SI3068405T1 - Pirolo (1,2,f)(1,2,4)triazini uporabni za zdavljenje okužb z respiratornim sincicijskim virusom - Google Patents

Pirolo (1,2,f)(1,2,4)triazini uporabni za zdavljenje okužb z respiratornim sincicijskim virusom

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Publication number
SI3068405T1
SI3068405T1 SI201431284T SI201431284T SI3068405T1 SI 3068405 T1 SI3068405 T1 SI 3068405T1 SI 201431284 T SI201431284 T SI 201431284T SI 201431284 T SI201431284 T SI 201431284T SI 3068405 T1 SI3068405 T1 SI 3068405T1
Authority
SI
Slovenia
Prior art keywords
pyrrolo
virus infections
treating respiratory
respiratory syncitial
syncitial virus
Prior art date
Application number
SI201431284T
Other languages
English (en)
Slovenian (sl)
Inventor
Michael O'neil Hanrahan Clarke
Edward Doerffler
Richard L. Mackman
Dustin Siegel
Original Assignee
Gilead Sciences, Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=52003049&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SI3068405(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Gilead Sciences, Inc. filed Critical Gilead Sciences, Inc.
Publication of SI3068405T1 publication Critical patent/SI3068405T1/sl

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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7052Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
    • A61K31/706Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/407Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/53Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with three nitrogens as the only ring hetero atoms, e.g. chlorazanil, melamine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/16Antivirals for RNA viruses for influenza or rhinoviruses
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/04Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6561Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H7/00Compounds containing non-saccharide radicals linked to saccharide radicals by a carbon-to-carbon bond
    • C07H7/06Heterocyclic radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Virology (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Biochemistry (AREA)
  • Epidemiology (AREA)
  • Biotechnology (AREA)
  • Engineering & Computer Science (AREA)
  • Genetics & Genomics (AREA)
  • Oncology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Communicable Diseases (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Saccharide Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
SI201431284T 2013-11-11 2014-11-06 Pirolo (1,2,f)(1,2,4)triazini uporabni za zdavljenje okužb z respiratornim sincicijskim virusom SI3068405T1 (sl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201361902544P 2013-11-11 2013-11-11
PCT/US2014/064412 WO2015069939A1 (en) 2013-11-11 2014-11-06 Pyrrolo [1,2,f] [1,2,4] triazines useful for treating respiratory syncitial virus infections
EP14806123.7A EP3068405B1 (en) 2013-11-11 2014-11-06 Pyrrolo [1,2,f][1,2,4]triazines useful for treating respiratory syncitial virus infections

Publications (1)

Publication Number Publication Date
SI3068405T1 true SI3068405T1 (sl) 2019-08-30

Family

ID=52003049

Family Applications (2)

Application Number Title Priority Date Filing Date
SI201431284T SI3068405T1 (sl) 2013-11-11 2014-11-06 Pirolo (1,2,f)(1,2,4)triazini uporabni za zdavljenje okužb z respiratornim sincicijskim virusom
SI201431978T SI3505173T1 (sl) 2013-11-11 2014-11-06 Pirolo(1,2-F)(1,2,4)triazini, uporabni za zdravljenje okužb z respiratornim sincicijskim virusom

Family Applications After (1)

Application Number Title Priority Date Filing Date
SI201431978T SI3505173T1 (sl) 2013-11-11 2014-11-06 Pirolo(1,2-F)(1,2,4)triazini, uporabni za zdravljenje okužb z respiratornim sincicijskim virusom

Country Status (36)

Country Link
US (5) US9388208B2 (OSRAM)
EP (3) EP3505173B1 (OSRAM)
JP (7) JP6234571B2 (OSRAM)
KR (4) KR102355881B1 (OSRAM)
CN (3) CN110003215B (OSRAM)
AP (1) AP2016009186A0 (OSRAM)
AU (5) AU2014346665A1 (OSRAM)
BR (1) BR112016010261B1 (OSRAM)
CA (1) CA2928674C (OSRAM)
CL (1) CL2016001120A1 (OSRAM)
CR (1) CR20160220A (OSRAM)
CU (1) CU20160065A7 (OSRAM)
CY (1) CY1121948T1 (OSRAM)
DK (2) DK3505173T3 (OSRAM)
DO (1) DOP2016000107A (OSRAM)
EA (2) EA039734B1 (OSRAM)
ES (2) ES2926155T3 (OSRAM)
GT (1) GT201600086A (OSRAM)
HR (2) HRP20191303T1 (OSRAM)
HU (2) HUE059683T2 (OSRAM)
IL (1) IL245324B (OSRAM)
LT (2) LT3505173T (OSRAM)
MD (1) MD4596C1 (OSRAM)
MX (2) MX376186B (OSRAM)
MY (2) MY197933A (OSRAM)
NZ (1) NZ719592A (OSRAM)
PE (1) PE20160670A1 (OSRAM)
PH (1) PH12016500867A1 (OSRAM)
PL (2) PL3068405T3 (OSRAM)
PT (2) PT3505173T (OSRAM)
SG (1) SG11201603427XA (OSRAM)
SI (2) SI3068405T1 (OSRAM)
TR (1) TR201910961T4 (OSRAM)
UA (1) UA119050C2 (OSRAM)
WO (1) WO2015069939A1 (OSRAM)
ZA (1) ZA201603123B (OSRAM)

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