UY34132A - Terapias combinadas para el tratamiento de neoplasias malignas hematológicas utilizando inhibidores de piridopirimidinona de pi3k/mtor con bendamustina y/o rituximab. - Google Patents
Terapias combinadas para el tratamiento de neoplasias malignas hematológicas utilizando inhibidores de piridopirimidinona de pi3k/mtor con bendamustina y/o rituximab.Info
- Publication number
- UY34132A UY34132A UY0001034132A UY34132A UY34132A UY 34132 A UY34132 A UY 34132A UY 0001034132 A UY0001034132 A UY 0001034132A UY 34132 A UY34132 A UY 34132A UY 34132 A UY34132 A UY 34132A
- Authority
- UY
- Uruguay
- Prior art keywords
- pyridopirimidinone
- malignal
- neoplasias
- bendamustine
- pi3k
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4184—1,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K39/00—Medicinal preparations containing antigens or antibodies
- A61K39/395—Antibodies; Immunoglobulins; Immune serum, e.g. antilymphocytic serum
- A61K39/39533—Antibodies; Immunoglobulins; Immune serum, e.g. antilymphocytic serum against materials from animals
- A61K39/39558—Antibodies; Immunoglobulins; Immune serum, e.g. antilymphocytic serum against materials from animals against tumor tissues, cells, antigens
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
Abstract
La invención proporciona un método para el tratamiento de cánceres incluyendo neoplasias malignas h ematológicas que comprende administrar un compuesto de Fórmula I, en combinación con uno o ambos de bendamustina y rituximab.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201161497356P | 2011-06-15 | 2011-06-15 | |
US201161510324P | 2011-07-21 | 2011-07-21 | |
FR1255114 | 2012-06-01 |
Publications (1)
Publication Number | Publication Date |
---|---|
UY34132A true UY34132A (es) | 2013-01-31 |
Family
ID=47357478
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
UY0001034132A UY34132A (es) | 2011-06-15 | 2012-06-15 | Terapias combinadas para el tratamiento de neoplasias malignas hematológicas utilizando inhibidores de piridopirimidinona de pi3k/mtor con bendamustina y/o rituximab. |
Country Status (9)
Country | Link |
---|---|
US (1) | US20140302012A1 (es) |
EP (1) | EP2793892A1 (es) |
JP (1) | JP2014517042A (es) |
CN (1) | CN103874494A (es) |
AR (1) | AR086955A1 (es) |
RU (1) | RU2014101071A (es) |
TW (1) | TW201306842A (es) |
UY (1) | UY34132A (es) |
WO (1) | WO2012174327A1 (es) |
Families Citing this family (22)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN106420743A (zh) | 2010-07-16 | 2017-02-22 | 埃克塞里艾克西斯公司 | C‑met调节剂药物组合物 |
WO2012037204A1 (en) | 2010-09-14 | 2012-03-22 | Exelixis, Inc. | Inhibitors of pi3k-delta and methods of their use and manufacture |
WO2012044572A1 (en) | 2010-09-27 | 2012-04-05 | Exelixis, Inc. | Dual inhibitors of met and vegf for the treatment of castration- resistant prostate cancer and osteoblastic bone metastases |
BR112013020362A2 (pt) | 2011-02-10 | 2018-05-29 | Exelixis Inc | processos para a preparação de compostos de quinolina, compostos e combinações farmacêuticas que os contem |
US20120252840A1 (en) | 2011-04-04 | 2012-10-04 | Exelixis, Inc. | Method of Treating Cancer |
KR20140025496A (ko) | 2011-05-02 | 2014-03-04 | 엑셀리시스, 인코포레이티드 | 암 및 뼈 암 통증의 치료방법 |
BR112014006702A2 (pt) | 2011-09-22 | 2017-06-13 | Exelixis Inc | método para tratar osteoporose |
CA2852771C (en) | 2011-10-20 | 2019-11-26 | Exelixis, Inc. | Process for preparing quinoline derivatives |
CN107375289A (zh) | 2011-11-01 | 2017-11-24 | 埃克塞利希斯股份有限公司 | 用于治疗淋巴组织增生性恶性肿瘤的作为磷脂酰肌醇3‑激酶抑制剂的化合物 |
