SI1720852T1 - Postopek za pripravo enantiomerno čistih substituiranih aminoalkoholov - Google Patents
Postopek za pripravo enantiomerno čistih substituiranih aminoalkoholovInfo
- Publication number
- SI1720852T1 SI1720852T1 SI200531602T SI200531602T SI1720852T1 SI 1720852 T1 SI1720852 T1 SI 1720852T1 SI 200531602 T SI200531602 T SI 200531602T SI 200531602 T SI200531602 T SI 200531602T SI 1720852 T1 SI1720852 T1 SI 1720852T1
- Authority
- SI
- Slovenia
- Prior art keywords
- aminoalcohols
- substituted
- preparation
- enantiomerically pure
- enantiomerically
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
- C07D333/14—Radicals substituted by singly bound hetero atoms other than halogen
- C07D333/20—Radicals substituted by singly bound hetero atoms other than halogen by nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C213/00—Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
- C07D307/04—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
- C07D307/18—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D307/22—Nitrogen atoms not forming part of a nitro radical
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
- C07D333/22—Radicals substituted by doubly bound hetero atoms, or by two hetero atoms other than halogen singly bound to the same carbon atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/07—Optical isomers
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Heterocyclic Compounds Containing Sulfur Atoms (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Furan Compounds (AREA)
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP04003809A EP1566383A1 (en) | 2004-02-19 | 2004-02-19 | Process for the preparation of enantiomerically pure 1-substituted-3-aminoalcohols |
EP04010043 | 2004-04-28 | ||
PCT/EP2005/001781 WO2005080370A1 (en) | 2004-02-19 | 2005-02-21 | Process for the preparation of enantiomerically pure 1-substituted-3-aminoalcohols |
EP05715425A EP1720852B1 (en) | 2004-02-19 | 2005-02-21 | Process for the preparation of enantiomerically pure 1-substituted-3-aminoalcohols |
Publications (1)
Publication Number | Publication Date |
---|---|
SI1720852T1 true SI1720852T1 (sl) | 2012-11-30 |
Family
ID=34889010
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SI200531602T SI1720852T1 (sl) | 2004-02-19 | 2005-02-21 | Postopek za pripravo enantiomerno čistih substituiranih aminoalkoholov |
Country Status (20)
Country | Link |
---|---|
US (3) | US7973182B2 (sl) |
EP (1) | EP1720852B1 (sl) |
JP (2) | JP2007523124A (sl) |
KR (1) | KR101160502B1 (sl) |
CN (1) | CN102627572A (sl) |
AU (1) | AU2005215906C1 (sl) |
BR (1) | BRPI0506796A (sl) |
CA (1) | CA2556891C (sl) |
CY (1) | CY1113261T1 (sl) |
DK (1) | DK1720852T3 (sl) |
EA (1) | EA200601513A1 (sl) |
ES (1) | ES2391399T3 (sl) |
IL (1) | IL177561A (sl) |
NO (1) | NO20064017L (sl) |
NZ (1) | NZ549381A (sl) |
PL (1) | PL1720852T3 (sl) |
PT (1) | PT1720852E (sl) |
SG (1) | SG135196A1 (sl) |
SI (1) | SI1720852T1 (sl) |
WO (1) | WO2005080370A1 (sl) |
Families Citing this family (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
BRPI0506796A (pt) | 2004-02-19 | 2007-05-22 | Lonza Ag | processo para a preparação de 1-substituìdos-3-aminoálcoois enantiomericamentente puros |
EP1868983A1 (en) * | 2005-02-21 | 2007-12-26 | Lonza Ag | Process for the preparation of enantiomerically pure 1-substituted-3-aminoalcohols |
