SK285594B6 - Gama-karbolín, spôsob jeho prípravy a kompozícia s jeho obsahom - Google Patents
Gama-karbolín, spôsob jeho prípravy a kompozícia s jeho obsahom Download PDFInfo
- Publication number
- SK285594B6 SK285594B6 SK299-2000A SK2992000A SK285594B6 SK 285594 B6 SK285594 B6 SK 285594B6 SK 2992000 A SK2992000 A SK 2992000A SK 285594 B6 SK285594 B6 SK 285594B6
- Authority
- SK
- Slovakia
- Prior art keywords
- formula
- alkyl
- radical
- hydrogen
- gamma
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Diabetes (AREA)
- Child & Adolescent Psychology (AREA)
- Anesthesiology (AREA)
- Hospice & Palliative Care (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP97202761A EP0905136A1 (fr) | 1997-09-08 | 1997-09-08 | Tétrahydro gamma-carbolines |
| PCT/EP1998/005710 WO1999012926A1 (fr) | 1997-09-08 | 1998-09-01 | Tetrahydro gamma-carbolines |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| SK2992000A3 SK2992000A3 (en) | 2001-03-12 |
| SK285594B6 true SK285594B6 (sk) | 2007-04-05 |
Family
ID=8228715
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SK299-2000A SK285594B6 (sk) | 1997-09-08 | 1998-09-01 | Gama-karbolín, spôsob jeho prípravy a kompozícia s jeho obsahom |
Country Status (28)
| Country | Link |
|---|---|
| US (2) | US6303614B1 (fr) |
| EP (2) | EP0905136A1 (fr) |
| JP (1) | JP2001515899A (fr) |
| KR (1) | KR100603896B1 (fr) |
| CN (1) | CN1110496C (fr) |
| AT (1) | ATE243209T1 (fr) |
| AU (1) | AU752410B2 (fr) |
| BR (1) | BR9811769A (fr) |
| CA (1) | CA2301807A1 (fr) |
| CZ (1) | CZ297220B6 (fr) |
| DE (1) | DE69815700T2 (fr) |
| EE (1) | EE04496B1 (fr) |
| ES (1) | ES2202902T3 (fr) |
| HK (1) | HK1029107A1 (fr) |
| HR (1) | HRP20000108A2 (fr) |
| HU (1) | HUP0003577A3 (fr) |
| ID (1) | ID23954A (fr) |
| IL (1) | IL134894A (fr) |
| MY (1) | MY129176A (fr) |
| NO (1) | NO315236B1 (fr) |
| NZ (1) | NZ503096A (fr) |
| PL (1) | PL191863B1 (fr) |
| RU (1) | RU2208614C2 (fr) |
| SK (1) | SK285594B6 (fr) |
| TR (1) | TR200000616T2 (fr) |
| TW (1) | TW531539B (fr) |
| WO (1) | WO1999012926A1 (fr) |
| ZA (1) | ZA988161B (fr) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1944306A1 (fr) * | 2003-09-17 | 2008-07-16 | Janssen Pharmaceutica, N.V. | Composés hétérocycliques fusionnés |
| CN1882590B (zh) * | 2003-09-17 | 2014-03-05 | 詹森药业有限公司 | 作为血清素受体调节剂的稠合杂环化合物 |
| CN103788089A (zh) * | 2003-09-17 | 2014-05-14 | 詹森药业有限公司 | 作为血清素受体调节剂的稠合杂环化合物 |
| EP1757605A4 (fr) * | 2004-04-12 | 2007-12-19 | Taisho Pharmaceutical Co Ltd | Composé amine cyclique |
| EP1856126A2 (fr) | 2005-02-17 | 2007-11-21 | Wyeth a Corporation of the State of Delaware | Derive d'indole, benzothiophene, benzofurane et indene a fusion cycloalkyle |
| FR2885905A1 (fr) * | 2005-05-23 | 2006-11-24 | Trophos Sa | Nouveaux composes chimiques et leurs utilisations comme medicament |
| WO2007009485A1 (fr) * | 2005-07-22 | 2007-01-25 | Pharma C S.A. | Derives de 8-phenoxy-y-carboline substitues a activite 5ht1 |
| WO2007058580A1 (fr) * | 2005-11-15 | 2007-05-24 | Astrazeneca Ab | Nouveaux derives de 2-aminopyrimidinone et leur utilisation |
| US7637410B2 (en) * | 2006-10-06 | 2009-12-29 | Tyco Healthcare Group Lp | Surgical instrument including a locking assembly |
| MX2010003149A (es) * | 2007-09-20 | 2010-11-10 | D2E Llc | Derivados que contienen fluor de pirido[4,3-b]indoles hidrogenados con propiedades neuroprotectoras y de mejoramiento de cognicion, proceso de preparacion y uso. |
| WO2009082268A2 (fr) | 2007-12-21 | 2009-07-02 | Alla Chem, Llc | Ligands dalpha-adrénorécepteurs, de récepteurs de dopamine, de l'histamine, d'imidazoline et de sérotonine ainsi que leurs procédés d'utilisation |
