AR081772A1 - Tratamiento de la artritis reumatoide con masitinib - Google Patents
Tratamiento de la artritis reumatoide con masitinibInfo
- Publication number
- AR081772A1 AR081772A1 ARP110101884A ARP110101884A AR081772A1 AR 081772 A1 AR081772 A1 AR 081772A1 AR P110101884 A ARP110101884 A AR P110101884A AR P110101884 A ARP110101884 A AR P110101884A AR 081772 A1 AR081772 A1 AR 081772A1
- Authority
- AR
- Argentina
- Prior art keywords
- treatment
- masitinib
- reumatoid arthritis
- arthritis
- reumatoid
- Prior art date
Links
- 239000002139 L01XE22 - Masitinib Substances 0.000 title abstract 2
- WJEOLQLKVOPQFV-UHFFFAOYSA-N masitinib Chemical compound C1CN(C)CCN1CC1=CC=C(C(=O)NC=2C=C(NC=3SC=C(N=3)C=3C=NC=CC=3)C(C)=CC=2)C=C1 WJEOLQLKVOPQFV-UHFFFAOYSA-N 0.000 title abstract 2
- 229960004655 masitinib Drugs 0.000 title abstract 2
- 206010003246 arthritis Diseases 0.000 title 1
- 210000003630 histaminocyte Anatomy 0.000 abstract 1
- 239000003112 inhibitor Substances 0.000 abstract 1
- 206010039073 rheumatoid arthritis Diseases 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 239000005483 tyrosine kinase inhibitor Substances 0.000 abstract 1
- 229940121358 tyrosine kinase inhibitor Drugs 0.000 abstract 1
- 150000004917 tyrosine kinase inhibitor derivatives Chemical class 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Epidemiology (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Immunology (AREA)
- Organic Chemistry (AREA)
- Rheumatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Physical Education & Sports Medicine (AREA)
Abstract
Un inhibidor de la tirosina quinasa o un inhibidor de los mastocitos, y en particular masitinib o una sal farmacéuticamente aceptable del mismo, para el tratamiento de la artritis reumatoide humana.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US35060310P | 2010-06-02 | 2010-06-02 |
Publications (1)
Publication Number | Publication Date |
---|---|
AR081772A1 true AR081772A1 (es) | 2012-10-17 |
Family
ID=44119407
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP110101884A AR081772A1 (es) | 2010-06-02 | 2011-06-01 | Tratamiento de la artritis reumatoide con masitinib |
Country Status (4)
Country | Link |
---|---|
US (1) | US20130267484A1 (es) |
AR (1) | AR081772A1 (es) |
TW (1) | TW201204719A (es) |
WO (1) | WO2011151372A1 (es) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6962940B2 (en) | 2002-03-20 | 2005-11-08 | Celgene Corporation | (+)-2-[1-(3-Ethoxy-4-methoxyphenyl)-2-methylsulfonylethyl]-4-acetylaminoisoindoline-1,3-dione: methods of using and compositions thereof |
WO2018045258A1 (en) * | 2016-09-02 | 2018-03-08 | The University Of Chicago | TREATMENT OF TNF-alpha CYTOTOXICITY |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
NZ530764A (en) * | 2001-07-09 | 2008-07-31 | Combinatorx Inc | Composition comprising a tricyclic antidepressant and a corticosteroid administered simutaneously or within 14 days for treatment of inflammatory disorders |
DK1525200T3 (da) | 2002-08-02 | 2007-12-03 | Ab Science | 2-(3-aminoaryl)amino-4-aryl-thiazoler til sygdomsbehandling |
US8450302B2 (en) * | 2002-08-02 | 2013-05-28 | Ab Science | 2-(3-aminoaryl) amino-4-aryl-thiazoles and their use as c-kit inhibitors |
US8073630B2 (en) * | 2006-08-30 | 2011-12-06 | Exagen Diagnostics, Inc. | Pharacogenetic method for prediction of the efficacy of methotrexate monotherapy in recent-onset arthritis |
NZ578944A (en) | 2007-02-13 | 2011-03-31 | Ab Science | PROCESS FOR THE SYNTHESIS OF 2-AMINOTHIAZOLE COMPOUNDS SUCH AS 4-(4-Methyl-piperazin-1-ylmethyl)-N-[4-methyl-3-(4-pyridin-3-yl-thiazol-2-ylamino)-phenyl]-benzamide AS KINASE INHIBITORS |
-
2011
- 2011-06-01 WO PCT/EP2011/059034 patent/WO2011151372A1/en active Application Filing
- 2011-06-01 US US13/700,788 patent/US20130267484A1/en not_active Abandoned
- 2011-06-01 AR ARP110101884A patent/AR081772A1/es unknown
- 2011-06-01 TW TW100119306A patent/TW201204719A/zh unknown
Also Published As
Publication number | Publication date |
---|---|
WO2011151372A1 (en) | 2011-12-08 |
US20130267484A1 (en) | 2013-10-10 |
TW201204719A (en) | 2012-02-01 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FB | Suspension of granting procedure |