CN101484435A (zh) | 2006-07-03 | 2009-07-15 | 兰贝克赛实验室有限公司 | 制备n-甲基-3-(1-萘氧基)-3-(2-噻吩基)丙胺及其纯对应异构体盐的方法 |
WO2010025238A2 (en) | 2008-08-27 | 2010-03-04 | Codexis, Inc. | Ketoreductase polypeptides for the production of a 3-aryl-3-hydroxypropanamine from a 3-aryl-3-ketopropanamine |
US8288141B2 (en) | 2008-08-27 | 2012-10-16 | Codexis, Inc. | Ketoreductase polypeptides for the production of 3-aryl-3-hydroxypropanamine from a 3-aryl-3-ketopropanamine |
SI2558455T1 (sl) | 2010-04-13 | 2017-12-29 | Krka, D.D., Novo Mesto | Sinteza duloksetina in/ali njegovih farmacevtsko sprejemljivih soli |
CN104056663B (zh) * | 2013-03-22 | 2016-12-28 | 上海交通大学 | 一种面手性双反应中心钌催化剂及其合成与应用 |
CN110054563A (zh) * | 2019-06-10 | 2019-07-26 | 江西隆莱生物制药有限公司 | 丁内酯类化合物的制备方法及其中间体 |
CN111793056A (zh) * | 2020-07-27 | 2020-10-20 | 广州康瑞泰药业有限公司 | 一种度洛西汀中间体的制备方法 |
Family Cites Families (21)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE3031248A1 (de) | 1980-08-19 | 1982-04-01 | Ruhrchemie Ag, 4200 Oberhausen | Verfahren zur herstellung von 3-dimethylamino-2,2-dimethylpropanal |
US5362866A (en) | 1983-09-02 | 1994-11-08 | Molecular Biosystems, Inc. | Oligonucleotide polymeric support system with an oxidation cleavable link |
KR880007433A (ko) * | 1986-12-22 | 1988-08-27 | 메리 앤 터커 | 3-아릴옥시-3-치환된 프로판아민 |
US4948813A (en) | 1987-11-30 | 1990-08-14 | E. I. Du Pont De Nemours And Company | Benzylketone phospholipase A2 inhibitors |
CA2042346A1 (en) * | 1990-05-17 | 1991-11-18 | Michael Alexander Staszak | Chiral synthesis of 1-aryl-3-aminopropan-1-ols |
JPH0570412A (ja) * | 1991-09-13 | 1993-03-23 | Fuji Yakuhin Kogyo Kk | 光学活性なβ−アミノアルコールの製造方法 |
US5491234A (en) * | 1992-03-30 | 1996-02-13 | Pfizer Inc. | Pyrimidine derivatives for enhancing antitumor activity |
ATE177427T1 (de) | 1993-10-08 | 1999-03-15 | Hoffmann La Roche | Optisch aktive phosphorverbindungen |
US5362886A (en) | 1993-10-12 | 1994-11-08 | Eli Lilly And Company | Asymmetric synthesis |
IT1270082B (it) * | 1994-07-12 | 1997-04-28 | Univ Degli Studi Milano | Difosfine eteroaromatiche come leganti chirali, complessi tra dette difosfine e metalli di transizione ed impiego di detti complessi come catalizzatori chirali |
TW514634B (en) * | 1997-10-14 | 2002-12-21 | Lilly Co Eli | Process to make chiral compounds |
US6008412A (en) * | 1997-10-14 | 1999-12-28 | Eli Lilly And Company | Process to make chiral compounds |
US6162929A (en) | 1997-12-23 | 2000-12-19 | Hoffmann-La Roche Inc. | Process for the manufacture of bisphosphine oxide and bisphosphonate compounds |
JP3549390B2 (ja) | 1998-03-23 | 2004-08-04 | 高砂香料工業株式会社 | ルテニウム−ホスフィン錯体及びその製造方法 |
DE69933904T2 (de) | 1998-05-08 | 2007-09-06 | Takasago International Corp. | Ruthenium-iodo optisch aktiver Phosphinkomplex |
FR2816946B1 (fr) | 2000-11-17 | 2004-04-02 | Ppg Sipsy | Diphosphines chirales dissymetriques, leurs utilisations pour la preparation de complexes diphosphino-metalliques, et les complexes diphosphino-metalliques ainsi obtenus |
DE10207586A1 (de) * | 2002-02-22 | 2003-09-11 | Degussa | Herstellung von N-Methyl-3-hydroxy-3-(2-thienyl)propanamin über neue carbamatgruppenhaltige Thiophenderivate als Zwischenprodukte |
WO2004005239A1 (en) | 2002-07-09 | 2004-01-15 | Lonza Ag | PROCESS FOR THE PREPARATION OF N-MONOSUBSTITUTED β-AMINO ALCOHOLS |
