SI1038863T1 - Novi substituirani dimerni derivati, postopek za njihovo pripravo in farmacevtski pripravki, ki jih vsebujejo - Google Patents

Novi substituirani dimerni derivati, postopek za njihovo pripravo in farmacevtski pripravki, ki jih vsebujejo

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Publication number
SI1038863T1
SI1038863T1 SI200030120T SI200030120T SI1038863T1 SI 1038863 T1 SI1038863 T1 SI 1038863T1 SI 200030120 T SI200030120 T SI 200030120T SI 200030120 T SI200030120 T SI 200030120T SI 1038863 T1 SI1038863 T1 SI 1038863T1
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SI
Slovenia
Prior art keywords
alkyl
indol
ring
heteroaryl
halogen
Prior art date
Application number
SI200030120T
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Unknown language ( )
English (en)
Inventor
Daniel Lesieur
Said Yous
Carole Descamps-Francois
Francois Lefoulon
Gerald Guillaumet
Marie-Claude Viaud
Caroline Bennejean
Philippe Delagrange
Pierre Renard
Original Assignee
Les Laboratoires Servier
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Publication date
Application filed by Les Laboratoires Servier filed Critical Les Laboratoires Servier
Publication of SI1038863T1 publication Critical patent/SI1038863T1/sl

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    • C07D339/00—Heterocyclic compounds containing rings having two sulfur atoms as the only ring hetero atoms
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
    • C07D307/79—Benzo [b] furans; Hydrogenated benzo [b] furans with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
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    • C07C233/16—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms
    • C07C233/17—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom
    • C07C233/18—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom having the carbon atom of the carboxamide group bound to a hydrogen atom or to a carbon atom of an acyclic saturated carbon skeleton
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    • C07C233/16—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms
    • C07C233/17—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom
    • C07C233/20—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom having the carbon atom of the carboxamide group bound to a carbon atom of an acyclic unsaturated carbon skeleton
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    • C07C233/36—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by amino groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom having the carbon atom of the carboxamide group bound to a hydrogen atom or to a carbon atom of an acyclic saturated carbon skeleton
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    • C07C233/60—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of rings other than six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms
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    • C07C233/68—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom
    • C07C233/73—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom of a carbon skeleton containing six-membered aromatic rings
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    • C07C235/34—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to acyclic carbon atoms and singly-bound oxygen atoms bound to the same carbon skeleton the carbon skeleton containing six-membered aromatic rings having the nitrogen atoms of the carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
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    • C07C271/10—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms
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    • C07D209/04—Indoles; Hydrogenated indoles
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    • C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
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    • C07D311/04—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
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    • C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
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    • C07C2602/04—One of the condensed rings being a six-membered aromatic ring
    • C07C2602/10—One of the condensed rings being a six-membered aromatic ring the other ring being six-membered, e.g. tetraline
SI200030120T 1999-03-25 2000-03-24 Novi substituirani dimerni derivati, postopek za njihovo pripravo in farmacevtski pripravki, ki jih vsebujejo SI1038863T1 (sl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9903717A FR2791344B1 (fr) 1999-03-25 1999-03-25 Nouveaux derives dimeriques substitues, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
EP00400813A EP1038863B1 (fr) 1999-03-25 2000-03-24 Nouveaux dérivés dimériques substitués, leur procédé de préparation et les compositions pharmaceutiques qui les contiennent

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SI1038863T1 true SI1038863T1 (sl) 2003-10-31

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KR (1) KR100450314B1 (sl)
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AU (1) AU761605B2 (sl)
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FR (1) FR2791344B1 (sl)
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HU (1) HUP0001249A3 (sl)
NO (1) NO20001541L (sl)
NZ (1) NZ503587A (sl)
PL (1) PL339184A1 (sl)
PT (1) PT1038863E (sl)
SI (1) SI1038863T1 (sl)
ZA (1) ZA200001502B (sl)

Families Citing this family (5)

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Publication number Priority date Publication date Assignee Title
US6653346B1 (en) * 2002-02-07 2003-11-25 Galileo Pharmaceuticals, Inc. Cytoprotective benzofuran derivatives
US7078541B2 (en) * 2002-02-07 2006-07-18 Galileo Pharmaceuticals, Inc. Benzofuran derivatives
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EP1038863A3 (fr) 2000-11-02
KR20010006873A (ko) 2001-01-26
BR0001419A (pt) 2000-09-26
EP1038863A2 (fr) 2000-09-27
AU2257700A (en) 2000-10-05
JP3688549B2 (ja) 2005-08-31
EP1038863B1 (fr) 2003-06-04
HU0001249D0 (en) 2000-06-28
US6635650B2 (en) 2003-10-21
US20020035114A1 (en) 2002-03-21
HK1032042A1 (en) 2001-07-06
AU761605B2 (en) 2003-06-05
NO20001541L (no) 2000-09-26
ES2200794T3 (es) 2004-03-16
NZ503587A (en) 2001-05-25
KR100450314B1 (ko) 2004-09-30
FR2791344B1 (fr) 2002-02-15
EA200000261A3 (ru) 2000-12-25
US6319930B1 (en) 2001-11-20
EA003300B1 (ru) 2003-04-24
NO20001541D0 (no) 2000-03-24
DE60003103D1 (de) 2003-07-10
EA200000261A2 (ru) 2000-10-30
CA2301990A1 (fr) 2000-09-25
PL339184A1 (en) 2000-10-09
DE60003103T2 (de) 2004-05-19
CA2301990C (fr) 2004-01-06
JP2000319242A (ja) 2000-11-21
HUP0001249A3 (en) 2003-05-28
FR2791344A1 (fr) 2000-09-29
PT1038863E (pt) 2003-09-30
CN1273967A (zh) 2000-11-22
DK1038863T3 (da) 2003-09-22
ATE242201T1 (de) 2003-06-15
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HUP0001249A2 (hu) 2000-10-28

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