| RU2374245C1 (ru) | 2008-08-22 | 2009-11-27 | Андрей Александрович Иващенко | Лиганд с широким спектром одновременной рецепторной активности, фармацевтическая композиция, способ ее получения и лекарственное средство |
| CN105399674B (zh) | 2015-12-31 | 2017-02-15 | 青岛清原化合物有限公司 | 吡唑类化合物或其盐、制备方法、除草剂组合物及用途 |
| CN106631941B (zh) * | 2016-12-30 | 2018-09-28 | 青岛瀚生生物科技股份有限公司 | 一种2-甲基-3氯苯基甲硫醚的制备方法 |
| GB201704325D0 (en) * | 2017-03-17 | 2017-05-03 | Argonaut Therapeutics Ltd | Compounds |
| CN110698474B (zh) * | 2019-11-14 | 2021-11-02 | 福州大学 | 一种α位取代四氢-γ-咔啉类化合物及其制备方法和应用 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3410286C2 (de) * | 1984-03-21 | 1986-01-23 | Fresenius AG, 6380 Bad Homburg | Verfahren zur Trennung von Blut sowie Vorrichtung zur Durchführung des Verfahrens |
| US4672117A (en) * | 1985-09-16 | 1987-06-09 | American Home Products Corporation | Antipsychotic gamma-carbolines |
| US4798896A (en) * | 1988-01-19 | 1989-01-17 | American Home Products Corporation | Antipsychotic gamma-carboline N-oxides |
| EP0705832B1 (fr) * | 1994-09-12 | 2003-08-13 | Eli Lilly And Company Limited | Modulateurs serotonergiques |
-
1997
- 1997-09-08 EP EP97202761A patent/EP0905136A1/fr not_active Withdrawn
-
1998
- 1998-09-01 CZ CZ20000726A patent/CZ297220B6/cs not_active IP Right Cessation
- 1998-09-01 TR TR2000/00616T patent/TR200000616T2/xx unknown
- 1998-09-01 CA CA002301807A patent/CA2301807A1/fr not_active Abandoned
- 1998-09-01 WO PCT/EP1998/005710 patent/WO1999012926A1/fr active IP Right Grant
- 1998-09-01 EE EEP200000059A patent/EE04496B1/xx not_active IP Right Cessation
- 1998-09-01 AU AU97421/98A patent/AU752410B2/en not_active Ceased
- 1998-09-01 RU RU2000109310/04A patent/RU2208614C2/ru not_active IP Right Cessation
- 1998-09-01 JP JP2000510733A patent/JP2001515899A/ja not_active Withdrawn
- 1998-09-01 ES ES98951365T patent/ES2202902T3/es not_active Expired - Lifetime
- 1998-09-01 CN CN98808818A patent/CN1110496C/zh not_active Expired - Fee Related
- 1998-09-01 KR KR1020007000970A patent/KR100603896B1/ko not_active IP Right Cessation
- 1998-09-01 PL PL339143A patent/PL191863B1/pl not_active IP Right Cessation
- 1998-09-01 BR BR9811769-6A patent/BR9811769A/pt not_active Application Discontinuation
- 1998-09-01 US US09/508,240 patent/US6303614B1/en not_active Expired - Fee Related
- 1998-09-01 DE DE69815700T patent/DE69815700T2/de not_active Expired - Fee Related
- 1998-09-01 EP EP98951365A patent/EP1015451B1/fr not_active Expired - Lifetime
- 1998-09-01 NZ NZ503096A patent/NZ503096A/en unknown
- 1998-09-01 AT AT98951365T patent/ATE243209T1/de not_active IP Right Cessation
- 1998-09-01 IL IL13489498A patent/IL134894A/xx not_active IP Right Cessation
- 1998-09-01 SK SK299-2000A patent/SK285594B6/sk unknown
- 1998-09-01 ID IDW20000432A patent/ID23954A/id unknown
- 1998-09-02 TW TW087114508A patent/TW531539B/zh not_active IP Right Cessation
- 1998-09-07 ZA ZA9808161A patent/ZA988161B/xx unknown
- 1998-09-07 MY MYPI98004080A patent/MY129176A/en unknown
- 1998-09-08 HU HU0003577A patent/HUP0003577A3/hu unknown
-
2000
- 2000-02-14 NO NO20000737A patent/NO315236B1/no unknown
- 2000-02-29 HR HR20000108A patent/HRP20000108A2/xx not_active Application Discontinuation
- 2000-11-10 HK HK00107165A patent/HK1029107A1/xx not_active IP Right Cessation
-
2001
- 2001-08-15 US US09/930,005 patent/US6506768B2/en not_active Expired - Fee Related
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