SK103193A3 - Piperidine derivatives, process for their preparation and pharmaceutical compositions containing these derivatives - Google Patents

Piperidine derivatives, process for their preparation and pharmaceutical compositions containing these derivatives Download PDF

Info

Publication number
SK103193A3
SK103193A3 SK1031-93A SK103193A SK103193A3 SK 103193 A3 SK103193 A3 SK 103193A3 SK 103193 A SK103193 A SK 103193A SK 103193 A3 SK103193 A3 SK 103193A3
Authority
SK
Slovakia
Prior art keywords
group
carbon atoms
alkyl
compounds
hydrogen
Prior art date
Application number
SK1031-93A
Other languages
English (en)
Slovak (sk)
Inventor
Samir Jegham
Itzchak Angel
Thomas Purcell
Johannes Schoemaker
Original Assignee
Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synthelabo filed Critical Synthelabo
Publication of SK103193A3 publication Critical patent/SK103193A3/sk

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
SK1031-93A 1992-09-28 1993-09-27 Piperidine derivatives, process for their preparation and pharmaceutical compositions containing these derivatives SK103193A3 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9211551A FR2696177B1 (fr) 1992-09-28 1992-09-28 Dérivés de pipéridine, leur préparation et leur application en thérapeutique.

Publications (1)

Publication Number Publication Date
SK103193A3 true SK103193A3 (en) 1994-08-10

Family

ID=9433967

Family Applications (1)

Application Number Title Priority Date Filing Date
SK1031-93A SK103193A3 (en) 1992-09-28 1993-09-27 Piperidine derivatives, process for their preparation and pharmaceutical compositions containing these derivatives

Country Status (24)

Country Link
US (1) US5434169A (de)
EP (1) EP0591027A1 (de)
JP (1) JPH06211838A (de)
KR (1) KR940007020A (de)
CN (1) CN1087339A (de)
AP (1) AP424A (de)
AU (1) AU658533B2 (de)
CA (1) CA2107061A1 (de)
CZ (1) CZ282080B6 (de)
DZ (1) DZ1718A1 (de)
FI (1) FI934221A (de)
FR (1) FR2696177B1 (de)
HU (2) HUT65303A (de)
IL (1) IL107133A (de)
MA (1) MA22981A1 (de)
MX (1) MX9305932A (de)
NO (1) NO933435L (de)
NZ (1) NZ248776A (de)
OA (1) OA09840A (de)
PL (1) PL172860B1 (de)
SK (1) SK103193A3 (de)
TN (1) TNSN93107A1 (de)
TW (1) TW272190B (de)
ZA (1) ZA937156B (de)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2231887A1 (en) * 1995-09-18 1997-03-27 Glaxo Group Limited 5-ht3 receptor antagonists for dyskinesia
AU714477B2 (en) * 1996-04-19 2000-01-06 Regents Of The University Of California, The Treatment of mood/affective disorders by glutamatergic upmodulators
FR2765221B1 (fr) * 1997-06-25 1999-07-30 Synthelabo Derives de 4-[(1h-imidazol-4-yl)piperidin-1-yl]anilide, leur preparation et leur application en therapeutique
US6013654A (en) * 1997-08-14 2000-01-11 Pharmacia & Upjohn Company Imidazo[1,2-A]pyridines for the treatment of CNS and cardiac diseases
GB9918425D0 (en) * 1999-08-04 1999-10-06 Novartis Ag Organic compounds
US6887870B1 (en) * 1999-10-12 2005-05-03 Bristol-Myers Squibb Company Heterocyclic sodium/proton exchange inhibitors and method
US7183305B2 (en) 2003-11-11 2007-02-27 Allergan, Inc. Process for the synthesis of imidazoles
US7880017B2 (en) 2003-11-11 2011-02-01 Allergan, Inc. Process for the synthesis of imidazoles
RU2422442C2 (ru) * 2005-07-29 2011-06-27 Ф. Хоффманн-Ля Рош Аг Производные индол-3-ил-карбонил-пиперидина и пиперазина
FR2925902B1 (fr) * 2008-01-02 2011-01-07 Sanofi Aventis DERIVES D'IMIDAZO°1,2-a!PYRIDINE-2-CARBOXAMIDES, LEUR PREPARATION ET LEUR APPLICATION EN THERAPEUTIQUE
WO2010080357A1 (en) * 2008-12-18 2010-07-15 Boehringer Ingelheim International Gmbh Serotonin 5-ht2b receptor inhibitors

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS61210080A (ja) * 1985-03-13 1986-09-18 Chisso Corp アルデヒドラクトンの製造法
FR2579596B1 (fr) * 1985-03-26 1987-11-20 Inst Nat Sante Rech Med (imidazolyl-4) piperidines, leur preparation et leur application en therapeutique
US5008390A (en) * 1985-05-23 1991-04-16 Smithkline Beckman Corporation Compounds for preparing 6-phenyl-2,3-dihydroimidazo[2,1-b]-thiazoles and corresponding thiazines
IT1230703B (it) * 1989-01-26 1991-10-29 Luso Farmaco Inst Derivati imidazolonici ad attivita' antiipertensiva, loro metodi di preparazione e composizioni farmaceutiche che li contengono.
US4925851A (en) * 1989-05-23 1990-05-15 Sandoz Pharmaceuticals Corp. 2- or 4-substituted-[2-(1H-imidazol-1-yl)ethyl]piperidines
FR2671083B1 (fr) * 1990-12-31 1994-12-23 Inst Nat Sante Rech Med Nouvelles 4-(4-imidazolyl) piperidines substituees en 1, leur preparation ainsi que leurs applications therapeutiques.

Also Published As

Publication number Publication date
PL300515A1 (en) 1994-04-05
CZ282080B6 (cs) 1997-05-14
TW272190B (de) 1996-03-11
NO933435D0 (no) 1993-09-27
ZA937156B (en) 1994-05-23
CN1087339A (zh) 1994-06-01
HU211249A9 (en) 1995-11-28
US5434169A (en) 1995-07-18
IL107133A (en) 1998-03-10
FI934221A0 (fi) 1993-09-27
FI934221A (fi) 1994-03-29
FR2696177A1 (fr) 1994-04-01
MX9305932A (es) 1994-04-29
AP9300575A0 (en) 1993-10-31
AP424A (en) 1995-11-04
PL172860B1 (pl) 1997-12-31
KR940007020A (ko) 1994-04-26
IL107133A0 (en) 1993-12-28
CZ9302015A3 (en) 1994-04-13
OA09840A (fr) 1994-08-15
EP0591027A1 (de) 1994-04-06
DZ1718A1 (fr) 2002-02-17
NO933435L (no) 1994-03-29
MA22981A1 (fr) 1994-04-01
AU4860693A (en) 1994-04-14
TNSN93107A1 (fr) 1994-03-17
AU658533B2 (en) 1995-04-13
HUT65303A (en) 1994-05-02
JPH06211838A (ja) 1994-08-02
HU9302727D0 (en) 1993-12-28
CA2107061A1 (en) 1994-03-29
FR2696177B1 (fr) 1995-05-12
NZ248776A (en) 1995-09-26

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