SI3830092T1 - Heteroaromatski NMDA receptorski modulatorji in njihove uporabe - Google Patents
Heteroaromatski NMDA receptorski modulatorji in njihove uporabeInfo
- Publication number
- SI3830092T1 SI3830092T1 SI201930580T SI201930580T SI3830092T1 SI 3830092 T1 SI3830092 T1 SI 3830092T1 SI 201930580 T SI201930580 T SI 201930580T SI 201930580 T SI201930580 T SI 201930580T SI 3830092 T1 SI3830092 T1 SI 3830092T1
- Authority
- SI
- Slovenia
- Prior art keywords
- heteroaromatic
- nmda receptor
- receptor modulators
- nmda
- modulators
- Prior art date
Links
- 102000004868 N-Methyl-D-Aspartate Receptors Human genes 0.000 title 1
- 108090001041 N-Methyl-D-Aspartate Receptors Proteins 0.000 title 1
- 125000001072 heteroaryl group Chemical group 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Psychiatry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Epidemiology (AREA)
- Hospice & Palliative Care (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Steroid Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pyridine Compounds (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201862714100P | 2018-08-03 | 2018-08-03 | |
EP19876025.8A EP3830092B1 (en) | 2018-08-03 | 2019-08-02 | Heteroaromatic nmda receptor modulators and uses thereof |
PCT/US2019/044814 WO2020086136A2 (en) | 2018-08-03 | 2019-08-02 | Heteroaromatic nmda receptor modulators and uses thereof |
Publications (1)
Publication Number | Publication Date |
---|---|
SI3830092T1 true SI3830092T1 (sl) | 2023-09-29 |
Family
ID=69228330
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SI201930580T SI3830092T1 (sl) | 2018-08-03 | 2019-08-02 | Heteroaromatski NMDA receptorski modulatorji in njihove uporabe |
Country Status (37)
Country | Link |
---|---|
US (4) | US10584131B2 (sl) |
EP (2) | EP4223760A1 (sl) |
JP (1) | JP7319369B2 (sl) |
KR (1) | KR20210039432A (sl) |
CN (1) | CN112513047B (sl) |
AR (1) | AR115905A1 (sl) |
AU (1) | AU2019368147B2 (sl) |
BR (1) | BR112021001967A2 (sl) |
CA (1) | CA3108519A1 (sl) |
CL (1) | CL2021000294A1 (sl) |
CO (1) | CO2021002898A2 (sl) |
CR (1) | CR20210125A (sl) |
CU (1) | CU24647B1 (sl) |
CY (1) | CY1126144T1 (sl) |
DK (1) | DK3830092T3 (sl) |
DO (1) | DOP2021000025A (sl) |
EA (1) | EA202190431A1 (sl) |
EC (1) | ECSP21014902A (sl) |
ES (1) | ES2951872T3 (sl) |
FI (1) | FI3830092T3 (sl) |
HR (1) | HRP20230774T1 (sl) |
HU (1) | HUE062566T2 (sl) |
IL (1) | IL280474B2 (sl) |
JO (1) | JOP20210020A1 (sl) |
LT (1) | LT3830092T (sl) |
MA (1) | MA53351B1 (sl) |
MX (1) | MX2021001367A (sl) |
PE (1) | PE20210948A1 (sl) |
PH (1) | PH12021550242A1 (sl) |
PL (1) | PL3830092T3 (sl) |
PT (1) | PT3830092T (sl) |
RS (1) | RS64359B1 (sl) |
SG (1) | SG11202101125VA (sl) |
SI (1) | SI3830092T1 (sl) |
TW (1) | TWI833783B (sl) |
WO (1) | WO2020086136A2 (sl) |
ZA (1) | ZA202101273B (sl) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP4006038A1 (en) | 2015-12-09 | 2022-06-01 | Cadent Therapeutics, Inc. | Thienopyrimidinone nmda receptor modulators and uses thereof |
JP7071917B2 (ja) * | 2015-12-09 | 2022-05-19 | カデント セラピューティクス,インコーポレーテッド | ヘテロ芳香族nmda受容体モジュレーターおよびその使用 |
