SI2366703T1 - Polimorfna oblika 2-amino (nitroaril) tiazolnega derivata - Google Patents

Polimorfna oblika 2-amino (nitroaril) tiazolnega derivata

Info

Publication number
SI2366703T1
SI2366703T1 SI200831294T SI200831294T SI2366703T1 SI 2366703 T1 SI2366703 T1 SI 2366703T1 SI 200831294 T SI200831294 T SI 200831294T SI 200831294 T SI200831294 T SI 200831294T SI 2366703 T1 SI2366703 T1 SI 2366703T1
Authority
SI
Slovenia
Prior art keywords
nitroaryl
amino
polymorph form
thiazole derivative
thiazole
Prior art date
Application number
SI200831294T
Other languages
English (en)
Inventor
Alain Moussy
Philippe Reginault
Francois Bellamy
Anne Lermet
Original Assignee
Ab Science
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ab Science filed Critical Ab Science
Publication of SI2366703T1 publication Critical patent/SI2366703T1/sl

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/10Drugs for disorders of the urinary system of the bladder
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/02Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/08Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A61P19/10Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/04Antineoplastic agents specific for metastasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Diabetes (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Oncology (AREA)
  • Hematology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Obesity (AREA)
  • Pulmonology (AREA)
  • Urology & Nephrology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Communicable Diseases (AREA)
  • Transplantation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Catalysts (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
SI200831294T 2007-02-13 2008-02-13 Polimorfna oblika 2-amino (nitroaril) tiazolnega derivata SI2366703T1 (sl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US88958707P 2007-02-13 2007-02-13
EP11170200.7A EP2366703B1 (en) 2007-02-13 2008-02-13 Polymorph form of 2-amino (nitroaryl) thiazole derivative

Publications (1)

Publication Number Publication Date
SI2366703T1 true SI2366703T1 (sl) 2014-10-30

Family

ID=39332208

Family Applications (2)

Application Number Title Priority Date Filing Date
SI200831294T SI2366703T1 (sl) 2007-02-13 2008-02-13 Polimorfna oblika 2-amino (nitroaril) tiazolnega derivata
SI200830399T SI2118099T1 (sl) 2007-02-13 2008-02-13 Postopek za sintezo 2-aminotiazolnih spojin kot kinaznih inhibitorjev

Family Applications After (1)

Application Number Title Priority Date Filing Date
SI200830399T SI2118099T1 (sl) 2007-02-13 2008-02-13 Postopek za sintezo 2-aminotiazolnih spojin kot kinaznih inhibitorjev

Country Status (23)

Country Link
US (3) US8153792B2 (sl)
EP (2) EP2366703B1 (sl)
JP (2) JP5568312B2 (sl)
KR (1) KR20090110851A (sl)
CN (2) CN101657446B (sl)
AR (1) AR065337A1 (sl)
AT (1) ATE515506T1 (sl)
AU (1) AU2008214679A1 (sl)
BR (1) BRPI0807626B1 (sl)
CA (2) CA2677586C (sl)
ES (2) ES2522169T3 (sl)
HR (2) HRP20110709T1 (sl)
IL (1) IL200320A0 (sl)
MA (1) MA31180B1 (sl)
MX (1) MX2009008665A (sl)
NZ (1) NZ578944A (sl)
PL (2) PL2118099T3 (sl)
RU (2) RU2456285C2 (sl)
SI (2) SI2366703T1 (sl)
TN (1) TN2009000342A1 (sl)
TW (1) TWI406862B (sl)
WO (1) WO2008098949A2 (sl)
ZA (1) ZA200905981B (sl)

