SI9500124A - Process for the preparation of Azithromycin Dihydrochloride - Google Patents

Process for the preparation of Azithromycin Dihydrochloride Download PDF

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Publication number
SI9500124A
SI9500124A SI9500124A SI9500124A SI9500124A SI 9500124 A SI9500124 A SI 9500124A SI 9500124 A SI9500124 A SI 9500124A SI 9500124 A SI9500124 A SI 9500124A SI 9500124 A SI9500124 A SI 9500124A
Authority
SI
Slovenia
Prior art keywords
azithromycin
dihydrochloride
preparation
hydrogen chloride
temperature
Prior art date
Application number
SI9500124A
Other languages
English (en)
Slovenian (sl)
Inventor
Nevenka Lopotar
Stjepan Mutak
Original Assignee
Pliva Pharm & Chem Works
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pliva Pharm & Chem Works filed Critical Pliva Pharm & Chem Works
Publication of SI9500124A publication Critical patent/SI9500124A/sl

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
SI9500124A 1994-04-15 1995-04-13 Process for the preparation of Azithromycin Dihydrochloride SI9500124A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
HR940251A HRP940251B1 (en) 1994-04-15 1994-04-15 Process for the preparation of azithromycin dihydrochloride

Publications (1)

Publication Number Publication Date
SI9500124A true SI9500124A (en) 1995-10-31

Family

ID=10946105

Family Applications (1)

Application Number Title Priority Date Filing Date
SI9500124A SI9500124A (en) 1994-04-15 1995-04-13 Process for the preparation of Azithromycin Dihydrochloride

Country Status (16)

Country Link
EP (1) EP0677530B1 (de)
JP (1) JP3075681B2 (de)
CN (1) CN1042033C (de)
AT (1) ATE154028T1 (de)
BG (1) BG61769B1 (de)
CA (1) CA2146475C (de)
DE (1) DE69500327T2 (de)
ES (1) ES2104441T3 (de)
HR (1) HRP940251B1 (de)
HU (1) HU217553B (de)
PL (1) PL177292B1 (de)
RO (1) RO113737B1 (de)
RU (1) RU2134271C1 (de)
SI (1) SI9500124A (de)
SK (1) SK281178B6 (de)
UA (1) UA41902C2 (de)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HRP20020231A2 (en) 2002-03-18 2003-12-31 Pliva D D ISOSTRUCTURAL PSEUDOPOLYMORPHS OF 9-DEOXO-9a-AZA-9a-METHYL-9a-HOMOERYTHROMYCIN A
US6861411B1 (en) 1997-12-02 2005-03-01 Pfizer, Inc. Method of treating eye infections with azithromycin
US7056893B2 (en) 1999-03-31 2006-06-06 Insite Vision, Inc. Topical treatment for prevention of ocular infections
US6239113B1 (en) 1999-03-31 2001-05-29 Insite Vision, Incorporated Topical treatment or prevention of ocular infections
US7572773B2 (en) 2003-07-24 2009-08-11 Pliva Hrvatska D.O.O. Single dose fast dissolving azithromycin
CN100343267C (zh) * 2005-08-05 2007-10-17 新昌国邦化学工业有限公司 阿奇霉素酒石酸盐的制备方法
CN100427499C (zh) * 2005-12-20 2008-10-22 山东诚创医药技术开发有限公司 一种阿奇霉素的可溶性盐及其制备方法
CN101092440B (zh) * 2007-07-19 2010-05-26 浙江尖峰药业有限公司 硫酸阿奇霉素的制备方法
CN102746350A (zh) * 2011-04-21 2012-10-24 常州泰康制药有限公司 盐酸阿奇霉素的制备方法
CN104045674B (zh) * 2014-05-21 2017-01-04 丽珠医药集团股份有限公司 一种阿奇霉素的制备方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1100504A (en) * 1967-08-16 1968-01-24 Pliva Pharm & Chem Works Erythromycin oxime and 9-amino-3-o-cladinosyl-5-o-desosaminyl-6,11,12-trihydroxy-2,4,6,8,10,12-hexamethylpentadecane-13-olide
US4474768A (en) * 1982-07-19 1984-10-02 Pfizer Inc. N-Methyl 11-aza-10-deoxo-10-dihydro-erytromycin A, intermediates therefor
YU43658B (en) * 1983-07-18 1989-10-31 Pliva Pharm & Chem Works Process for preparing 7,16-dioxa-2-aza-10-0-cladinosyl-12,0-desosaminyl-4,5-dihydroxy-6-ethyl-3,5,9,11,13,15-hexamethyl-bicyclo(11.2.1)hexadeca-1(2)-ene-8

Also Published As

Publication number Publication date
ATE154028T1 (de) 1997-06-15
BG99580A (bg) 1995-12-29
BG61769B1 (bg) 1998-05-29
EP0677530B1 (de) 1997-06-04
ES2104441T3 (es) 1997-10-01
JP3075681B2 (ja) 2000-08-14
HU9501084D0 (en) 1995-06-28
HU217553B (hu) 2000-02-28
HRP940251A2 (en) 1997-06-30
SK281178B6 (sk) 2000-12-11
DE69500327T2 (de) 1998-01-08
CN1042033C (zh) 1999-02-10
UA41902C2 (uk) 2001-10-15
PL177292B1 (pl) 1999-10-29
HRP940251B1 (en) 1998-12-31
EP0677530A1 (de) 1995-10-18
SK49195A3 (en) 1995-11-08
RU2134271C1 (ru) 1999-08-10
HUT71840A (en) 1996-02-28
RO113737B1 (ro) 1998-10-30
JPH0841058A (ja) 1996-02-13
RU95105596A (ru) 1997-01-10
DE69500327D1 (de) 1997-07-10
CA2146475C (en) 1999-06-29
CN1112566A (zh) 1995-11-29
PL308095A1 (en) 1995-10-16
CA2146475A1 (en) 1995-10-16

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