IL109655A - 2-aminopyrazine-5-carboxamide derivatives their preparation and pharmaceutical compositions containing them - Google Patents

2-aminopyrazine-5-carboxamide derivatives their preparation and pharmaceutical compositions containing them

Info

Publication number
IL109655A
IL109655A IL10965594A IL10965594A IL109655A IL 109655 A IL109655 A IL 109655A IL 10965594 A IL10965594 A IL 10965594A IL 10965594 A IL10965594 A IL 10965594A IL 109655 A IL109655 A IL 109655A
Authority
IL
Israel
Prior art keywords
group
general formula
compound
hydrogen atom
carries
Prior art date
Application number
IL10965594A
Other languages
English (en)
Other versions
IL109655A0 (en
Original Assignee
Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synthelabo filed Critical Synthelabo
Publication of IL109655A0 publication Critical patent/IL109655A0/xx
Publication of IL109655A publication Critical patent/IL109655A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/02Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/08Drugs for disorders of the urinary system of the prostate
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D241/00Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/02Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
    • C07D241/10Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
    • C07D241/14Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D241/24Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D241/26Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals with nitrogen atoms directly attached to ring carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Urology & Nephrology (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
IL10965594A 1993-05-17 1994-05-15 2-aminopyrazine-5-carboxamide derivatives their preparation and pharmaceutical compositions containing them IL109655A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9305930A FR2705344B1 (fr) 1993-05-17 1993-05-17 Dérivés de 2-aminopyrazine-5-carboxamide, leur préparation et leur application en thérapeutique.

Publications (2)

Publication Number Publication Date
IL109655A0 IL109655A0 (en) 1994-08-26
IL109655A true IL109655A (en) 1999-03-12

Family

ID=9447217

Family Applications (1)

Application Number Title Priority Date Filing Date
IL10965594A IL109655A (en) 1993-05-17 1994-05-15 2-aminopyrazine-5-carboxamide derivatives their preparation and pharmaceutical compositions containing them

Country Status (19)

Country Link
US (1) US5420130A (ru)
EP (1) EP0625514B1 (ru)
JP (1) JPH06329645A (ru)
CN (1) CN1104637A (ru)
AT (1) ATE183742T1 (ru)
AU (1) AU671361B2 (ru)
CA (1) CA2123668A1 (ru)
CZ (1) CZ283499B6 (ru)
DE (1) DE69420179D1 (ru)
FI (1) FI942265A (ru)
FR (1) FR2705344B1 (ru)
HU (1) HUT69711A (ru)
IL (1) IL109655A (ru)
NO (1) NO941830L (ru)
NZ (1) NZ260531A (ru)
PL (1) PL173309B1 (ru)
RU (1) RU2128176C1 (ru)
SK (1) SK57494A3 (ru)
ZA (1) ZA943353B (ru)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MXPA00010805A (es) * 1998-05-06 2002-05-08 Univ Duke Metodo para el tratamiento de sindromes de la vejiga y del tracto urinario inferior.
CZ301763B6 (cs) 1998-08-20 2010-06-16 Toyama Chemical Co., Ltd. Protivirový prostredek a derivát dusíkatého heterocyklického karboxamidu

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4041032A (en) * 1974-01-16 1977-08-09 Yamanouchi Pharmaceutical Co., Ltd. Pyrazine derivatives
FR2656609B1 (fr) * 1989-12-28 1992-03-27 Synthelabo Derives de 2-aminopyrimidine-4-carboxamide, leur preparation et leur application en therapeutique.

Also Published As

Publication number Publication date
RU94016363A (ru) 1996-04-10
JPH06329645A (ja) 1994-11-29
FR2705344B1 (fr) 1995-06-30
ZA943353B (en) 1995-03-28
FI942265A (fi) 1994-11-18
AU6312694A (en) 1994-11-24
EP0625514B1 (fr) 1999-08-25
SK57494A3 (en) 1995-07-11
DE69420179D1 (de) 1999-09-30
CZ119594A3 (en) 1994-12-15
FI942265A0 (fi) 1994-05-16
AU671361B2 (en) 1996-08-22
NO941830L (no) 1994-11-18
ATE183742T1 (de) 1999-09-15
IL109655A0 (en) 1994-08-26
RU2128176C1 (ru) 1999-03-27
CN1104637A (zh) 1995-07-05
FR2705344A1 (fr) 1994-11-25
CZ283499B6 (cs) 1998-04-15
HU9401512D0 (en) 1994-08-29
US5420130A (en) 1995-05-30
NO941830D0 (no) 1994-05-16
HUT69711A (en) 1995-09-28
CA2123668A1 (en) 1994-11-18
NZ260531A (en) 1995-10-26
EP0625514A1 (fr) 1994-11-23
PL173309B1 (pl) 1998-02-27

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Legal Events

Date Code Title Description
FF Patent granted
RH Patent void