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WO2011131705A1 (en) 2010-04-20 2011-10-27 Ab Science Treatment of multiple sclerosis with masitinib
AR081772A1 (es) 2010-06-02 2012-10-17 Ab Science Tratamiento de la artritis reumatoide con masitinib
US10045978B2 (en) 2010-11-05 2018-08-14 Ab Science Treatment of mastocytosis with masitinib
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TW201605449A (zh) 2013-12-02 2016-02-16 Ab化學公司 馬賽替尼治療結腸直腸癌的用途
EP2886543A1 (en) 2013-12-18 2015-06-24 Sandoz Ag Crystalline form of mastinib mesylate
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EP3359195B1 (en) 2015-10-05 2024-05-29 AB Science Treatment of severe systemic mastocytosis with masitinib
HUE057398T2 (hu) 2016-03-25 2022-05-28 Ab Science A masitinib alkalmazása egy amiotrófiás laterálszklerózisos beteg alpopuláció kezelésére
CN110678464A (zh) * 2017-03-31 2020-01-10 桑多斯股份公司 马赛替尼的晶型
US10696638B2 (en) 2017-12-26 2020-06-30 Industrial Technology Research Institute Compounds for inhibiting AGC kinase and pharmaceutical compositions comprising the same
US20230000838A1 (en) 2019-11-22 2023-01-05 Ab Science Masitinib for the treatment of sickle cell disease
EP3831384A1 (en) 2019-12-02 2021-06-09 AB Science Use of masitinib for the treatment of eosinophilic asthma
IL294817A (en) 2020-02-20 2022-09-01 Ab Science Masitinib for the treatment of a subpopulation of multiple sclerosis patients
KR20230014681A (ko) 2020-04-10 2023-01-30 에이비 사이언스 코로나바이러스 질환 2019(covid-19)의 치료를 위한 마시티닙의 용도
WO2022129410A1 (en) 2020-12-16 2022-06-23 Ab Science Masitinib for the treatment of alzheimer's disease
US20230321081A1 (en) 2021-05-17 2023-10-12 Ab Science Masitinib for the treatment of castrate-resistant prostate cancer
CN115850258A (zh) * 2022-12-27 2023-03-28 东北林业大学 一种马赛替尼的合成方法

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Also Published As

Publication number Publication date
EP2118099B1 (en) 2011-07-06
CN101657446B (zh) 2013-05-15
CN101657446A (zh) 2010-02-24
US8153792B2 (en) 2012-04-10
TN2009000342A1 (en) 2010-12-31
PL2118099T3 (pl) 2011-12-30
ZA200905981B (en) 2010-11-24
CN103342701A (zh) 2013-10-09
RU2491286C1 (ru) 2013-08-27
CA2677586A1 (en) 2008-08-21
PL2366703T3 (pl) 2015-02-27
CA2970628C (en) 2019-08-27
MX2009008665A (es) 2009-08-21
IL200320A0 (en) 2010-04-29
US8492545B2 (en) 2013-07-23
HRP20110709T1 (hr) 2011-11-30
US20130289045A1 (en) 2013-10-31
US8940894B2 (en) 2015-01-27
JP5784073B2 (ja) 2015-09-24
TW200848419A (en) 2008-12-16
RU2009132186A (ru) 2011-03-20
NZ578944A (en) 2011-03-31
HRP20140986T1 (hr) 2014-11-21
ES2369617T3 (es) 2011-12-02
TWI406862B (zh) 2013-09-01
KR20090110851A (ko) 2009-10-22
CN103342701B (zh) 2016-09-21
MA31180B1 (fr) 2010-02-01
US20100121063A1 (en) 2010-05-13
SI2118099T1 (sl) 2011-11-30
ATE515506T1 (de) 2011-07-15
EP2118099A2 (en) 2009-11-18
EP2366703B1 (en) 2014-07-30
US20120196871A1 (en) 2012-08-02
CA2677586C (en) 2017-07-25
AR065337A1 (es) 2009-06-03
JP5568312B2 (ja) 2014-08-06
JP2010518141A (ja) 2010-05-27
WO2008098949A2 (en) 2008-08-21
BRPI0807626A2 (pt) 2014-11-25
ES2522169T3 (es) 2014-11-13
RU2456285C2 (ru) 2012-07-20
WO2008098949A3 (en) 2008-10-02
EP2366703A1 (en) 2011-09-21
BRPI0807626B1 (pt) 2022-03-03
JP2013177437A (ja) 2013-09-09
CA2970628A1 (en) 2008-08-21
AU2008214679A1 (en) 2008-08-21

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