JP7332472B2 (ja) | 2016-12-22 | 2023-08-23 | ノバルティス アーゲー | Nmda受容体モジュレーターおよびその使用 |
CN112513047B (zh) | 2018-08-03 | 2023-10-20 | 诺华股份有限公司 | 芳香杂环nmda受体调节剂及其用途 |
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WO2017188694A1 (ko) | 2016-04-25 | 2017-11-02 | 이뮤노메트테라퓨틱스 인코포레이티드 | 질소를 포함하는 헤테로아릴 화합물 및 이의 용도 |
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2019
- 2019-08-02 CN CN201980051645.9A patent/CN112513047B/zh active Active
- 2019-08-02 EA EA202190431A patent/EA202190431A1/ru unknown
- 2019-08-02 AU AU2019368147A patent/AU2019368147B2/en active Active
- 2019-08-02 WO PCT/US2019/044814 patent/WO2020086136A2/en active Application Filing
- 2019-08-02 PT PT198760258T patent/PT3830092T/pt unknown
- 2019-08-02 DK DK19876025.8T patent/DK3830092T3/da active
- 2019-08-02 TW TW108127473A patent/TWI833783B/zh active
- 2019-08-02 SG SG11202101125VA patent/SG11202101125VA/en unknown
- 2019-08-02 CA CA3108519A patent/CA3108519A1/en active Pending
- 2019-08-02 RS RS20230563A patent/RS64359B1/sr unknown
- 2019-08-02 HU HUE19876025A patent/HUE062566T2/hu unknown
- 2019-08-02 IL IL280474A patent/IL280474B2/en unknown
- 2019-08-02 JP JP2021529249A patent/JP7319369B2/ja active Active
- 2019-08-02 ES ES19876025T patent/ES2951872T3/es active Active
- 2019-08-02 MX MX2021001367A patent/MX2021001367A/es unknown
- 2019-08-02 AR ARP190102209A patent/AR115905A1/es unknown
- 2019-08-02 HR HRP20230774TT patent/HRP20230774T1/hr unknown
- 2019-08-02 MA MA53351A patent/MA53351B1/fr unknown
- 2019-08-02 LT LTEPPCT/US2019/044814T patent/LT3830092T/lt unknown
- 2019-08-02 CU CU2021000013A patent/CU24647B1/es unknown
- 2019-08-02 PE PE2021000151A patent/PE20210948A1/es unknown
- 2019-08-02 EP EP23165151.4A patent/EP4223760A1/en active Pending
- 2019-08-02 SI SI201930580T patent/SI3830092T1/sl unknown
- 2019-08-02 US US16/530,274 patent/US10584131B2/en active Active
- 2019-08-02 FI FIEP19876025.8T patent/FI3830092T3/fi active
- 2019-08-02 JO JOP/2021/0020A patent/JOP20210020A1/ar unknown
- 2019-08-02 CR CR20210125A patent/CR20210125A/es unknown
- 2019-08-02 BR BR112021001967-7A patent/BR112021001967A2/pt unknown
- 2019-08-02 KR KR1020217006300A patent/KR20210039432A/ko active Search and Examination
- 2019-08-02 PL PL19876025.8T patent/PL3830092T3/pl unknown
- 2019-08-02 EP EP19876025.8A patent/EP3830092B1/en active Active
- 2019-11-08 US US16/678,806 patent/US10752633B2/en active Active
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2021
- 2021-02-01 PH PH12021550242A patent/PH12021550242A1/en unknown
- 2021-02-02 DO DO2021000025A patent/DOP2021000025A/es unknown
- 2021-02-03 CL CL2021000294A patent/CL2021000294A1/es unknown
- 2021-02-12 US US17/174,826 patent/US11542264B2/en active Active
- 2021-02-25 ZA ZA2021/01273A patent/ZA202101273B/en unknown
- 2021-03-03 EC ECSENADI202114902A patent/ECSP21014902A/es unknown
- 2021-03-03 CO CONC2021/0002898A patent/CO2021002898A2/es unknown
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2023
- 2023-07-13 US US18/221,694 patent/US20240199617A1/en active Pending
- 2023-08-02 CY CY20231100387T patent/CY1126144T1/el unknown
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