-21-carboxylic acid gamma-lactones
FR2451923A1 (fr) * 1979-03-22 1980-10-17 Roussel Uclaf Nouveaux derives steroides 7-alkyles, leur procede de preparation et leur application comme medicament

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
Патент US № 4258039, кл. 4241241, опублик. 24.03.81. *

Also Published As

Publication number Publication date
FR2496669A1 (fr) 1982-06-25
FI77463B (fi) 1988-11-30
EP0055170A1 (fr) 1982-06-30
FI814109L (fi) 1982-06-24
AU549260B2 (en) 1986-01-23
FI77463C (fi) 1989-03-10
KR870001937B1 (ko) 1987-10-22
CA1196910A (fr) 1985-11-19
ATE10004T1 (de) 1984-11-15
AU7877281A (en) 1982-07-01
US4396614A (en) 1983-08-02
DK569281A (da) 1982-06-24
ES516143A0 (es) 1983-08-01
FR2496669B1 ( ) 1983-10-28
PT74184A (fr) 1982-01-01
IL64503A0 (en) 1982-03-31
IE52462B1 (en) 1987-11-11
GR77629B ( ) 1984-09-25
ES507890A0 (es) 1984-01-01
ES8401989A1 (es) 1984-01-01
PT74184B (fr) 1984-01-05
KR830007713A (ko) 1983-11-04
ZA818673B (en) 1982-10-27
JPS57163399A (en) 1982-10-07
DE3166872D1 (en) 1984-11-29
JPH0133115B2 ( ) 1989-07-11
EP0055170B1 (fr) 1984-10-24
ES8307837A1 (es) 1983-08-01
IE813077L (en) 1982-06-23
HU184974B (en) 1984-11-28

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