SI1544199T1 - Spojina, ki ima kondenziran obroč in vsebuje dušik, in njena uporaba kot inhibitor HIV integraze - Google Patents
Spojina, ki ima kondenziran obroč in vsebuje dušik, in njena uporaba kot inhibitor HIV integrazeInfo
- Publication number
- SI1544199T1 SI1544199T1 SI200430973T SI200430973T SI1544199T1 SI 1544199 T1 SI1544199 T1 SI 1544199T1 SI 200430973 T SI200430973 T SI 200430973T SI 200430973 T SI200430973 T SI 200430973T SI 1544199 T1 SI1544199 T1 SI 1544199T1
- Authority
- SI
- Slovenia
- Prior art keywords
- ring compound
- hiv integrase
- integrase inhibitor
- nitrogenous condensed
- nitrogenous
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Communicable Diseases (AREA)
- Virology (AREA)
- Oncology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- AIDS & HIV (AREA)
- Tropical Medicine & Parasitology (AREA)
- Molecular Biology (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2003293117 | 2003-08-13 | ||
JP2004134896 | 2004-04-28 | ||
EP04771830A EP1544199B1 (en) | 2003-08-13 | 2004-08-12 | Nitrogenous condensed-ring compound and use thereof as hiv integrase inhibitor |
PCT/JP2004/011869 WO2005016927A1 (ja) | 2003-08-13 | 2004-08-12 | 含窒素縮合環化合物及びそのhivインテグラーゼ阻害剤としての利用 |
Publications (1)
Publication Number | Publication Date |
---|---|
SI1544199T1 true SI1544199T1 (sl) | 2009-04-30 |
Family
ID=34197143
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SI200430973T SI1544199T1 (sl) | 2003-08-13 | 2004-08-12 | Spojina, ki ima kondenziran obroč in vsebuje dušik, in njena uporaba kot inhibitor HIV integraze |
Country Status (15)
Country | Link |
---|---|
US (3) | US20050054645A1 (sl) |
EP (2) | EP2042502A1 (sl) |
JP (1) | JP3814631B2 (sl) |
AR (1) | AR045367A1 (sl) |
AT (1) | ATE411315T1 (sl) |
CA (1) | CA2577239A1 (sl) |
CL (1) | CL2004002061A1 (sl) |
DE (1) | DE602004017108D1 (sl) |
DK (1) | DK1544199T3 (sl) |
ES (1) | ES2315700T3 (sl) |
PE (1) | PE20050361A1 (sl) |
PT (1) | PT1544199E (sl) |
SI (1) | SI1544199T1 (sl) |
TW (1) | TW200510425A (sl) |
WO (1) | WO2005016927A1 (sl) |
Families Citing this family (119)
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US7732616B2 (en) * | 2003-11-19 | 2010-06-08 | Array Biopharma Inc. | Dihydropyridine and dihydropyridazine derivatives as inhibitors of MEK and methods of use thereof |
US7517994B2 (en) * | 2003-11-19 | 2009-04-14 | Array Biopharma Inc. | Heterocyclic inhibitors of MEK and methods of use thereof |
WO2005051302A2 (en) * | 2003-11-19 | 2005-06-09 | Array Biopharma Inc. | Bicyclic inhibitors of mek and methods of use thereof |
US20050182252A1 (en) | 2004-02-13 | 2005-08-18 | Reddy K. R. | Novel 2'-C-methyl nucleoside derivatives |
CA2557926A1 (en) * | 2004-03-09 | 2005-09-22 | Monica Donghi | Hiv integrase inhibitors |
WO2005092099A1 (en) * | 2004-03-09 | 2005-10-06 | Merck & Co., Inc. | Hiv integrase inhibitors |
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AU2005222391B2 (en) * | 2004-03-09 | 2010-11-11 | Merck Sharp & Dohme Corp. | HIV integrase inhibitors |
