SK4795A3 - Derivatives of macrolides antibiotics with 16-membered ring separated and used for treatment of illnesses and prarmaceutical agents on their base - Google Patents
Derivatives of macrolides antibiotics with 16-membered ring separated and used for treatment of illnesses and prarmaceutical agents on their baseInfo
- Publication number
- SK4795A3 SK4795A3 SK47-95A SK4795A SK4795A3 SK 4795 A3 SK4795 A3 SK 4795A3 SK 4795 A SK4795 A SK 4795A SK 4795 A3 SK4795 A3 SK 4795A3
- Authority
- SK
- Slovakia
- Prior art keywords
- derivatives
- pct
- membered ring
- prarmaceutical
- illnesses
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
- A61K31/7048—Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Molecular Biology (AREA)
- Genetics & Genomics (AREA)
- Engineering & Computer Science (AREA)
- Biotechnology (AREA)
- Biochemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
- Radiation-Therapy Devices (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US91424292A | 1992-07-15 | 1992-07-15 | |
| US99624392A | 1992-12-23 | 1992-12-23 | |
| PCT/US1993/005210 WO1994002496A1 (en) | 1992-07-15 | 1993-06-07 | Derivatives of 16-membered ring antibiotic macrolides |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| SK4795A3 true SK4795A3 (en) | 1995-07-11 |
Family
ID=27129638
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SK47-95A SK4795A3 (en) | 1992-07-15 | 1993-06-07 | Derivatives of macrolides antibiotics with 16-membered ring separated and used for treatment of illnesses and prarmaceutical agents on their base |
Country Status (22)
| Country | Link |
|---|---|
| US (1) | US5545624A (de) |
| EP (1) | EP0649430B1 (de) |
| JP (1) | JP2836964B2 (de) |
| KR (1) | KR950702570A (de) |
| CN (1) | CN1083068A (de) |
| AT (1) | ATE161265T1 (de) |
| AU (1) | AU4401093A (de) |
| BR (1) | BR9306741A (de) |
| CA (1) | CA2140243A1 (de) |
| CZ (1) | CZ9995A3 (de) |
| DE (1) | DE69315839T2 (de) |
| DK (1) | DK0649430T3 (de) |
| FI (1) | FI933204A (de) |
| GR (1) | GR3026064T3 (de) |
| HU (1) | HUT65330A (de) |
| IL (1) | IL106263A0 (de) |
| MX (1) | MX9304301A (de) |
| PL (1) | PL307137A1 (de) |
| SK (1) | SK4795A3 (de) |
| TW (1) | TW226373B (de) |
| UY (1) | UY23617A1 (de) |
| WO (1) | WO1994002496A1 (de) |
Families Citing this family (21)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5677287A (en) * | 1993-03-18 | 1997-10-14 | Pfizer Inc. | Antibacterial 16-membered ring macrolides containing olefins at C-20 |
| DE69402714T2 (de) * | 1993-07-15 | 1997-07-31 | Pfizer | Amid-derivate von 16-gliedrige heterocyclen als antibiotische macrolide |
| ES2076107B1 (es) * | 1993-09-20 | 1996-04-01 | Pfizer | Derivados de antibioticos macrolidos de anillos de 16 miembros. |
| AU3121095A (en) * | 1994-09-22 | 1996-04-09 | Pfizer Inc. | Antibiotic macrolides |
| EP0778283A3 (de) * | 1995-12-05 | 1998-01-28 | Pfizer Inc. | Antibiotische Makrolide |