FR2841899A1 (fr) | 2002-07-05 | 2004-01-09 | Ppg Sipsy | Procede de resolution asymetrique d'un racemique faisant intervenir l'acide diprogulique et utilisation dudit acide comme agent de resolution asymetrique |
WO2004005307A1 (en) * | 2002-07-09 | 2004-01-15 | Lonza Ag | Process for the preparation of optically active 3-n-methylamino-1-(2-thienyl)-1-propanol |
BRPI0506796A (pt) | 2004-02-19 | 2007-05-22 | Lonza Ag | processo para a preparação de 1-substituìdos-3-aminoálcoois enantiomericamentente puros |
-
2005
- 2005-02-21 BR BRPI0506796-0A patent/BRPI0506796A/pt not_active IP Right Cessation
- 2005-02-21 WO PCT/EP2005/001781 patent/WO2005080370A1/en active Application Filing
- 2005-02-21 PL PL05715425T patent/PL1720852T3/pl unknown
- 2005-02-21 JP JP2006553562A patent/JP2007523124A/ja active Pending
- 2005-02-21 CA CA2556891A patent/CA2556891C/en not_active Expired - Fee Related
- 2005-02-21 US US10/590,140 patent/US7973182B2/en not_active Expired - Fee Related
- 2005-02-21 PT PT05715425T patent/PT1720852E/pt unknown
- 2005-02-21 NZ NZ549381A patent/NZ549381A/en not_active IP Right Cessation
- 2005-02-21 SG SG200706103-9A patent/SG135196A1/en unknown
- 2005-02-21 ES ES05715425T patent/ES2391399T3/es active Active
- 2005-02-21 CN CN2012100464149A patent/CN102627572A/zh active Pending
- 2005-02-21 SI SI200531602T patent/SI1720852T1/sl unknown
- 2005-02-21 EP EP05715425A patent/EP1720852B1/en not_active Not-in-force
- 2005-02-21 EA EA200601513A patent/EA200601513A1/ru unknown
- 2005-02-21 DK DK05715425.4T patent/DK1720852T3/da active
- 2005-02-21 KR KR1020067018840A patent/KR101160502B1/ko not_active IP Right Cessation
- 2005-02-21 AU AU2005215906A patent/AU2005215906C1/en not_active Ceased
-
2006
- 2006-08-17 IL IL177561A patent/IL177561A/en not_active IP Right Cessation
- 2006-09-06 NO NO20064017A patent/NO20064017L/no not_active Application Discontinuation
-
2011
- 2011-03-08 US US13/064,146 patent/US8198468B2/en not_active Expired - Fee Related
- 2011-03-08 US US13/064,147 patent/US8193380B2/en not_active Expired - Fee Related
-
2012
- 2012-06-14 JP JP2012134968A patent/JP2012229223A/ja not_active Withdrawn
- 2012-10-10 CY CY20121100937T patent/CY1113261T1/el unknown
Also Published As
Publication number | Publication date |
---|---|
PT1720852E (pt) | 2012-10-22 |
PL1720852T3 (pl) | 2012-12-31 |
IL177561A (en) | 2011-12-29 |
SG135196A1 (en) | 2007-09-28 |
US8198468B2 (en) | 2012-06-12 |
US8193380B2 (en) | 2012-06-05 |
CA2556891C (en) | 2012-12-18 |
AU2005215906C1 (en) | 2012-03-01 |
EP1720852A1 (en) | 2006-11-15 |
JP2012229223A (ja) | 2012-11-22 |
BRPI0506796A (pt) | 2007-05-22 |
AU2005215906B2 (en) | 2011-08-18 |
KR20070009587A (ko) | 2007-01-18 |
CY1113261T1 (el) | 2016-04-13 |
US20110207946A1 (en) | 2011-08-25 |
NZ549381A (en) | 2010-05-28 |
NO20064017L (no) | 2006-09-15 |
EP1720852B1 (en) | 2012-07-11 |
US7973182B2 (en) | 2011-07-05 |
ES2391399T3 (es) | 2012-11-26 |
CA2556891A1 (en) | 2005-09-01 |
WO2005080370A1 (en) | 2005-09-01 |
US20080154047A1 (en) | 2008-06-26 |
KR101160502B1 (ko) | 2012-06-28 |
DK1720852T3 (da) | 2012-10-22 |
AU2005215906A1 (en) | 2005-09-01 |
IL177561A0 (en) | 2006-12-10 |
CN102627572A (zh) | 2012-08-08 |
JP2007523124A (ja) | 2007-08-16 |
EA200601513A1 (ru) | 2007-02-27 |
US20110207945A1 (en) | 2011-08-25 |
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