SK57494A3 - 5-aminopyrazine-2-carboxamide derivatives, method of their preparation and pharmaceutical composition containing these derivatives - Google Patents

5-aminopyrazine-2-carboxamide derivatives, method of their preparation and pharmaceutical composition containing these derivatives Download PDF

Info

Publication number
SK57494A3
SK57494A3 SK574-94A SK57494A SK57494A3 SK 57494 A3 SK57494 A3 SK 57494A3 SK 57494 A SK57494 A SK 57494A SK 57494 A3 SK57494 A3 SK 57494A3
Authority
SK
Slovakia
Prior art keywords
group
formula
compound
carboxamide
mol
Prior art date
Application number
SK574-94A
Other languages
English (en)
Slovak (sk)
Inventor
Pascal George
Benoit Marabout
Jacques Froissant
Original Assignee
Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synthelabo filed Critical Synthelabo
Publication of SK57494A3 publication Critical patent/SK57494A3/sk

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/02Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/08Drugs for disorders of the urinary system of the prostate
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D241/00Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/02Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
    • C07D241/10Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
    • C07D241/14Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D241/24Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D241/26Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals with nitrogen atoms directly attached to ring carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Urology & Nephrology (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
SK574-94A 1993-05-17 1994-05-16 5-aminopyrazine-2-carboxamide derivatives, method of their preparation and pharmaceutical composition containing these derivatives SK57494A3 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9305930A FR2705344B1 (fr) 1993-05-17 1993-05-17 Dérivés de 2-aminopyrazine-5-carboxamide, leur préparation et leur application en thérapeutique.

Publications (1)

Publication Number Publication Date
SK57494A3 true SK57494A3 (en) 1995-07-11

Family

ID=9447217

Family Applications (1)

Application Number Title Priority Date Filing Date
SK574-94A SK57494A3 (en) 1993-05-17 1994-05-16 5-aminopyrazine-2-carboxamide derivatives, method of their preparation and pharmaceutical composition containing these derivatives

Country Status (19)

Country Link
US (1) US5420130A (ru)
EP (1) EP0625514B1 (ru)
JP (1) JPH06329645A (ru)
CN (1) CN1104637A (ru)
AT (1) ATE183742T1 (ru)
AU (1) AU671361B2 (ru)
CA (1) CA2123668A1 (ru)
CZ (1) CZ283499B6 (ru)
DE (1) DE69420179D1 (ru)
FI (1) FI942265A (ru)
FR (1) FR2705344B1 (ru)
HU (1) HUT69711A (ru)
IL (1) IL109655A (ru)
NO (1) NO941830L (ru)
NZ (1) NZ260531A (ru)
PL (1) PL173309B1 (ru)
RU (1) RU2128176C1 (ru)
SK (1) SK57494A3 (ru)
ZA (1) ZA943353B (ru)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1075486A1 (en) * 1998-05-06 2001-02-14 Duke University Method of treating bladder and lower urinary tract syndromes
PL200955B1 (pl) 1998-08-20 2009-02-27 Toyama Chemical Co Ltd Przeciwwirusowa kompozycja farmaceutyczna i jej zastosowanie oraz zawierająca azot heterocykliczna pochodna karboksamidu

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4041032A (en) * 1974-01-16 1977-08-09 Yamanouchi Pharmaceutical Co., Ltd. Pyrazine derivatives
FR2656609B1 (fr) * 1989-12-28 1992-03-27 Synthelabo Derives de 2-aminopyrimidine-4-carboxamide, leur preparation et leur application en therapeutique.

Also Published As

Publication number Publication date
FI942265A0 (fi) 1994-05-16
CA2123668A1 (en) 1994-11-18
PL173309B1 (pl) 1998-02-27
AU671361B2 (en) 1996-08-22
HU9401512D0 (en) 1994-08-29
HUT69711A (en) 1995-09-28
IL109655A0 (en) 1994-08-26
US5420130A (en) 1995-05-30
FR2705344A1 (fr) 1994-11-25
CZ119594A3 (en) 1994-12-15
ATE183742T1 (de) 1999-09-15
NO941830D0 (no) 1994-05-16
JPH06329645A (ja) 1994-11-29
RU2128176C1 (ru) 1999-03-27
NO941830L (no) 1994-11-18
NZ260531A (en) 1995-10-26
AU6312694A (en) 1994-11-24
FR2705344B1 (fr) 1995-06-30
FI942265A (fi) 1994-11-18
ZA943353B (en) 1995-03-28
DE69420179D1 (de) 1999-09-30
EP0625514B1 (fr) 1999-08-25
CN1104637A (zh) 1995-07-05
EP0625514A1 (fr) 1994-11-23
RU94016363A (ru) 1996-04-10
IL109655A (en) 1999-03-12
CZ283499B6 (cs) 1998-04-15

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