| US6605599B1 (en) | 1997-07-08 | 2003-08-12 | Bristol-Myers Squibb Company | Epothilone derivatives |
| ES2213597T3 (es) * | 1999-08-30 | 2004-09-01 | Zaidan Hojin Biseibutsu Kagaku Kenkyu Kai | Antibioticos macrolidos y tratamiento de la pasteurelosis. |
| US20020111317A1 (en) * | 2000-09-25 | 2002-08-15 | Leonard Katz | Sixteen-membered macrolide compounds |
| US6664240B2 (en) * | 2001-11-15 | 2003-12-16 | Enanta Pharmaceuticals, Inc. | Tylosin derivatives having antibacterial activity |
| DK1483251T3 (da) | 2002-03-12 | 2010-04-12 | Bristol Myers Squibb Co | C3-cyano-epothilon-derivater |
| US7247617B2 (en) * | 2004-07-13 | 2007-07-24 | Kosan Biosciences Incorporated | Sixteen-member macrolide antiinfective agents |
| AU2007278195B2 (en) | 2006-07-28 | 2012-09-13 | Intervet International B.V. | Macrolide synthesis process |
| CN101506220B (zh) * | 2006-07-28 | 2012-10-17 | 英特威国际有限公司 | 大环内酯合成方法 |
| PT2782922T (pt) | 2011-11-25 | 2018-02-05 | The Kitasato Inst | Derivados antibacterianos de tilosina e processos para a sua preparação |
| FR2995605B1 (fr) * | 2012-09-18 | 2014-09-19 | Sanofi Sa | Derives de macrolides, leur preparation et leur application therapeutique. |
| AU2014270353B2 (en) * | 2013-05-23 | 2018-09-20 | Elanco Animal Health Gmbh | Tylosin derivatives and method for preparation thereof |
| CN108864228B (zh) * | 2014-01-22 | 2021-02-02 | 镇江威特药业有限责任公司 | 十六元环三胺内酯衍生物及其应用 |
| CN105777828A (zh) * | 2014-12-22 | 2016-07-20 | 菏泽市方明制药有限公司 | 一种用低质量的泰乐菌素制备高质量替米考星的方法 |
| US10287275B2 (en) | 2015-04-16 | 2019-05-14 | Victor Pharma Co., Ltd. Zhenjiang | 16-member triamilide derivatives and uses thereof |
| CN117510561B (zh) * | 2023-11-30 | 2024-04-02 | 中国农业科学院饲料研究所 | 一种泰乐菌素衍生物及其制备方法与应用 |
| CN117304241B (zh) * | 2023-11-30 | 2024-03-01 | 中国农业科学院饲料研究所 | 一种大环内酯类化合物及其制备方法与应用 |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3975372A (en) * | 1975-02-28 | 1976-08-17 | Schering Corporation | Preparation of 12,13-desepoxy-12,13-dehydrorosamicin |
| AU561147B2 (en) * | 1982-09-13 | 1987-04-30 | Eli Lilly And Company | 20-amino macrolide antibiotics |
| US4443436A (en) * | 1982-09-13 | 1984-04-17 | Eli Lilly And Company | C-20-Modified macrolide derivatives of the macrolide antibiotics tylosin, desmycosin, macrocin, and lactenocin |
| JPS59225199A (ja) * | 1983-02-10 | 1984-12-18 | Microbial Chem Res Found | ２０，２３−ジデオキシ−２３−アルキレンイミノ−２０−置換アミノマイカミノシルレロノライド |
| IL71032A0 (en) * | 1983-02-28 | 1984-05-31 | Lilly Co Eli | C-20 and c-23-modified macrolide derivatives |
| US4468511A (en) * | 1983-02-28 | 1984-08-28 | Eli Lilly And Company | C-20- And C-23-Modified macrolide derivatives |
| JPS59181299A (ja) * | 1983-03-31 | 1984-10-15 | Microbial Chem Res Found | ２０，２３−ジデオキシ−２０，２３−ビス置換アミノ−マイカミノシルレロノライド |
| US4921947A (en) * | 1986-03-31 | 1990-05-01 | Eli Lilly And Company | Process for preparing macrolide derivatives |
| US4820694A (en) * | 1986-09-29 | 1989-04-11 | Eli Lilly And Company | Modifications of 3-O-demethylmycinose in macrocin and lactenocin |