JP2015515988A (ja) | 2012-05-02 | 2015-06-04 | エクセリクシス, インク. | 溶骨性骨転移を治療するためのmet−vegf二重調節剤 |
TW201521792A (zh) * | 2013-03-05 | 2015-06-16 | Sanofi Sa | PI3Kα抑制劑之錠劑調配物 |
MX366003B (es) | 2013-03-15 | 2019-06-24 | Exelixis Inc | Metabolitos de n-(4-{[6,7-bis(metiloxi)quinolin-4-il]oxi}fenil)-n' -(4-fluorofenil)ciclopropan-1,1-dicarboxamida. |
US11564915B2 (en) | 2013-04-04 | 2023-01-31 | Exelixis, Inc. | Cabozantinib dosage form and use in the treatment of cancer |
GB201321717D0 (en) | 2013-12-09 | 2014-01-22 | Pharmachemie Bv | Inhalable Medicaments |
MX2021001583A (es) | 2014-02-14 | 2023-02-08 | Exelixis Inc | Formas sólidas cristalinas de n-{4-[(6,7-dimetoxiquinolin-4-il)oxi ] fenil}-n'-(4-fluorofenil)ciclopropan-1,1-dicarboxamida, procesos para elaboración y métodos de uso. |
US10159666B2 (en) | 2014-03-17 | 2018-12-25 | Exelixis, Inc. | Dosing of cabozantinib formulations |
MA40250A (fr) * | 2014-07-04 | 2017-05-10 | Lupin Ltd | Dérivés de quinolizinone utilisés comme inhibiteurs de pi3k |
CN106715397B (zh) | 2014-07-31 | 2021-07-23 | 埃克塞里艾克西斯公司 | 制备氟-18标记的卡博替尼及其类似物的方法 |
EP3177311A1 (en) | 2014-08-05 | 2017-06-14 | Exelixis, Inc. | Drug combinations to treat multiple myeloma |
EP3442531A1 (en) | 2016-04-15 | 2019-02-20 | Exelixis, Inc. | Method of treating renal cell carcinoma using n-(4-(6,7-dimethoxyquinolin-4-yloxy) phenyl)-n'-(4-fluoropheny)cyclopropane-1,1-dicarboxamide, (2s)-hydroxybutanedioate |
LT3497103T (lt) * | 2016-08-15 | 2021-07-26 | Pfizer Inc. | Piridopirimidinono cdk2/4/6 inhibitoriai |
WO2018060804A1 (en) | 2016-09-29 | 2018-04-05 | Telefonaktiebolaget Lm Ericsson (Publ) | Active time handling with 2-step granting |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US20060128777A1 (en) * | 2004-11-05 | 2006-06-15 | Bendall Heather H | Cancer treatments |
BRPI0617159B8 (pt) * | 2005-10-07 | 2021-05-25 | Exelixis Inc | compostos de piridopirimidinone inibidores de pi3ka, composições que os contem e processo para preparo |
WO2008032162A1 (en) * | 2006-09-15 | 2008-03-20 | Pfizer Products Inc. | Pyrido (2, 3-d) pyrimidin0ne compounds and their use as pi3 inhibitors |
UA100979C2 (ru) * | 2007-04-10 | 2013-02-25 | Экселиксис, Инк. | Применение пиридопиримидиноновых ингибиторов pi3k альфа для лечения рака |
WO2012065019A2 (en) * | 2010-11-12 | 2012-05-18 | Exelixis, Inc. | Pyridopyrimidinone inhibitors of p13k alpha |
-
2012
- 2012-06-14 TW TW101121374A patent/TW201306842A/zh unknown
- 2012-06-15 JP JP2014516010A patent/JP2014517042A/ja active Pending
- 2012-06-15 WO PCT/US2012/042582 patent/WO2012174327A1/en active Application Filing
- 2012-06-15 AR ARP120102139A patent/AR086955A1/es unknown
- 2012-06-15 US US14/126,181 patent/US20140302012A1/en not_active Abandoned
- 2012-06-15 RU RU2014101071/15A patent/RU2014101071A/ru unknown
- 2012-06-15 UY UY0001034132A patent/UY34132A/es not_active Application Discontinuation
- 2012-06-15 EP EP12731817.8A patent/EP2793892A1/en not_active Withdrawn
- 2012-06-15 CN CN201280040054.XA patent/CN103874494A/zh active Pending
Also Published As
Publication number | Publication date |
---|---|
CN103874494A (zh) | 2014-06-18 |
AR086955A1 (es) | 2014-02-05 |
WO2012174327A1 (en) | 2012-12-20 |
JP2014517042A (ja) | 2014-07-17 |
TW201306842A (zh) | 2013-02-16 |
EP2793892A1 (en) | 2014-10-29 |
US20140302012A1 (en) | 2014-10-09 |
RU2014101071A (ru) | 2015-07-20 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
109 | Application deemed to be withdrawn |
Effective date: 20201020 |