PL2593090T3 - Kompozycje farmaceutyczne modulatora c-Met - Google Patents

Kompozycje farmaceutyczne modulatora c-Met

Info

Publication number
PL2593090T3
PL2593090T3 PL11740764T PL11740764T PL2593090T3 PL 2593090 T3 PL2593090 T3 PL 2593090T3 PL 11740764 T PL11740764 T PL 11740764T PL 11740764 T PL11740764 T PL 11740764T PL 2593090 T3 PL2593090 T3 PL 2593090T3
Authority
PL
Poland
Prior art keywords
pharmaceutical compositions
modulator pharmaceutical
met
met modulator
compositions
Prior art date
Application number
PL11740764T
Other languages
English (en)
Inventor
Jo Ann WILSON
Original Assignee
Exelixis, Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=45469828&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PL2593090(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Exelixis, Inc. filed Critical Exelixis, Inc.
Publication of PL2593090T3 publication Critical patent/PL2593090T3/pl

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2009Inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • A61K9/2018Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2095Tabletting processes; Dosage units made by direct compression of powders or specially processed granules, by eliminating solvents, by melt-extrusion, by injection molding, by 3D printing
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2893Tablet coating processes
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/286Polysaccharides, e.g. gums; Cyclodextrin
    • A61K9/2866Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
PL11740764T 2010-07-16 2011-07-18 Kompozycje farmaceutyczne modulatora c-Met PL2593090T3 (pl)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US36525310P 2010-07-16 2010-07-16
US37084310P 2010-08-05 2010-08-05
EP11740764.3A EP2593090B1 (en) 2010-07-16 2011-07-18 C-met modulator pharmaceutical compositions
PCT/US2011/044378 WO2012009722A1 (en) 2010-07-16 2011-07-18 C-met modulator pharmaceutical compositions

Publications (1)

Publication Number Publication Date
PL2593090T3 true PL2593090T3 (pl) 2022-02-21

Family

ID=45469828

Family Applications (1)

Application Number Title Priority Date Filing Date
PL11740764T PL2593090T3 (pl) 2010-07-16 2011-07-18 Kompozycje farmaceutyczne modulatora c-Met

Country Status (23)

Country Link
US (9) US9724342B2 (pl)
EP (2) EP4014971A1 (pl)
JP (3) JP5934204B2 (pl)
KR (6) KR20190042768A (pl)
CN (3) CN106420743A (pl)
AR (1) AR082252A1 (pl)
AU (4) AU2011278950C1 (pl)
BR (1) BR112013000980B1 (pl)
CA (1) CA2805645C (pl)
DK (1) DK2593090T3 (pl)
EA (1) EA030435B1 (pl)
ES (1) ES2904646T3 (pl)
HU (1) HUE057184T2 (pl)
IL (2) IL224189A (pl)
LT (1) LT2593090T (pl)
MX (1) MX336741B (pl)
NZ (1) NZ607118A (pl)
PL (1) PL2593090T3 (pl)
PT (1) PT2593090T (pl)
SG (2) SG10201609324UA (pl)
TW (3) TWI619495B (pl)
WO (1) WO2012009722A1 (pl)
ZA (1) ZA201300458B (pl)

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Also Published As

Publication number Publication date
US9724342B2 (en) 2017-08-08
AR082252A1 (es) 2012-11-21
EA201300146A1 (ru) 2013-06-28
PT2593090T (pt) 2021-11-04
JP2019142879A (ja) 2019-08-29
EP2593090A1 (en) 2013-05-22
WO2012009722A1 (en) 2012-01-19
SG187060A1 (en) 2013-02-28
LT2593090T (lt) 2022-01-10
US20200121671A1 (en) 2020-04-23
AU2018220045B2 (en) 2020-03-05
CA2805645A1 (en) 2012-01-19
TW201219371A (en) 2012-05-16
ZA201300458B (en) 2013-09-25
EP4014971A1 (en) 2022-06-22
KR20220005631A (ko) 2022-01-13
JP2013531045A (ja) 2013-08-01
TW201735925A (zh) 2017-10-16
JP5934204B2 (ja) 2016-06-15
DK2593090T3 (da) 2021-10-25
EA030435B1 (ru) 2018-08-31
US20130337015A1 (en) 2013-12-19
AU2011278950B2 (en) 2016-07-21
IL253333A0 (en) 2017-09-28
BR112013000980B1 (pt) 2022-08-16
US20210379050A1 (en) 2021-12-09
KR20200029633A (ko) 2020-03-18
AU2011278950C1 (en) 2018-11-22
NZ607118A (en) 2015-05-29
TWI516477B (zh) 2016-01-11
EP2593090B1 (en) 2021-10-13
CN114209699A (zh) 2022-03-22
AU2016247044A1 (en) 2016-11-03
CN106420743A (zh) 2017-02-22
US20170266178A1 (en) 2017-09-21
KR20130137586A (ko) 2013-12-17
US20170143689A1 (en) 2017-05-25
US10039757B2 (en) 2018-08-07
IL224189A (en) 2017-07-31
AU2011278950A1 (en) 2013-03-07
ES2904646T3 (es) 2022-04-05
KR20190042768A (ko) 2019-04-24
KR20180056807A (ko) 2018-05-29
KR101862324B1 (ko) 2018-05-29
BR112013000980A2 (pt) 2018-03-13
TW201602083A (zh) 2016-01-16
CA2805645C (en) 2019-05-07
SG10201609324UA (en) 2017-01-27
KR20210014770A (ko) 2021-02-09
US20180311229A1 (en) 2018-11-01
MX2013000567A (es) 2013-05-01
AU2018220045A1 (en) 2018-09-06
MX336741B (es) 2016-01-29
AU2020203645A1 (en) 2020-06-25
US20220031688A1 (en) 2022-02-03
TWI619495B (zh) 2018-04-01
US11123338B2 (en) 2021-09-21
US10034873B2 (en) 2018-07-31
HUE057184T2 (hu) 2022-04-28
US20220370436A1 (en) 2022-11-24
JP2016188215A (ja) 2016-11-04
US20220087999A1 (en) 2022-03-24
US10548888B2 (en) 2020-02-04
JP6503317B2 (ja) 2019-04-17
CN103221035A (zh) 2013-07-24

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