| EP0262903A3 (de) * | 1986-09-29 | 1988-11-02 | Eli Lilly And Company | Acylderivate von 20-modifiziertem Tylosin und Desmycosin-Derivate |
| US4920103A (en) * | 1986-09-29 | 1990-04-24 | Eli Lilly And Company | Modifications of mycinose and 3-O-demethylmycinose in tylosin-type macrolides |
| FR2638458A1 (fr) * | 1988-10-27 | 1990-05-04 | Adir | Nouveaux derives de la tylosine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
-
1993
- 1993-05-25 TW TW082104137A patent/TW226373B/zh active
- 1993-06-07 KR KR1019950700159A patent/KR950702570A/ko not_active Application Discontinuation
- 1993-06-07 JP JP6504438A patent/JP2836964B2/ja not_active Expired - Lifetime
- 1993-06-07 AU AU44010/93A patent/AU4401093A/en not_active Abandoned
- 1993-06-07 AT AT93914300T patent/ATE161265T1/de not_active IP Right Cessation
- 1993-06-07 DK DK93914300.4T patent/DK0649430T3/da active
- 1993-06-07 US US08/362,496 patent/US5545624A/en not_active Expired - Fee Related
- 1993-06-07 EP EP93914300A patent/EP0649430B1/de not_active Expired - Lifetime
- 1993-06-07 WO PCT/US1993/005210 patent/WO1994002496A1/en not_active Application Discontinuation
- 1993-06-07 DE DE69315839T patent/DE69315839T2/de not_active Expired - Fee Related
- 1993-06-07 SK SK47-95A patent/SK4795A3/sk unknown
- 1993-06-07 CA CA002140243A patent/CA2140243A1/en not_active Abandoned
- 1993-06-07 PL PL93307137A patent/PL307137A1/xx unknown
- 1993-06-07 BR BR9306741A patent/BR9306741A/pt not_active Application Discontinuation
- 1993-06-07 CZ CZ9599A patent/CZ9995A3/cs unknown
- 1993-07-07 IL IL106263A patent/IL106263A0/xx unknown
- 1993-07-14 CN CN93108458A patent/CN1083068A/zh active Pending
- 1993-07-14 HU HU9302016A patent/HUT65330A/hu unknown
- 1993-07-14 UY UY23617A patent/UY23617A1/es unknown
- 1993-07-14 FI FI933204A patent/FI933204A/fi unknown
- 1993-07-15 MX MX9304301A patent/MX9304301A/es unknown
-
1998
- 1998-02-04 GR GR980400232T patent/GR3026064T3/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| GR3026064T3 (en) | 1998-05-29 |
| AU4401093A (en) | 1994-02-14 |
| US5545624A (en) | 1996-08-13 |
| EP0649430A1 (de) | 1995-04-26 |
| WO1994002496A1 (en) | 1994-02-03 |
| MX9304301A (es) | 1994-02-28 |
| FI933204A (fi) | 1994-01-16 |
| CN1083068A (zh) | 1994-03-02 |
| KR950702570A (ko) | 1995-07-29 |
| JP2836964B2 (ja) | 1998-12-14 |
| HU9302016D0 (en) | 1993-10-28 |
| DK0649430T3 (da) | 1998-02-09 |
| IL106263A0 (en) | 1993-11-15 |
| HUT65330A (en) | 1994-05-02 |
| DE69315839D1 (de) | 1998-01-29 |
| TW226373B (de) | 1994-07-11 |
| CZ9995A3 (en) | 1995-07-12 |
| JPH07504922A (ja) | 1995-06-01 |
| DE69315839T2 (de) | 1998-04-09 |
| PL307137A1 (en) | 1995-05-02 |
| UY23617A1 (es) | 1994-01-05 |
| CA2140243A1 (en) | 1994-02-03 |
| ATE161265T1 (de) | 1998-01-15 |
| EP0649430B1 (de) | 1997-12-17 |
| BR9306741A (pt) | 1998-12-08 |
| FI933204A0 (fi) | 1993-07-14 |
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