SI1476141T1 - Naprave za transdermalno dajanje opoida, zaščitene pred nedovoljenimi posegi - Google Patents
Naprave za transdermalno dajanje opoida, zaščitene pred nedovoljenimi posegiInfo
- Publication number
- SI1476141T1 SI1476141T1 SI200331243T SI200331243T SI1476141T1 SI 1476141 T1 SI1476141 T1 SI 1476141T1 SI 200331243 T SI200331243 T SI 200331243T SI 200331243 T SI200331243 T SI 200331243T SI 1476141 T1 SI1476141 T1 SI 1476141T1
- Authority
- SI
- Slovenia
- Prior art keywords
- tamper
- patient
- pharmaceutically acceptable
- acceptable salt
- opioid
- Prior art date
Links
- 150000003839 salts Chemical class 0.000 abstract 3
- 230000037317 transdermal delivery Effects 0.000 abstract 3
- 125000002252 acyl group Chemical group 0.000 abstract 2
- 238000000034 method Methods 0.000 abstract 1
- 239000003887 narcotic antagonist Substances 0.000 abstract 1
- 239000003401 opiate antagonist Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/70—Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
- A61K9/7023—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
- A61K9/703—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
- A61K9/7084—Transdermal patches having a drug layer or reservoir, and one or more separate drug-free skin-adhesive layers, e.g. between drug reservoir and skin, or surrounding the drug reservoir; Liquid-filled reservoir patches
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/485—Morphinan derivatives, e.g. morphine, codeine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/36—Opioid-abuse
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D489/00—Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula:
- C07D489/06—Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula: with a hetero atom directly attached in position 14
- C07D489/08—Oxygen atom
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- Dermatology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Addiction (AREA)
- Emergency Medicine (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US35714102P | 2002-02-19 | 2002-02-19 | |
| US35713902P | 2002-02-19 | 2002-02-19 | |
| PCT/US2003/004999 WO2003070191A2 (en) | 2002-02-19 | 2003-02-19 | Tamper-resistant transdermal opioid delivery devices |
| EP03742830A EP1476141B1 (en) | 2002-02-19 | 2003-02-19 | Tamper-resistant transdermal opioid delivery devices |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| SI1476141T1 true SI1476141T1 (sl) | 2008-08-31 |
Family
ID=27760456
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SI200331243T SI1476141T1 (sl) | 2002-02-19 | 2003-02-19 | Naprave za transdermalno dajanje opoida, zaščitene pred nedovoljenimi posegi |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US20040033253A1 (enExample) |
| EP (1) | EP1476141B1 (enExample) |
| JP (3) | JP4874523B2 (enExample) |
| AT (1) | ATE392892T1 (enExample) |
| AU (1) | AU2003216321A1 (enExample) |
| CY (1) | CY1108201T1 (enExample) |
| DE (1) | DE60320530T2 (enExample) |
| DK (1) | DK1476141T3 (enExample) |
| ES (1) | ES2305480T3 (enExample) |
| PT (1) | PT1476141E (enExample) |
| SI (1) | SI1476141T1 (enExample) |
| WO (1) | WO2003070191A2 (enExample) |
Families Citing this family (71)
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| US8790689B2 (en) * | 2003-04-30 | 2014-07-29 | Purdue Pharma L.P. | Tamper resistant transdermal dosage form |
| DE102005005446A1 (de) | 2005-02-04 | 2006-08-10 | Grünenthal GmbH | Bruchfeste Darreichungsformen mit retardierter Freisetzung |
| US20070048228A1 (en) | 2003-08-06 | 2007-03-01 | Elisabeth Arkenau-Maric | Abuse-proofed dosage form |
| DE10361596A1 (de) | 2003-12-24 | 2005-09-29 | Grünenthal GmbH | Verfahren zur Herstellung einer gegen Missbrauch gesicherten Darreichungsform |
| DE10336400A1 (de) | 2003-08-06 | 2005-03-24 | Grünenthal GmbH | Gegen Missbrauch gesicherte Darreichungsform |
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-
2003
- 2003-02-14 US US10/366,394 patent/US20040033253A1/en not_active Abandoned
- 2003-02-19 WO PCT/US2003/004999 patent/WO2003070191A2/en not_active Ceased
- 2003-02-19 JP JP2003569151A patent/JP4874523B2/ja not_active Expired - Fee Related
- 2003-02-19 EP EP03742830A patent/EP1476141B1/en not_active Expired - Lifetime
- 2003-02-19 PT PT03742830T patent/PT1476141E/pt unknown
- 2003-02-19 AT AT03742830T patent/ATE392892T1/de active
- 2003-02-19 ES ES03742830T patent/ES2305480T3/es not_active Expired - Lifetime
- 2003-02-19 SI SI200331243T patent/SI1476141T1/sl unknown
- 2003-02-19 DK DK03742830T patent/DK1476141T3/da active
- 2003-02-19 AU AU2003216321A patent/AU2003216321A1/en not_active Abandoned
- 2003-02-19 DE DE60320530T patent/DE60320530T2/de not_active Expired - Lifetime
-
2008
- 2008-07-17 CY CY20081100746T patent/CY1108201T1/el unknown
-
2010
- 2010-03-29 JP JP2010075835A patent/JP5453151B2/ja not_active Expired - Fee Related
-
2013
- 2013-08-02 JP JP2013160887A patent/JP2013237692A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| DK1476141T3 (da) | 2008-08-18 |
| JP5453151B2 (ja) | 2014-03-26 |
| JP2013237692A (ja) | 2013-11-28 |
| EP1476141A2 (en) | 2004-11-17 |
| DE60320530T2 (de) | 2009-06-10 |
| JP2010189403A (ja) | 2010-09-02 |
| WO2003070191A8 (en) | 2004-06-10 |
| DE60320530D1 (de) | 2008-06-05 |
| EP1476141B1 (en) | 2008-04-23 |
| ATE392892T1 (de) | 2008-05-15 |
| PT1476141E (pt) | 2008-07-03 |
| WO2003070191A3 (en) | 2004-09-10 |
| JP4874523B2 (ja) | 2012-02-15 |
| JP2006502967A (ja) | 2006-01-26 |
| ES2305480T3 (es) | 2008-11-01 |
| AU2003216321A1 (en) | 2003-09-09 |
| WO2003070191A2 (en) | 2003-08-28 |
| CY1108201T1 (el) | 2014-02-12 |
| AU2003216321A8 (en) | 2003-09-09 |
| US20040033253A1 (en) | 2004-02-19 |
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