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US7745459B2 (en) * | 2004-09-21 | 2010-06-29 | Japan Tobacco Inc. | Quinolizinone compound and use thereof as HIV integrase inhibitor |
EP1852434B1 (en) * | 2005-02-21 | 2011-07-13 | Shionogi Co., Ltd. | Bicyclic carbamoylpyridone derivative having hiv integrase inhibiting activity |
CA2600832C (en) * | 2005-03-31 | 2011-12-13 | Istituto Di Ricerche Di Biologia Molecolare P. Angeletti S.P.A. | Hiv integrase inhibitors |
DK2465580T3 (en) | 2005-04-28 | 2014-03-10 | Viiv Healthcare Co | POLYCYCLIC CARBAMOYL PYRIDONE DERIVATIVES WITH HIV INTEGRASE INHIBITIVE ACTIVITY |
CA2606195C (en) | 2005-05-02 | 2015-03-31 | Merck And Co., Inc. | Hcv ns3 protease inhibitors |
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-
2004
- 2004-08-11 TW TW093124129A patent/TW200510425A/zh unknown
- 2004-08-12 ES ES04771830T patent/ES2315700T3/es not_active Expired - Lifetime
- 2004-08-12 PT PT04771830T patent/PT1544199E/pt unknown
- 2004-08-12 SI SI200430973T patent/SI1544199T1/sl unknown
- 2004-08-12 DK DK04771830T patent/DK1544199T3/da active
- 2004-08-12 DE DE602004017108T patent/DE602004017108D1/de not_active Expired - Lifetime
- 2004-08-12 EP EP08166109A patent/EP2042502A1/en not_active Withdrawn
- 2004-08-12 CA CA002577239A patent/CA2577239A1/en not_active Abandoned
- 2004-08-12 EP EP04771830A patent/EP1544199B1/en not_active Expired - Lifetime
- 2004-08-12 JP JP2005513209A patent/JP3814631B2/ja not_active Expired - Fee Related
- 2004-08-12 WO PCT/JP2004/011869 patent/WO2005016927A1/ja active Application Filing
- 2004-08-12 AT AT04771830T patent/ATE411315T1/de not_active IP Right Cessation
- 2004-08-13 AR ARP040102913A patent/AR045367A1/es unknown
- 2004-08-13 CL CL200402061A patent/CL2004002061A1/es unknown
- 2004-08-13 PE PE2004000787A patent/PE20050361A1/es not_active Application Discontinuation
- 2004-10-05 US US10/958,225 patent/US20050054645A1/en not_active Abandoned
-
2005
- 2005-10-13 US US11/255,605 patent/US7211572B2/en active Active
-
2007
- 2007-04-06 US US11/783,270 patent/US20080161311A1/en not_active Abandoned
Also Published As
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TW200510425A (en) | 2005-03-16 |
US20080161311A1 (en) | 2008-07-03 |
ES2315700T3 (es) | 2009-04-01 |
WO2005016927A1 (ja) | 2005-02-24 |
US20050054645A1 (en) | 2005-03-10 |
DK1544199T3 (da) | 2009-01-12 |
EP2042502A1 (en) | 2009-04-01 |
JP3814631B2 (ja) | 2006-08-30 |
AR045367A1 (es) | 2005-10-26 |
ATE411315T1 (de) | 2008-10-15 |
JPWO2005016927A1 (ja) | 2006-10-12 |
PT1544199E (pt) | 2008-12-03 |
EP1544199A4 (en) | 2006-07-26 |
US7211572B2 (en) | 2007-05-01 |
DE602004017108D1 (de) | 2008-11-27 |
EP1544199B1 (en) | 2008-10-15 |
CL2004002061A1 (es) | 2005-06-03 |
US20060052361A1 (en) | 2006-03-09 |
PE20050361A1 (es) | 2005-06-27 |
EP1544199A1 (en) | 2005-06-22 |
CA2577239A1 (en) | 2005-02-24 |
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