SI21507A - Postopek za pripravo spojin z ace inhibitornim delovanjem - Google Patents
Postopek za pripravo spojin z ace inhibitornim delovanjem Download PDFInfo
- Publication number
- SI21507A SI21507A SI200300123A SI200300123A SI21507A SI 21507 A SI21507 A SI 21507A SI 200300123 A SI200300123 A SI 200300123A SI 200300123 A SI200300123 A SI 200300123A SI 21507 A SI21507 A SI 21507A
- Authority
- SI
- Slovenia
- Prior art keywords
- preparation
- compounds
- ace inhibitory
- activated
- inhibitory activity
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D207/16—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
- C07D209/42—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Peptides Or Proteins (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Priority Applications (8)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
SI200300123A SI21507A (sl) | 2003-05-16 | 2003-05-16 | Postopek za pripravo spojin z ace inhibitornim delovanjem |
DE602004030112T DE602004030112D1 (de) | 2003-05-16 | 2004-05-07 | Verfahren zur herstellung von ace hemmern |
PCT/SI2004/000021 WO2004101515A1 (fr) | 2003-05-16 | 2004-05-07 | Procede de preparation de composes ayant une action inhibitrice sur ace |
EP04731808A EP1628956B1 (fr) | 2003-05-16 | 2004-05-07 | Procede de preparation de composes ayant une action inhibitrice sur ace |
US10/556,986 US7671215B2 (en) | 2003-05-16 | 2004-05-07 | Process for the preparation of compounds having an ace inhibitory action |
SI200431600T SI1628956T1 (sl) | 2003-05-16 | 2004-05-07 | Postopek za pripravo spojin z ACE inhibitornim delovanjem |
AT04731808T ATE488498T1 (de) | 2003-05-16 | 2004-05-07 | Verfahren zur herstellung von ace hemmern |
RU2005139158/04A RU2377236C2 (ru) | 2003-05-16 | 2004-05-07 | Способ получения соединений, обладающих апф ингибиторной активностью |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
SI200300123A SI21507A (sl) | 2003-05-16 | 2003-05-16 | Postopek za pripravo spojin z ace inhibitornim delovanjem |
Publications (1)
Publication Number | Publication Date |
---|---|
SI21507A true SI21507A (sl) | 2004-12-31 |
Family
ID=33448812
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SI200300123A SI21507A (sl) | 2003-05-16 | 2003-05-16 | Postopek za pripravo spojin z ace inhibitornim delovanjem |
SI200431600T SI1628956T1 (sl) | 2003-05-16 | 2004-05-07 | Postopek za pripravo spojin z ACE inhibitornim delovanjem |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SI200431600T SI1628956T1 (sl) | 2003-05-16 | 2004-05-07 | Postopek za pripravo spojin z ACE inhibitornim delovanjem |
Country Status (7)
Country | Link |
---|---|
US (1) | US7671215B2 (fr) |
EP (1) | EP1628956B1 (fr) |
AT (1) | ATE488498T1 (fr) |
DE (1) | DE602004030112D1 (fr) |
RU (1) | RU2377236C2 (fr) |
SI (2) | SI21507A (fr) |
WO (1) | WO2004101515A1 (fr) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US20080188545A1 (en) * | 2006-12-21 | 2008-08-07 | Alimardanov Asaf R | Synthesis of pyrrolidine compounds |
US20090076126A1 (en) * | 2007-09-17 | 2009-03-19 | Protia, Llc | Deuterium-enriched enalapril |
RU2012103753A (ru) | 2009-07-16 | 2013-08-27 | Эбботт Лабораториз | Способ синтеза (2s, 3ar, 7as)-октагидро-1н-индол-карбоновой кислоты в качестве промежуточного соединения для получения трандолаприла |
ES2670854T3 (es) * | 2012-10-10 | 2018-06-01 | Piramal Enterprises Limited | Un proceso mejorado para la preparación de perindoprilo intermedio |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
NL4915C (fr) | 1913-08-18 | |||
FR2620709B1 (fr) * | 1987-09-17 | 1990-09-07 | Adir | Procede de synthese industrielle du perindopril et de ses principaux intermediaires de synthese |
US5864040A (en) | 1996-01-11 | 1999-01-26 | American Home Products Corporation | Benzimidazole phosphono-amino acids |
GB9710612D0 (en) | 1997-05-23 | 1997-07-16 | Glaxo Group Ltd | Synthesis of acridine derivatives |
UA73553C2 (en) | 2000-03-31 | 2005-08-15 | Pfizer Prod Inc | Piperazine derivatives |
GB2375762B (en) * | 2001-05-21 | 2003-10-01 | Fermenta Biotech Ltd | Stereospecific synthesis of 2-hydroxy-4-phenyl-butyric acid esters |
WO2002094857A1 (fr) | 2001-05-23 | 2002-11-28 | The Curators Of The University Of Missouri | Synthese peptidique en phase solide inverse |
AR036187A1 (es) * | 2001-07-24 | 2004-08-18 | Adir | Un proceso para la preparacion de perindopril, compuestos analogos y sus sales, compuesto intermediario 2,5-dioxo-oxazolidina y proceso para preparar un intermediario |
GB0119795D0 (en) | 2001-08-14 | 2001-10-03 | Smithkline Beecham Plc | Novel process |
-
2003
- 2003-05-16 SI SI200300123A patent/SI21507A/sl not_active IP Right Cessation
-
2004
- 2004-05-07 SI SI200431600T patent/SI1628956T1/sl unknown
- 2004-05-07 DE DE602004030112T patent/DE602004030112D1/de not_active Expired - Lifetime
- 2004-05-07 AT AT04731808T patent/ATE488498T1/de not_active IP Right Cessation
- 2004-05-07 RU RU2005139158/04A patent/RU2377236C2/ru not_active IP Right Cessation
- 2004-05-07 EP EP04731808A patent/EP1628956B1/fr not_active Expired - Lifetime
- 2004-05-07 WO PCT/SI2004/000021 patent/WO2004101515A1/fr active Application Filing
- 2004-05-07 US US10/556,986 patent/US7671215B2/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
RU2005139158A (ru) | 2007-06-27 |
SI1628956T1 (sl) | 2011-03-31 |
WO2004101515A1 (fr) | 2004-11-25 |
ATE488498T1 (de) | 2010-12-15 |
DE602004030112D1 (de) | 2010-12-30 |
RU2377236C2 (ru) | 2009-12-27 |
EP1628956B1 (fr) | 2010-11-17 |
US20070072919A1 (en) | 2007-03-29 |
US7671215B2 (en) | 2010-03-02 |
EP1628956A1 (fr) | 2006-03-01 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
IF | Valid on the event date | ||
OO00 | Grant of patent |
Effective date: 20031011 |
|
KO00 | Lapse of patent |
Effective date: 20130523 |